KR20110042356A - 제약 조성물 및 그의 투여 - Google Patents

제약 조성물 및 그의 투여 Download PDF

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Publication number
KR20110042356A
KR20110042356A KR1020117005734A KR20117005734A KR20110042356A KR 20110042356 A KR20110042356 A KR 20110042356A KR 1020117005734 A KR1020117005734 A KR 1020117005734A KR 20117005734 A KR20117005734 A KR 20117005734A KR 20110042356 A KR20110042356 A KR 20110042356A
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South Korea
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composition
solid dispersion
pharmaceutical composition
amorphous compound
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Korean (ko)
Inventor
윌리엄 로우
패트리시아 허터
크리스토퍼 영
커크 다인하트
마리누스 야코부스 페르비스
커크 오버호프
페터 디. 제이. 그루테누이스
마틴 보트필드
알프레도 그로시
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버텍스 파마슈티칼스 인코포레이티드
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Application filed by 버텍스 파마슈티칼스 인코포레이티드 filed Critical 버텍스 파마슈티칼스 인코포레이티드
Publication of KR20110042356A publication Critical patent/KR20110042356A/ko
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    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
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  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Emergency Medicine (AREA)
KR1020117005734A 2008-08-13 2009-08-13 제약 조성물 및 그의 투여 Ceased KR20110042356A (ko)

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
US8870408P 2008-08-13 2008-08-13
US61/088,704 2008-08-13
US8880108P 2008-08-14 2008-08-14
US61/088,801 2008-08-14
US9009608P 2008-08-19 2008-08-19
US61/090,096 2008-08-19
US14616309P 2009-01-21 2009-01-21
US61/146,163 2009-01-21
US18152709P 2009-05-27 2009-05-27
US61/181,527 2009-05-27
US18334509P 2009-06-02 2009-06-02
US61/183,345 2009-06-02

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020177016117A Division KR20170072950A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여

Publications (1)

Publication Number Publication Date
KR20110042356A true KR20110042356A (ko) 2011-04-26

Family

ID=41206223

Family Applications (5)

Application Number Title Priority Date Filing Date
KR1020117005734A Ceased KR20110042356A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020197037948A Ceased KR20190143497A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020247015082A Pending KR20240066199A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020177016117A Ceased KR20170072950A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020227014317A Ceased KR20220057663A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여

Family Applications After (4)

Application Number Title Priority Date Filing Date
KR1020197037948A Ceased KR20190143497A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020247015082A Pending KR20240066199A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020177016117A Ceased KR20170072950A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여
KR1020227014317A Ceased KR20220057663A (ko) 2008-08-13 2009-08-13 제약 조성물 및 그의 투여

Country Status (27)

Country Link
US (1) US20120220625A1 (enExample)
EP (3) EP3345625B1 (enExample)
JP (2) JP5575768B2 (enExample)
KR (5) KR20110042356A (enExample)
CN (1) CN102231990B (enExample)
AU (2) AU2009282419B2 (enExample)
BR (1) BRPI0916877A2 (enExample)
CA (1) CA2733908C (enExample)
CY (2) CY1119945T1 (enExample)
DK (2) DK2328618T3 (enExample)
EA (1) EA021706B1 (enExample)
ES (2) ES2660143T3 (enExample)
HR (2) HRP20180328T1 (enExample)
HU (2) HUE035931T2 (enExample)
IL (3) IL211203A (enExample)
LT (2) LT2328618T (enExample)
ME (1) ME03019B (enExample)
MX (3) MX366161B (enExample)
NO (1) NO2328618T3 (enExample)
NZ (1) NZ591535A (enExample)
PL (2) PL3345625T3 (enExample)
PT (2) PT3345625T (enExample)
RS (2) RS56894B1 (enExample)
SI (2) SI2328618T1 (enExample)
SM (2) SMT201800074T1 (enExample)
WO (1) WO2010019239A2 (enExample)
ZA (1) ZA201101097B (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20150080609A (ko) * 2012-11-02 2015-07-09 버텍스 파마슈티칼스 인코포레이티드 Cftr 매개된 질환의 치료를 위한 약제학적 조성물
KR20160047522A (ko) * 2013-08-27 2016-05-02 길리애드 파마셋 엘엘씨 2종의 항바이러스 화합물의 조합 제제
US12065432B2 (en) 2007-12-07 2024-08-20 Vertex Pharmaceuticals Incorporated Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid

Families Citing this family (115)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2006111093A (ru) 2003-09-06 2007-10-27 Вертекс Фармасьютикалз Инкорпорейтед (Us) Модуляторы атр-связывающих кассетных транспортеров
US7977322B2 (en) 2004-08-20 2011-07-12 Vertex Pharmaceuticals Incorporated Modulators of ATP-binding cassette transporters
PL2489659T3 (pl) 2004-06-24 2018-06-29 Vertex Pharma Modulatory transporterów posiadających kasetę wiążącą atp
KR20080053297A (ko) 2005-08-11 2008-06-12 버텍스 파마슈티칼스 인코포레이티드 낭포성 섬유종 트랜스막 전도도 조정자의 조절자
DK2774925T3 (en) 2005-11-08 2017-02-27 Vertex Pharma Heterocyclic modulators of ATP binding cassette transporters
NZ569327A (en) 2005-12-28 2011-09-30 Vertex Pharma 1-(benzo [d] [1,3] dioxol-5-yl) -n- (phenyl) cyclopropane- carboxamide derivatives and related compounds as modulators of ATP-binding cassette transporters for the treatment of cystic fibrosis
PT1993360T (pt) 2005-12-28 2017-05-25 Vertex Pharma Formas sólidas de n-[2,4-bis(1,1-dimetiletil)-5-hidroxifenil]-1,4-di-hidro-4-oxoquinolina-3-carboxamida
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