LU82468A1 - Derives de l'acide penicillanique utiles comme medicaments,compositions therapeutiques les contenant et procedes de leur preparation - Google Patents

Derives de l'acide penicillanique utiles comme medicaments,compositions therapeutiques les contenant et procedes de leur preparation Download PDF

Info

Publication number
LU82468A1
LU82468A1 LU82468A LU82468A LU82468A1 LU 82468 A1 LU82468 A1 LU 82468A1 LU 82468 A LU82468 A LU 82468A LU 82468 A LU82468 A LU 82468A LU 82468 A1 LU82468 A1 LU 82468A1
Authority
LU
Luxembourg
Prior art keywords
salt
acid
penicillanate
bromo
iodo
Prior art date
Application number
LU82468A
Other languages
English (en)
French (fr)
Inventor
W Daehne
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of LU82468A1 publication Critical patent/LU82468A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LU82468A 1979-05-21 1980-05-20 Derives de l'acide penicillanique utiles comme medicaments,compositions therapeutiques les contenant et procedes de leur preparation LU82468A1 (fr)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
GB7917665 1979-05-21
GB7917665 1979-05-21
GB7930819 1979-09-05
GB7930819 1979-09-05
GB7941252 1979-11-29
GB7941252 1979-11-29
GB8006681 1980-02-27
GB8006681 1980-02-27

Publications (1)

Publication Number Publication Date
LU82468A1 true LU82468A1 (fr) 1980-12-16

Family

ID=27449123

Family Applications (1)

Application Number Title Priority Date Filing Date
LU82468A LU82468A1 (fr) 1979-05-21 1980-05-20 Derives de l'acide penicillanique utiles comme medicaments,compositions therapeutiques les contenant et procedes de leur preparation

Country Status (19)

Country Link
US (3) US4446144A (de)
JP (1) JPS55154977A (de)
AU (3) AU534754B2 (de)
BE (1) BE883390A (de)
CA (1) CA1265787A (de)
DE (3) DE3051038C2 (de)
DK (2) DK158669C (de)
FI (1) FI801618A (de)
FR (2) FR2457294A1 (de)
GR (1) GR68372B (de)
IE (2) IE49770B1 (de)
IL (1) IL59948A0 (de)
IT (1) IT1133091B (de)
LU (1) LU82468A1 (de)
NL (1) NL8002911A (de)
NZ (1) NZ193597A (de)
PH (2) PH17959A (de)
PT (1) PT71273A (de)
SE (3) SE452465B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51846B1 (en) * 1980-11-17 1987-04-15 Leo Pharm Prod Ltd Pharmaceutical preparation for veterinary use and an appliance containing it
US4521533A (en) * 1984-07-12 1985-06-04 Pfizer Inc. Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics
GB8522156D0 (en) * 1985-09-06 1985-10-09 Leo Pharm Prod Ltd Producing chemical compounds
US5589354A (en) * 1994-12-20 1996-12-31 Biopure Corporation Halogenation of cephalexin with haloperoxidase from Rathayibacter biopuresis
US5695951A (en) * 1994-12-20 1997-12-09 Biopure Corporation Chlorination of cephalexin with chloroperoxidase from Rathayibacter biopuresis
DK0971690T4 (en) 1996-12-18 2015-07-13 Bimeda Res & Dev Ltd Anti-infective intramammary veterinary composition.
US20020035107A1 (en) * 2000-06-20 2002-03-21 Stefan Henke Highly concentrated stable meloxicam solutions
CA2501395C (en) * 2002-10-25 2011-05-24 Akzo Nobel Nv Prolonged release pharmaceutical composition
EP1568369A1 (de) 2004-02-23 2005-08-31 Boehringer Ingelheim Vetmedica Gmbh Verwendung von Meloxicam zur Behandlung von Atemwegserkrankungen bei Schweinen
DE102004025324A1 (de) * 2004-05-19 2005-12-08 Boehringer Ingelheim Vetmedica Gmbh Flüssige Zubereitung für die Veterinärmedizin, Verfahren zu deren Herstellung und deren Verwendung
WO2014014364A1 (en) * 2012-07-17 2014-01-23 Bayer New Zealand Limited Injectable antibiotic formulations and their methods of use
MY172561A (en) * 2012-07-17 2019-12-03 Bayer New Zealand Ltd Injectable antibiotic formulations and their methods of use
BR112015014963B1 (pt) * 2012-12-20 2022-04-12 Alleva Animal Health Limited Formulação de suspensão injetável veterinária
EP4265241A1 (de) * 2022-04-20 2023-10-25 Bilim Ilac Sanayii Ve Ticaret A.S. Tablettenformulierungen zur behandlung von harnwegsinfektionen und verfahren zur herstellung solcher formulierungen

