KR20190070956A - Ssao/vap-1 억제제 및 sglt2 억제제를 포함하는 복합제제 및 이의 용도 - Google Patents
Ssao/vap-1 억제제 및 sglt2 억제제를 포함하는 복합제제 및 이의 용도 Download PDFInfo
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- KR20190070956A KR20190070956A KR1020197014347A KR20197014347A KR20190070956A KR 20190070956 A KR20190070956 A KR 20190070956A KR 1020197014347 A KR1020197014347 A KR 1020197014347A KR 20197014347 A KR20197014347 A KR 20197014347A KR 20190070956 A KR20190070956 A KR 20190070956A
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Landscapes
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Applications Claiming Priority (3)
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| EP16194572 | 2016-10-19 | ||
| PCT/EP2017/076300 WO2018073154A1 (en) | 2016-10-19 | 2017-10-16 | Combinations comprising an ssao/vap-1 inhibitor and a sglt2 inhibitor, uses thereof |
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| KR20190110740A (ko) | 2018-03-21 | 2019-10-01 | 주식회사유한양행 | 신규의 아릴 또는 헤테로아릴 트라이아졸론 유도체 또는 이의 염 및 이를 포함하는 약학 조성물 |
| SG11202103062UA (en) * | 2018-09-28 | 2021-04-29 | Acucela Inc | Inhibitors of vap-1 |
| MX2021003731A (es) | 2018-09-28 | 2021-08-05 | Acucela Inc | Inhibidores de vap-1. |
| JP7414230B2 (ja) * | 2018-11-09 | 2024-01-16 | 国立大学法人 琉球大学 | 抗血液悪性腫瘍薬 |
| CN121081472A (zh) | 2018-12-13 | 2025-12-09 | 拓臻股份有限公司 | 一种THRβ受体激动剂化合物及其制备方法和用途 |
| TWI835945B (zh) * | 2018-12-14 | 2024-03-21 | 南韓商柳韓洋行股份有限公司 | 3,3-二氟烯丙胺化物或其鹽及包含彼的醫藥組合物 |
| TW202039486A (zh) * | 2018-12-14 | 2020-11-01 | 南韓商柳韓洋行股份有限公司 | 三唑并吡啶-3-酮化物或其鹽及包含彼之醫藥組合物 |
| CN114375193B (zh) | 2019-09-12 | 2024-05-14 | 拓臻制药公司 | 甲状腺激素受体β激动剂化合物 |
| EP4051669A4 (en) | 2019-10-29 | 2023-12-13 | Eccogene (Shanghai) Co., Ltd. | SSAO INHIBITORS AND THEIR USE |
| CN115666577A (zh) * | 2020-03-25 | 2023-01-31 | 拓臻股份有限公司 | 呼吸道病症的治疗 |
| KR20230023642A (ko) * | 2020-05-13 | 2023-02-17 | 테른스 파마슈티칼스, 인크. | 간 장애의 조합 치료 |
| CN113893256A (zh) * | 2020-07-06 | 2022-01-07 | 诺未科技(北京)有限公司 | 化合物或其可药用盐、二聚体或三聚体在制备治疗癌症的药物中的应用 |
| AU2021332217A1 (en) | 2020-08-25 | 2023-05-11 | Eli Lilly And Company | Polymorphs of an ssao inhibitor |
| US20240148767A1 (en) * | 2021-03-04 | 2024-05-09 | The Governors Of The University Of Alberta | The use of empagliflozin for the treatment of ulcerative colitis and crohn's disease |
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| ES2567571T3 (es) | 2003-03-14 | 2016-04-25 | Astellas Pharma Inc. | Derivados de C-glucósido y sales de los mismos |
| EP2514756B1 (en) | 2003-08-01 | 2014-12-17 | Mitsubishi Tanabe Pharma Corporation | Novel compounds having inhibitory activity against sodium-dependant glucose transporter |
| PL1730131T3 (pl) | 2004-03-16 | 2012-10-31 | Boehringer Ingelheim Int | Glukopiranozylo-podstawione pochodne benzenu, środki lecznicze zawierające te związki, ich zastosowanie i sposób ich wytwarzania |
| TW200637839A (en) | 2005-01-07 | 2006-11-01 | Taisho Pharmaceutical Co Ltd | 1-thio-d-glucitol derivatives |
| TW200637869A (en) | 2005-01-28 | 2006-11-01 | Chugai Pharmaceutical Co Ltd | The spiroketal derivatives and the use as therapeutical agent for diabetes of the same |
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| ATE517099T1 (de) | 2006-02-15 | 2011-08-15 | Boehringer Ingelheim Int | Glucopyranosyl-substituierte benzonitril-derivate,pharmazeutische zusammensetzungen mit derartigen verbindungen, ihre verwendung und herstellungsverfahren dafür |
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2017
- 2017-10-16 US US16/341,460 patent/US20210212968A1/en not_active Abandoned
- 2017-10-16 EP EP17804068.9A patent/EP3528800A1/en not_active Withdrawn
- 2017-10-16 MX MX2019004549A patent/MX2019004549A/es unknown
- 2017-10-16 CA CA3041169A patent/CA3041169A1/en not_active Abandoned
- 2017-10-16 EA EA201990951A patent/EA201990951A1/ru unknown
- 2017-10-16 CN CN201780063937.5A patent/CN109843279A/zh active Pending
- 2017-10-16 JP JP2019520691A patent/JP2019531320A/ja active Pending
- 2017-10-16 WO PCT/EP2017/076300 patent/WO2018073154A1/en not_active Ceased
- 2017-10-16 KR KR1020197014347A patent/KR20190070956A/ko not_active Withdrawn
- 2017-10-16 BR BR112019005930A patent/BR112019005930A2/pt not_active IP Right Cessation
- 2017-10-16 AU AU2017344882A patent/AU2017344882A1/en not_active Abandoned
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2019
- 2019-04-08 CL CL2019000935A patent/CL2019000935A1/es unknown
- 2019-04-11 IL IL265989A patent/IL265989A/en unknown
- 2019-04-17 PH PH12019500845A patent/PH12019500845A1/en unknown
Also Published As
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|---|---|
| CA3041169A1 (en) | 2018-04-26 |
| CN109843279A (zh) | 2019-06-04 |
| IL265989A (en) | 2019-06-30 |
| BR112019005930A2 (pt) | 2019-06-11 |
| PH12019500845A1 (en) | 2019-12-02 |
| US20210212968A1 (en) | 2021-07-15 |
| EP3528800A1 (en) | 2019-08-28 |
| WO2018073154A1 (en) | 2018-04-26 |
| EA201990951A1 (ru) | 2019-11-29 |
| JP2019531320A (ja) | 2019-10-31 |
| CL2019000935A1 (es) | 2019-08-09 |
| AU2017344882A1 (en) | 2019-03-28 |
| MX2019004549A (es) | 2019-06-12 |
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