KR20120101411A - 치환된 3-페닐프로피온산 및 그의 용도 - Google Patents

치환된 3-페닐프로피온산 및 그의 용도 Download PDF

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KR20120101411A
KR20120101411A KR1020127013589A KR20127013589A KR20120101411A KR 20120101411 A KR20120101411 A KR 20120101411A KR 1020127013589 A KR1020127013589 A KR 1020127013589A KR 20127013589 A KR20127013589 A KR 20127013589A KR 20120101411 A KR20120101411 A KR 20120101411A
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South Korea
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mmol
methyl
mixture
ethyl
added
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Inventor
토마스 람페
마이클 한
조한네스-피터 스타스츠
칼-하인즈 슐레머
프랑크 분데르
셰리프 엘 쉬이크
볼크하트 민-지안 리
에바-마리아 베커
프라이데라이크 스톨
안드레아스 크노르
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바이엘 파마 악티엔게젤샤프트
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    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • C07C205/35—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/36—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/38—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to a carbon atom of a six-membered aromatic ring, e.g. nitrodiphenyl ethers
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    • C07C231/00—Preparation of carboxylic acid amides
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    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • C07C233/55—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a carbon atom of an unsaturated carbon skeleton
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    • C07D305/04—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D305/06—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring atoms
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
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  • Ophthalmology & Optometry (AREA)
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  • Communicable Diseases (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
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  • Vascular Medicine (AREA)
  • Obesity (AREA)
KR1020127013589A 2009-10-28 2010-10-21 치환된 3-페닐프로피온산 및 그의 용도 Ceased KR20120101411A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102009046115A DE102009046115A1 (de) 2009-10-28 2009-10-28 Substituierte 3-Phenylpropansäuren und ihre Verwendung
DE102009046115.9 2009-10-28

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KR20120101411A true KR20120101411A (ko) 2012-09-13

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KR1020127013589A Ceased KR20120101411A (ko) 2009-10-28 2010-10-21 치환된 3-페닐프로피온산 및 그의 용도

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US (2) US20110130445A1 (https=)
EP (1) EP2493845B1 (https=)
JP (1) JP5801312B2 (https=)
KR (1) KR20120101411A (https=)
CN (1) CN102712577B (https=)
AR (1) AR079015A1 (https=)
AU (1) AU2010311678B2 (https=)
BR (1) BR112012010057A2 (https=)
CA (1) CA2777152C (https=)
DE (1) DE102009046115A1 (https=)
DK (1) DK2493845T3 (https=)
ES (1) ES2446970T3 (https=)
HR (1) HRP20140270T1 (https=)
IL (1) IL218989A (https=)
MX (1) MX2012004951A (https=)
PL (1) PL2493845T3 (https=)
PT (1) PT2493845E (https=)
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