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1089385B (de) 1954-06-21 1960-09-22 Biochemie Gmbh Verfahren zur Herstellung von in Wasser schwer loeslichen, besonders fuer die Oraltherapie geeigneten Salzen des Penicillins mit organischen Basen
DE1031795B (de) 1955-09-29 1958-06-12 Chimiotherapie Lab Franc Verfahren zur Herstellung eines Salzes aus Penicillin und einer Piperazinbase
US3206469A (en) * 1961-08-15 1965-09-14 Lepetit Spa 6-halopenicillanic acid
GB1297555A (de) * 1970-09-22 1972-11-22
GB1377817A (en) * 1971-06-09 1974-12-18 Beecham Group Ltd Penicillins and cephalosporins
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IN149747B (de) * 1977-06-07 1982-04-03 Pfizer
US4180506A (en) * 1978-01-18 1979-12-25 Rex Pratt 6β-Bromo penicillanic acid
CA1158639A (en) 1978-12-11 1983-12-13 Eric M. Gordon 6-bromopenicillanic acid sulfone
US4203992A (en) * 1978-12-11 1980-05-20 E. R. Squibb & Sons, Inc. β-Bromopenicillanic acid sulfone
IL59081A0 (en) * 1979-01-10 1980-05-30 Schering Corp 2-penem compounds and a method for preparing them
DE3068390D1 (en) * 1979-01-10 1984-08-09 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
US4518530A (en) * 1979-03-05 1985-05-21 Pfizer Inc. 6-β-Substituted penicillanic acids as β-lactamase inhibitors
US4397783A (en) * 1979-03-05 1983-08-09 Pfizer Inc. Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
US4432970A (en) * 1979-11-23 1984-02-21 Pfizer Inc. 6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors

Also Published As

Publication number Publication date
SE8406201D0 (sv) 1984-12-06
AU541323B2 (en) 1985-01-03
BE883390A (fr) 1980-11-20
NL8002911A (nl) 1980-11-25
DK562589D0 (da) 1989-11-10
SE462097B (sv) 1990-05-07
DE3051037C2 (de) 1989-03-30
FR2499575B1 (de) 1985-03-01
AU534754B2 (en) 1984-02-16
DK218580A (da) 1980-11-22
IE49770B1 (en) 1985-12-11
IE800868L (en) 1980-11-21
AU1848683A (en) 1983-12-22
DE3019244C2 (de) 1989-04-06
US4446144A (en) 1984-05-01
PT71273A (en) 1980-06-01
AU541322B2 (en) 1985-01-03
IE49768B1 (en) 1985-12-11
IT8067790A0 (it) 1980-05-20
IL59948A0 (en) 1980-06-30
SE8406202L (sv) 1984-12-06
DK158669C (da) 1991-01-21
DE3051038C2 (de) 1989-04-13
SE8406201L (sv) 1984-12-06
DK158670C (da) 1991-01-07
CA1265787A (en) 1990-02-13
IT1133091B (it) 1986-07-09
FR2457294B1 (de) 1984-01-13
JPH0140837B2 (de) 1989-08-31
SE462096B (sv) 1990-05-07
US4672114A (en) 1987-06-09
DE3051038A1 (de) 1986-03-20
DK158670B (da) 1990-07-02
DE3019244A1 (de) 1980-12-04
DK158669B (da) 1990-07-02
FI801618A (fi) 1980-11-22
AU1848783A (en) 1983-12-22
FR2499575A1 (fr) 1982-08-13
SE452465B (sv) 1987-11-30
PH17959A (en) 1985-02-20
SE8003722L (sv) 1980-11-22
FR2457294A1 (fr) 1980-12-19
IE842559L (en) 1980-11-21
DK562589A (da) 1989-11-10
NZ193597A (en) 1985-04-30
JPS55154977A (en) 1980-12-02
AU5858480A (en) 1980-11-27
SE8406202D0 (sv) 1984-12-06
GR68372B (de) 1981-12-28
PH19005A (en) 1985-12-03
US4594246A (en) 1986-06-10

