KR900005131B1 - N-포르밀 및 n-하이드록시메틸-3-펜옥시-1-아제티딘카복스아미드, 이의 제조방법 및 이를 함유하는 약제학적 조성물 - Google Patents

N-포르밀 및 n-하이드록시메틸-3-펜옥시-1-아제티딘카복스아미드, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Download PDF

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Publication number
KR900005131B1
KR900005131B1 KR1019830004080A KR830004080A KR900005131B1 KR 900005131 B1 KR900005131 B1 KR 900005131B1 KR 1019830004080 A KR1019830004080 A KR 1019830004080A KR 830004080 A KR830004080 A KR 830004080A KR 900005131 B1 KR900005131 B1 KR 900005131B1
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KR
South Korea
Prior art keywords
phenoxy
azetidinecarboxamide
trifluoromethyl
compound
hydroxymethyl
Prior art date
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Expired
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KR1019830004080A
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English (en)
Korean (ko)
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KR840006203A (ko
Inventor
죠셉 라이트 죠지
첸 텡 리나
Original Assignee
에이.에치.로빈스 캄파니, 인코포레이티드
존 씨.고돈
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Publication date
Application filed by 에이.에치.로빈스 캄파니, 인코포레이티드, 존 씨.고돈 filed Critical 에이.에치.로빈스 캄파니, 인코포레이티드
Publication of KR840006203A publication Critical patent/KR840006203A/ko
Application granted granted Critical
Publication of KR900005131B1 publication Critical patent/KR900005131B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019830004080A 1982-09-02 1983-08-31 N-포르밀 및 n-하이드록시메틸-3-펜옥시-1-아제티딘카복스아미드, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Expired KR900005131B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/414,101 US4505907A (en) 1982-09-02 1982-09-02 N-Formyl and N-hydroxymethyl-3-phenoxy-1-azetidinecarboxamides
US414101 2003-04-16

Publications (2)

Publication Number Publication Date
KR840006203A KR840006203A (ko) 1984-11-22
KR900005131B1 true KR900005131B1 (ko) 1990-07-20

Family

ID=23639965

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019830004080A Expired KR900005131B1 (ko) 1982-09-02 1983-08-31 N-포르밀 및 n-하이드록시메틸-3-펜옥시-1-아제티딘카복스아미드, 이의 제조방법 및 이를 함유하는 약제학적 조성물

Country Status (25)

Country Link
US (1) US4505907A (enExample)
EP (1) EP0102740B1 (enExample)
JP (1) JPS601161A (enExample)
KR (1) KR900005131B1 (enExample)
AU (1) AU553472B2 (enExample)
CA (1) CA1185983A (enExample)
CS (1) CS240974B2 (enExample)
DE (1) DE3367385D1 (enExample)
DK (1) DK166297C (enExample)
EG (1) EG16473A (enExample)
ES (2) ES8504697A1 (enExample)
FI (1) FI77226C (enExample)
GR (1) GR79337B (enExample)
HK (1) HK47587A (enExample)
HU (1) HU189740B (enExample)
IE (1) IE55770B1 (enExample)
IL (1) IL68743A0 (enExample)
IN (1) IN161222B (enExample)
NO (1) NO157977C (enExample)
NZ (1) NZ205448A (enExample)
PH (1) PH20572A (enExample)
PL (2) PL145986B1 (enExample)
PT (1) PT77281B (enExample)
YU (1) YU44747B (enExample)
ZA (1) ZA834410B (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4571393A (en) * 1982-08-19 1986-02-18 A. H. Robins Company, Incorporated 3-Phenoxy-1-azetidinecarboxamides
US4594189A (en) * 1983-07-06 1986-06-10 A. H. Robins Company, Inc. Process for preparing 3-phenoxy-1-azetidines and carboxamide derivatives
IN162808B (enExample) * 1985-02-28 1988-07-09 Robins Co Inc A H
ZA861210B (en) * 1985-02-28 1987-10-28 Robins Co Inc A H 3-aryloxyazetidinecarboxamides as anticonvulsants and antiepileptics
US4956359A (en) * 1985-02-28 1990-09-11 A. H. Robins Company, Inc. 3-aryloxy and 3-arylthioazetidinecarboxamides as anticonvulsants and antiepileptics
FI87559C (fi) * 1985-02-28 1993-01-25 Robins Co Inc A H Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider
US5068231A (en) * 1985-02-28 1991-11-26 A. H. Robins Company Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US5130309A (en) * 1991-04-12 1992-07-14 A. H. Robins Company, Incorporated Aryloxy and aryloxyalklazetidines as antiarrhythmic and anticonvulsant agents
JP3178922B2 (ja) * 1992-12-03 2001-06-25 小松ゼノア株式会社 エンジンの吸気装置
GB9801501D0 (en) * 1998-01-23 1998-03-18 Cerebrus Ltd Chemical compounds - II
EP1049670B1 (en) 1998-01-23 2002-07-17 Vernalis Research Limited Azetidinecarboxamide derivatives for treating cns disorders
ATE250027T1 (de) 1998-01-23 2003-10-15 Vernalis Res Ltd Azetidincarboxamidderivate zur behandlung von zns-erkrankungen
GB9917385D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-I
GB9917386D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-II
WO2009051244A1 (ja) * 2007-10-18 2009-04-23 Takeda Pharmaceutical Company Limited 複素環化合物
US10365007B2 (en) 2014-09-30 2019-07-30 Fujitsu General Limited Ceiling-embedded air conditioner
US10288302B2 (en) 2015-03-31 2019-05-14 Fujitsu General Limited Ceiling-embedded air conditioner with airflow guide vane
JP6504349B2 (ja) 2015-03-31 2019-04-24 株式会社富士通ゼネラル 天井埋込型空気調和機
JP6516095B2 (ja) 2015-04-27 2019-05-22 株式会社富士通ゼネラル 天井埋込型空気調和機

