KR20010103798A - 피리딘 및 피리미딘 유도체와 이들의 사이토킨 매개질환의 억제제로서 용도 - Google Patents

피리딘 및 피리미딘 유도체와 이들의 사이토킨 매개질환의 억제제로서 용도 Download PDF

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Publication number
KR20010103798A
KR20010103798A KR1020017012093A KR20017012093A KR20010103798A KR 20010103798 A KR20010103798 A KR 20010103798A KR 1020017012093 A KR1020017012093 A KR 1020017012093A KR 20017012093 A KR20017012093 A KR 20017012093A KR 20010103798 A KR20010103798 A KR 20010103798A
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South Korea
Prior art keywords
alkyl
amino
alkoxy
formula
pyrimidinyl
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KR1020017012093A
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English (en)
Korean (ko)
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쿠밍존그라함
Original Assignee
다비드 에 질레스
아스트라제네카 아베
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Publication of KR20010103798A publication Critical patent/KR20010103798A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Vascular Medicine (AREA)
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  • Gastroenterology & Hepatology (AREA)
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KR1020017012093A 1999-03-23 2000-03-17 피리딘 및 피리미딘 유도체와 이들의 사이토킨 매개질환의 억제제로서 용도 KR20010103798A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9906566.6A GB9906566D0 (en) 1999-03-23 1999-03-23 Chemical compounds
GB9906566.6 1999-03-23
PCT/GB2000/001006 WO2000056738A1 (en) 1999-03-23 2000-03-17 Pyridine and pyrimidine derivatives and their use as inhibitors of cytokine mediated disease

Publications (1)

Publication Number Publication Date
KR20010103798A true KR20010103798A (ko) 2001-11-23

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ID=10850125

Family Applications (1)

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KR1020017012093A KR20010103798A (ko) 1999-03-23 2000-03-17 피리딘 및 피리미딘 유도체와 이들의 사이토킨 매개질환의 억제제로서 용도

Country Status (20)

Country Link
US (1) US6784174B1 (de)
EP (1) EP1165566B1 (de)
JP (1) JP2002540112A (de)
KR (1) KR20010103798A (de)
CN (3) CN1911931A (de)
AT (1) ATE247661T1 (de)
AU (1) AU757028B2 (de)
BR (1) BR0009223A (de)
CA (1) CA2367866A1 (de)
DE (1) DE60004655T2 (de)
DK (1) DK1165566T3 (de)
ES (1) ES2204539T3 (de)
GB (1) GB9906566D0 (de)
HK (2) HK1041886A1 (de)
IL (1) IL145303A0 (de)
NO (1) NO20014589L (de)
NZ (1) NZ514042A (de)
PT (1) PT1165566E (de)
WO (1) WO2000056738A1 (de)
ZA (1) ZA200107501B (de)

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NO20014589D0 (no) 2001-09-21
WO2000056738A1 (en) 2000-09-28
CN1911931A (zh) 2007-02-14
HK1078849A1 (en) 2006-03-24
CN1308329C (zh) 2007-04-04
ATE247661T1 (de) 2003-09-15
ZA200107501B (en) 2003-02-26
EP1165566A1 (de) 2002-01-02
PT1165566E (pt) 2004-01-30
DK1165566T3 (da) 2003-11-24
US6784174B1 (en) 2004-08-31
AU757028B2 (en) 2003-01-30
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NO20014589L (no) 2001-11-21
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AU3440100A (en) 2000-10-09
CN1351604A (zh) 2002-05-29
CN1660849A (zh) 2005-08-31
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