Similar Documents

Publication Publication Date Title
Baltzer et al. Mutual pro-drugs of β-lactam antibiotics and β-lactamase inhibitors
LU82468A1 (fr) Derives de l'acide penicillanique utiles comme medicaments,compositions therapeutiques les contenant et procedes de leur preparation
LU79774A1 (fr) Procede de preparation de 1,1-dioxydes de l'acide penicillanique et de ses esters utiles comme inhibiteurs de la b-lactamase
LU82164A1 (fr) -lactames derives de l acide penicillanique, leur preparation et leurs utilisations therapeutiques
FR2479229A1 (fr) Nouveaux derives des cephalosporines, leur procede de preparation et les medicaments utilisables comme antibiotiques qui contiennent lesdits derives
JPH08505645A (ja) 結晶性ペニシリン誘導体並びにその製造及び使用
JPS6224435B2 (de)
EP0080944B1 (de) Cephalosporinderivate substituiert in Position 3 von einer thiomethylheterocyclischen Gruppe, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Verbindungen
BE875054A (fr) Composes analogues aux cephalosporines
FR2491474A1 (fr) Napsylate de (d-a-amino a-phenylacetamido)-6 penicillanate de dioxo-1,1 penicillanoyloxymethyle cristallin et ses formes hydratees, leurs procedes de preparation et des medicaments antimicrobiens les contenant comme produits actifs
LU82163A1 (fr) Nouveaux derives d'acide penicillanique utile notamment comme antibiotiques et leurs procedes de preparation
US4511512A (en) Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
FR2520362A1 (fr) Nouveaux composes de type b-lactame, y compris leurs sels formes avec des acides ou des bases acceptables en pharmacie, procedes pour produire ces composes, medicaments les contenant et leur utilisation pour combattre les maladies infectieuses
GB2051046A (en) Penicillanic acid derivatives
LU84739A1 (fr) Nouveaux antibiotiques de type carbapenem
BE862211A (fr) Agents antibacteriens
BE821243A (fr) Derives de la penicilline
LU86105A1 (fr) Carbapenemes antibiotiques
LU81795A1 (fr) Nouvelle penicilline semi-synthetique,son procede de production et composition pharmaceutique la contenant
CA1207752A (en) PROCESS FOR PREPARING DERIVATIVES OF .beta.-LACTAM AND DERIVATIVES SO PRODUCED
FR2485540A1 (fr) Nouveaux derives antibiotiques des cephalosporines, leur procede de preparation et les medicaments en contenant
FR2539130A1 (fr) Esters de type penem, procede pour les preparer, medicament les contenant
JPH05194528A (ja) 新規な１−オキサペネム−３−カルボン酸類及びそのβ−ラクタマーゼ阻害薬としての用途
GB2125038A (en) Amine salts of 6 beta -halopenicillanic acids
FR2498189A1 (fr) Nouveaux derives de l'acide cephalosporanique, leur preparation et leur application comme medicaments