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB872447A (en) * 1958-12-23 1961-07-12 Lepetit Spa 1-carbamyl-3-substituted azetidines
DE2053333A1 (de) * 1970-10-30 1972-05-04 Farbenfabriken Bayer Ag, 5090 Lever Kusen Herbizide Mittel
US4031221A (en) * 1974-06-17 1977-06-21 American Hoechst Corporation Method of treating pain and hypertension
US4379151A (en) * 1978-03-14 1983-04-05 A. H. Robins Company, Inc. 3-Phenoxyazetidines for anorexigenic activity
US4226861A (en) * 1978-04-18 1980-10-07 A. H. Robins Company, Inc. N-Lower-alkyl 3-phenoxy-1-azetidinecarboxamides

Also Published As

Publication number Publication date
EG16473A (en) 1990-12-30
FI833126L (fi) 1984-03-03
EP0102740A1 (en) 1984-03-14
GR79337B (enExample) 1984-10-22
FI77226B (fi) 1988-10-31
DK398783A (da) 1984-03-03
NZ205448A (en) 1985-08-30
ES537668A0 (es) 1985-09-16
YU44747B (en) 1991-02-28
PT77281B (en) 1986-02-04
IE55770B1 (en) 1991-01-16
IL68743A0 (en) 1983-09-30
PH20572A (en) 1987-02-18
ES8600234A1 (es) 1985-09-16
AU553472B2 (en) 1986-07-17
FI833126A0 (fi) 1983-09-01
KR840006203A (ko) 1984-11-22
CA1185983A (en) 1985-04-23
FI77226C (fi) 1989-02-10
PT77281A (en) 1983-10-01
DK166297B (da) 1993-03-29
PL145986B1 (en) 1988-12-31
CS614183A2 (en) 1985-06-13
PL243555A1 (en) 1984-08-27
US4505907A (en) 1985-03-19
AU1459883A (en) 1984-03-08
EP0102740B1 (en) 1986-11-05
HK47587A (en) 1987-06-26
NO157977C (no) 1988-06-22
IN161222B (enExample) 1987-10-24
JPS601161A (ja) 1985-01-07
DK398783D0 (da) 1983-09-01
IE831652L (en) 1984-03-02
ZA834410B (en) 1984-03-28
ES523194A0 (es) 1985-04-16
PL142643B1 (en) 1987-11-30
DE3367385D1 (en) 1986-12-11
ES8504697A1 (es) 1985-04-16
HU189740B (en) 1986-07-28
NO833135L (no) 1984-03-05
NO157977B (no) 1988-03-14
DK166297C (da) 1993-08-30
JPH0452264B2 (enExample) 1992-08-21
CS240974B2 (en) 1986-03-13
YU170483A (en) 1986-04-30

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