LV10269B - Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use - Google Patents

Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use Download PDF

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Publication number
LV10269B
LV10269B LVP-93-820A LV930820A LV10269B LV 10269 B LV10269 B LV 10269B LV 930820 A LV930820 A LV 930820A LV 10269 B LV10269 B LV 10269B
Authority
LV
Latvia
Prior art keywords
methyl
compound
pyridinyl
benzimidazole
preparation
Prior art date
Application number
LVP-93-820A
Other languages
English (en)
Latvian (lv)
Other versions
LV10269A (lv
Inventor
Brandstrim Arne Elof
Lindberg Per Lennart
Sunden Gunnel Elisabeth
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9002206A external-priority patent/SE9002206D0/xx
Priority claimed from SE9002207A external-priority patent/SE9002207D0/xx
Application filed by Astra Ab filed Critical Astra Ab
Publication of LV10269A publication Critical patent/LV10269A/xx
Publication of LV10269B publication Critical patent/LV10269B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
LVP-93-820A 1990-06-20 1993-06-30 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use LV10269B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9002206A SE9002206D0 (sv) 1990-06-20 1990-06-20 New compounds
SE9002207A SE9002207D0 (sv) 1990-06-20 1990-06-20 New compounds i
PCT/SE1991/000416 WO1991019712A1 (en) 1990-06-20 1991-06-11 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use

Publications (2)

Publication Number Publication Date
LV10269A LV10269A (lv) 1994-10-20
LV10269B true LV10269B (en) 1995-10-20

Family

ID=26660803

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-93-820A LV10269B (en) 1990-06-20 1993-06-30 Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use

Country Status (29)

Country Link
US (1) US5430042A (es)
EP (1) EP0593463B1 (es)
JP (1) JP3049367B2 (es)
CN (1) CN1058213A (es)
AP (1) AP253A (es)
AT (1) ATE184602T1 (es)
AU (1) AU649456B2 (es)
BG (1) BG97198A (es)
CA (1) CA2083606C (es)
CZ (1) CZ279434B6 (es)
DE (1) DE69131627T2 (es)
EG (1) EG19752A (es)
ES (1) ES2140391T3 (es)
FI (1) FI925767A0 (es)
HU (1) HUT62882A (es)
IE (1) IE912026A1 (es)
IL (1) IL98472A (es)
IS (1) IS3720A7 (es)
LV (1) LV10269B (es)
MA (1) MA22198A1 (es)
NO (1) NO924650D0 (es)
NZ (1) NZ238545A (es)
OA (1) OA09683A (es)
PL (2) PL165898B1 (es)
PT (1) PT98036A (es)
RO (1) RO110497B1 (es)
TN (1) TNSN91050A1 (es)
WO (1) WO1991019712A1 (es)
YU (1) YU104091A (es)

