LU88714I2 - Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique - Google Patents

Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique

Info

Publication number
LU88714I2
LU88714I2 LU88714C LU88714C LU88714I2 LU 88714 I2 LU88714 I2 LU 88714I2 LU 88714 C LU88714 C LU 88714C LU 88714 C LU88714 C LU 88714C LU 88714 I2 LU88714 I2 LU 88714I2
Authority
LU
Luxembourg
Prior art keywords
amino
hydroxybutane
diphosphonic
alkali metal
organic base
Prior art date
Application number
LU88714C
Other languages
English (en)
French (fr)
Original Assignee
Gentili Ist Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11171970&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU88714(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gentili Ist Spa filed Critical Gentili Ist Spa
Publication of LU88714I2 publication Critical patent/LU88714I2/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839Polyphosphonic acids
    • C07F9/3873Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839Polyphosphonic acids
    • C07F9/3856Polyphosphonic acids containing halogen or nitro(so) substituents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LU88714C 1982-04-15 1983-04-13 Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique LU88714I2 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8220781A IT1201087B (it) 1982-04-15 1982-04-15 Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche

Publications (1)

Publication Number Publication Date
LU88714I2 true LU88714I2 (fr) 1996-08-23

Family

ID=11171970

Family Applications (2)

Application Number Title Priority Date Filing Date
LU84746A LU84746A1 (fr) 1982-04-15 1983-04-13 Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique
LU88714C LU88714I2 (fr) 1982-04-15 1983-04-13 Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique

Family Applications Before (1)

Application Number Title Priority Date Filing Date
LU84746A LU84746A1 (fr) 1982-04-15 1983-04-13 Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique

Country Status (12)

Country Link
US (1) US4621077A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS58189193A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE896453A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH661437A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2525223B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB2118042B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HK (1) HK79390A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1201087B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
LU (2) LU84746A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX9203428A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (5) NL192562C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE463239B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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CN106687118A (zh) 2014-07-02 2017-05-17 配体药物公司 前药化合物及其用途
US11970482B2 (en) 2018-01-09 2024-04-30 Ligand Pharmaceuticals Inc. Acetal compounds and therapeutic uses thereof

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SE8302130D0 (sv) 1983-04-15
FR2525223A1 (fr) 1983-10-21
NL192562B (nl) 1997-06-02
BE896453A (fr) 1983-08-01
MX9203428A (es) 1992-07-01
LU84746A1 (fr) 1983-11-17
NL980004I1 (nl) 1998-04-01
NL970038I2 (nl) 2000-11-01
NL192562C (nl) 1997-10-03
IT1201087B (it) 1989-01-27
NL980010I1 (nl) 1998-05-06
JPH0213645B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1990-04-04
GB2118042B (en) 1986-01-15
JPS58189193A (ja) 1983-11-04
NL980005I1 (nl) 1998-04-01
SE463239B (sv) 1990-10-29
GB2118042A (en) 1983-10-26
NL8301324A (nl) 1983-11-01
NL970038I1 (nl) 1998-01-05
US4621077A (en) 1986-11-04
IT8220781A0 (it) 1982-04-15
HK79390A (en) 1990-10-12
SE8302130L (sv) 1983-10-16
CH661437A5 (it) 1987-07-31
FR2525223B1 (fr) 1986-04-25
GB8308791D0 (en) 1983-05-11

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