KR20200094142A - 혈장 칼리크레인 저해제 및 그 염의 고체 형태 - Google Patents
혈장 칼리크레인 저해제 및 그 염의 고체 형태 Download PDFInfo
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- KR20200094142A KR20200094142A KR1020207015220A KR20207015220A KR20200094142A KR 20200094142 A KR20200094142 A KR 20200094142A KR 1020207015220 A KR1020207015220 A KR 1020207015220A KR 20207015220 A KR20207015220 A KR 20207015220A KR 20200094142 A KR20200094142 A KR 20200094142A
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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| MX2020005168A (es) | 2017-11-29 | 2020-08-20 | Kalvista Pharmaceuticals Ltd | Formas de dosificacion que contienen un inhibidor calicreina de plasma. |
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| GB201609601D0 (en) | 2016-06-01 | 2016-07-13 | Nucana Biomed Ltd | Phosphoramidate compounds |
| GB201609602D0 (en) | 2016-06-01 | 2016-07-13 | Nucuna Biomed Ltd | Chemical compounds |
| GB201609607D0 (en) | 2016-06-01 | 2016-07-13 | Kalvista Pharmaceuticals Ltd | Polymorphs of N-(3-Fluoro-4-methoxypyridin-2-yl)methyl)-3-(methoxymethyl)-1-({4-((2-oxopy ridin-1-yl)methyl)phenyl}methyl)pyrazole-4-carboxamide and salts |
| WO2018011628A1 (en) | 2016-07-11 | 2018-01-18 | Lifesci Pharmaceuticals, Inc. | Therapeutic inhibitory compounds |
| GB201713660D0 (en) | 2017-08-25 | 2017-10-11 | Kalvista Pharmaceuticals Ltd | Pharmaceutical compositions |
| GB201721515D0 (en) | 2017-12-21 | 2018-02-07 | Kalvista Pharmaceuticals Ltd | Dosage forms comprising a plasma kallikrein inhibtor |
| TW201925188A (zh) | 2017-11-29 | 2019-07-01 | 英商卡爾維斯塔製藥有限公司 | 酶抑制劑 |
| GB201719882D0 (en) | 2017-11-29 | 2018-01-10 | Kalvista Pharmaceuticals Ltd | Solid forms of a plasma kallikrein inhibitor and salts thereof |
| GB201719881D0 (en) | 2017-11-29 | 2018-01-10 | Kalvista Pharmaceuticals Ltd | Solid forms of plasma kallikrein inhibitor and salts thereof |
| GB201910125D0 (en) | 2019-07-15 | 2019-08-28 | Kalvista Pharmaceuticals Ltd | Treatments of angioedema |
| GB201910116D0 (en) | 2019-07-15 | 2019-08-28 | Kalvista Pharmaceuticals Ltd | Treatments of hereditary angioedema |
| EP4010333A1 (en) | 2019-08-09 | 2022-06-15 | Kalvista Pharmaceuticals Limited | Plasma kallikrein inhibitors |
| WO2021032936A1 (en) | 2019-08-21 | 2021-02-25 | Kalvista Pharmaceuticals Limited | Enzyme inhibitors |
| WO2021032935A1 (en) | 2019-08-21 | 2021-02-25 | Kalvista Pharmaceuticals Limited | Enzyme inhibitors |
| BR112022001341A2 (pt) | 2019-08-21 | 2022-03-22 | Kalvista Pharmaceuticals Ltd | Inibidores de enzima |
| EP4017586A1 (en) | 2019-08-21 | 2022-06-29 | Kalvista Pharmaceuticals Limited | Enzyme inhibitors |
| GB201918994D0 (en) | 2019-12-20 | 2020-02-05 | Kalvista Pharmaceuticals Ltd | Treatments of diabetic macular edema and impaired visual acuity |
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2017
- 2017-11-29 GB GBGB1719881.3A patent/GB201719881D0/en not_active Ceased
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2018
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- 2018-11-29 RU RU2020121150A patent/RU2020121150A/ru unknown
- 2018-11-29 EP EP18815306.8A patent/EP3717469A1/en not_active Withdrawn
- 2018-11-29 CA CA3082304A patent/CA3082304A1/en active Pending
- 2018-11-29 MX MX2020005422A patent/MX2020005422A/es unknown
- 2018-11-29 WO PCT/GB2018/053466 patent/WO2019106377A1/en not_active Ceased
- 2018-11-29 CN CN201880077596.1A patent/CN111433197A/zh active Pending
- 2018-11-29 KR KR1020207015220A patent/KR20200094142A/ko not_active Withdrawn
- 2018-11-29 BR BR112020010064-1A patent/BR112020010064A2/pt not_active IP Right Cessation
- 2018-11-29 AU AU2018374541A patent/AU2018374541B2/en not_active Withdrawn - After Issue
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2020
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2023
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| US20230203012A1 (en) | 2023-06-29 |
| IL274555A (en) | 2020-06-30 |
| GB201719881D0 (en) | 2018-01-10 |
| JP2021504310A (ja) | 2021-02-15 |
| MX2020005422A (es) | 2020-08-27 |
| RU2020121150A (ru) | 2021-12-29 |
| US11584735B2 (en) | 2023-02-21 |
| CA3082304A1 (en) | 2019-06-06 |
| CN111433197A (zh) | 2020-07-17 |
| WO2019106377A1 (en) | 2019-06-06 |
| EP3717469A1 (en) | 2020-10-07 |
| AU2018374541A1 (en) | 2020-05-28 |
| BR112020010064A2 (pt) | 2020-11-03 |
| AU2018374541B2 (en) | 2022-12-22 |
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