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US5817338A (en) * 1994-07-08 1998-10-06 Astra Aktiebolag Multiple unit tableted dosage form of omeprazole
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US6645988B2 (en) 1996-01-04 2003-11-11 Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US6699885B2 (en) * 1996-01-04 2004-03-02 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and methods of using same
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TWI367759B (en) * 2003-02-20 2012-07-11 Santarus Inc A novel formulation, omeprazole antacid complex-immediate release, for rapid and sustained suppression of gastric acid
CA2529984C (en) * 2003-06-26 2012-09-25 Isa Odidi Oral multi-functional pharmaceutical capsule preparations of proton pump inhibitors
US8993599B2 (en) * 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
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JP4919801B2 (ja) 2003-09-26 2012-04-18 アルザ・コーポレーシヨン 高い薬剤配合量を提供する薬剤コーティング及びそれを提供する方法
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BRPI0507784A (pt) * 2004-02-18 2007-07-17 Allergan Inc métodos e composições para a administração de pró-fármacos de inibidores da bomba de prótons
BRPI0507837A (pt) * 2004-02-18 2007-07-10 Allergan Inc métodos e composições para a administração intravenosa de compostos relacionados a inibidores de bomba de prótons
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US8815916B2 (en) * 2004-05-25 2014-08-26 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8906940B2 (en) * 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
US8394409B2 (en) 2004-07-01 2013-03-12 Intellipharmaceutics Corp. Controlled extended drug release technology
JP3921497B2 (ja) * 2004-08-06 2007-05-30 エーザイ・アール・アンド・ディー・マネジメント株式会社 ベンズイミダゾール誘導体とアミンとの塩およびその製造方法
US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
US8541026B2 (en) 2004-09-24 2013-09-24 Abbvie Inc. Sustained release formulations of opioid and nonopioid analgesics
US20070015782A1 (en) 2005-04-15 2007-01-18 Eisai Co., Ltd. Benzimidazole compound
US9040564B2 (en) 2005-04-28 2015-05-26 Eisai R&D Management Co., Ltd. Stabilized composition
US7981908B2 (en) 2005-05-11 2011-07-19 Vecta, Ltd. Compositions and methods for inhibiting gastric acid secretion
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JP5457830B2 (ja) 2006-04-03 2014-04-02 オディディ，イサ オルガノゾル被膜を含む制御放出送達デバイス
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US20090092658A1 (en) * 2007-10-05 2009-04-09 Santarus, Inc. Novel formulations of proton pump inhibitors and methods of using these formulations
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JP2009196894A (ja) * 2006-10-13 2009-09-03 Eisai R & D Management Co Ltd スルフィニルベンズイミダゾール化合物またはその塩の製造方法
US20080103169A1 (en) 2006-10-27 2008-05-01 The Curators Of The University Of Missouri Compositions comprising acid labile proton pump inhibiting agents, at least one other pharmaceutically active agent and methods of using same
US20080194307A1 (en) * 2007-02-13 2008-08-14 Jeff Sanger Sports-based game of chance
JP2011512416A (ja) 2008-02-20 2011-04-21 ザ・キュレイターズ・オブ・ザ・ユニバーシティー・オブ・ミズーリ オメプラゾール及びランソプラゾールの組合せと緩衝剤を含んでなる組成物とそれを使用する方法
CN102209529A (zh) 2008-09-09 2011-10-05 阿斯利康(瑞典)有限公司 将药物组合物递送至有需要的患者的方法
EP2445499A4 (en) 2009-06-25 2013-02-27 Astrazeneca Ab METHOD FOR TREATING A PATIENT WITH RISK OF DEVELOPING A NSAID-ASSOCIATED SPURGE
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US4359465A (en) * 1980-07-28 1982-11-16 The Upjohn Company Methods for treating gastrointestinal inflammation
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Also Published As

Publication number Publication date
CA2083606C (en) 2001-08-21
CA2083606A1 (en) 1991-12-21
OA09683A (en) 1993-05-15
AP253A (en) 1993-05-03
IE912026A1 (en) 1992-01-01
JP3049367B2 (ja) 2000-06-05
RO110497B1 (ro) 1996-01-30
EP0593463A1 (en) 1994-04-27
ES2140391T3 (es) 2000-03-01
PL165898B1 (pl) 1995-02-28
NO924650L (no) 1992-12-02
IS3720A7 (is) 1991-12-21
JPH05507714A (ja) 1993-11-04
AP9100286A0 (en) 1991-07-31
PL297295A1 (es) 1992-07-13
WO1991019712A1 (en) 1991-12-26
PT98036A (pt) 1992-03-31
MA22198A1 (fr) 1992-04-01
CS189391A3 (en) 1992-06-17
LV10269A (lv) 1994-10-20
HU9204034D0 (en) 1993-03-29
NZ238545A (en) 1993-08-26
FI925767A (fi) 1992-12-18
US5430042A (en) 1995-07-04
TNSN91050A1 (fr) 1992-10-25
HUT62882A (en) 1993-06-28
PL166209B1 (pl) 1995-04-28
ATE184602T1 (de) 1999-10-15
PL297294A1 (es) 1992-07-13
AU649456B2 (en) 1994-05-26
YU104091A (sh) 1994-01-20
AU8061791A (en) 1992-01-07
EG19752A (en) 1996-01-31
IL98472A0 (en) 1992-07-15
BG97198A (bg) 1993-12-24
NO924650D0 (no) 1992-12-02
FI925767A0 (fi) 1992-12-18
CZ279434B6 (cs) 1995-04-12
EP0593463B1 (en) 1999-09-15
IL98472A (en) 1995-08-31
CN1058213A (zh) 1992-01-29
DE69131627D1 (de) 1999-10-21
DE69131627T2 (de) 2000-04-27

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