KR20170008846A - 글루코코르티코이드 및 edo-s101을 포함하는 조합물 - Google Patents

글루코코르티코이드 및 edo-s101을 포함하는 조합물 Download PDF

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Publication number
KR20170008846A
KR20170008846A KR1020167035845A KR20167035845A KR20170008846A KR 20170008846 A KR20170008846 A KR 20170008846A KR 1020167035845 A KR1020167035845 A KR 1020167035845A KR 20167035845 A KR20167035845 A KR 20167035845A KR 20170008846 A KR20170008846 A KR 20170008846A
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KR
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Prior art keywords
combination
compound
formula
pharmaceutically acceptable
glucocorticoid
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Ceased
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KR1020167035845A
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English (en)
Korean (ko)
Inventor
토마스 요르크 메를링
엔리케 마리아 오시오
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유로-셀띠끄 소시에떼 아노님
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Publication of KR20170008846A publication Critical patent/KR20170008846A/ko
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
KR1020167035845A 2014-05-28 2015-05-26 글루코코르티코이드 및 edo-s101을 포함하는 조합물 Ceased KR20170008846A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1409485.8A GB201409485D0 (en) 2014-05-28 2014-05-28 Pharmaceutical composition
GB1409485.8 2014-05-28
PCT/EP2015/061572 WO2015181157A1 (en) 2014-05-28 2015-05-26 Combination comprising a glucocorticoid and edo-s101

Publications (1)

Publication Number Publication Date
KR20170008846A true KR20170008846A (ko) 2017-01-24

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KR1020167035845A Ceased KR20170008846A (ko) 2014-05-28 2015-05-26 글루코코르티코이드 및 edo-s101을 포함하는 조합물

Country Status (20)

Country Link
US (4) US10744120B2 (https=)
EP (1) EP3148584B1 (https=)
JP (2) JP2017518292A (https=)
KR (1) KR20170008846A (https=)
CN (1) CN106488776B (https=)
AU (1) AU2015266053B2 (https=)
BR (1) BR112016027043B1 (https=)
CA (1) CA2950340C (https=)
DK (1) DK3148584T3 (https=)
EA (1) EA038323B1 (https=)
ES (1) ES2885429T3 (https=)
GB (1) GB201409485D0 (https=)
IL (1) IL249230A0 (https=)
MX (1) MX383254B (https=)
PH (1) PH12016502352A1 (https=)
SG (2) SG10201810404XA (https=)
TW (1) TWI731837B (https=)
UA (1) UA121392C2 (https=)
WO (1) WO2015181157A1 (https=)
ZA (1) ZA201607489B (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20200015563A (ko) * 2017-06-13 2020-02-12 유로-셀띠끄 소시에떼 아노님 T-세포 전림프구성 백혈병의 치료에 사용하기 위한 티노스타무스틴

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20200015563A (ko) * 2017-06-13 2020-02-12 유로-셀띠끄 소시에떼 아노님 T-세포 전림프구성 백혈병의 치료에 사용하기 위한 티노스타무스틴

Also Published As

Publication number Publication date
ZA201607489B (en) 2026-03-25
US20210059989A1 (en) 2021-03-04
BR112016027043B1 (pt) 2023-01-31
US10744120B2 (en) 2020-08-18
JP2021046446A (ja) 2021-03-25
EA038323B1 (ru) 2021-08-10
AU2015266053B2 (en) 2020-07-02
CA2950340A1 (en) 2015-12-03
US11541038B2 (en) 2023-01-03
DK3148584T3 (da) 2021-08-30
IL249230A0 (en) 2017-02-28
MX2016015437A (es) 2017-06-23
EP3148584B1 (en) 2021-05-26
AU2015266053A1 (en) 2016-11-17
EA201692481A1 (ru) 2017-04-28
CA2950340C (en) 2023-10-17
UA121392C2 (uk) 2020-05-25
US20230285363A1 (en) 2023-09-14
BR112016027043A2 (pt) 2017-08-15
US20170296513A1 (en) 2017-10-19
TWI731837B (zh) 2021-07-01
MX383254B (es) 2025-03-13
SG11201609362YA (en) 2016-12-29
BR112016027043A8 (pt) 2021-07-20
US20250049762A1 (en) 2025-02-13
EP3148584A1 (en) 2017-04-05
CN106488776A (zh) 2017-03-08
ES2885429T3 (es) 2021-12-13
GB201409485D0 (en) 2014-07-09
CN106488776B (zh) 2021-01-22
WO2015181157A1 (en) 2015-12-03
JP2017518292A (ja) 2017-07-06
PH12016502352A1 (en) 2017-02-13
US12064417B2 (en) 2024-08-20
TW201613577A (en) 2016-04-16
SG10201810404XA (en) 2018-12-28

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