KR20160106684A - 히드록시포름아미드 유도체 및 그의 용도 - Google Patents

히드록시포름아미드 유도체 및 그의 용도 Download PDF

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Publication number
KR20160106684A
KR20160106684A KR1020167021496A KR20167021496A KR20160106684A KR 20160106684 A KR20160106684 A KR 20160106684A KR 1020167021496 A KR1020167021496 A KR 1020167021496A KR 20167021496 A KR20167021496 A KR 20167021496A KR 20160106684 A KR20160106684 A KR 20160106684A
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South Korea
Prior art keywords
methyl
hydroxyformamido
heptanamido
furan
carbamoyl
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Korean (ko)
Inventor
사라 이. 다우델
힐러리 쉔크 에이댐
마크 엘반
라이언 마이클 폭스
마를리스 함몬드
마크 에이. 힐피커
트램 에이취. 호앙
라라 에스. 칼랜더
브라이언 그리핀 로혼
사라다 만스
조앤 필프
데이비드 쥐. 와쉬번
구오센 예
Original Assignee
글락소스미스클라인 인털렉츄얼 프로퍼티 (넘버 2) 리미티드
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Publication of KR20160106684A publication Critical patent/KR20160106684A/ko
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    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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KR1020167021496A 2014-01-10 2015-01-09 히드록시포름아미드 유도체 및 그의 용도 Withdrawn KR20160106684A (ko)

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US201461925848P 2014-01-10 2014-01-10
US61/925,848 2014-01-10
PCT/IB2015/050179 WO2015104684A1 (en) 2014-01-10 2015-01-09 Hydroxy formamide derivatives and their use

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US (2) US10450288B2 (OSRAM)
EP (1) EP3092233A1 (OSRAM)
JP (2) JP2017507915A (OSRAM)
KR (1) KR20160106684A (OSRAM)
CN (2) CN106103431B (OSRAM)
AU (1) AU2015205370B2 (OSRAM)
BR (1) BR112016016130A2 (OSRAM)
CA (1) CA2936467A1 (OSRAM)
CL (1) CL2016001746A1 (OSRAM)
CR (1) CR20160316A (OSRAM)
DO (1) DOP2016000170A (OSRAM)
EA (1) EA031654B1 (OSRAM)
IL (1) IL246653A0 (OSRAM)
MA (1) MA39171A1 (OSRAM)
MX (1) MX2016009064A (OSRAM)
PE (1) PE20160998A1 (OSRAM)
PH (1) PH12016501349A1 (OSRAM)
SG (1) SG11201605539SA (OSRAM)
TW (1) TW201620887A (OSRAM)
UA (1) UA118278C2 (OSRAM)
WO (1) WO2015104684A1 (OSRAM)

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JP2017507915A (ja) * 2014-01-10 2017-03-23 グラクソスミスクライン、インテレクチュアル、プロパティー、（ナンバー２）、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ （Ｎｏ．２） Ｌｉｍｉｔｅｄ ヒドロキシホルムアミド誘導体およびそれらの使用
WO2017006295A1 (en) * 2015-07-08 2017-01-12 Glaxosmithkline Intellectual Property (No.2) Limited Hydroxy formamide derivatives and their use
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