DK1165566T3 - Pyridin- og pyrimidinderivater og deres anvendelse som inhibitorer af cytokin-medieret sygdom - Google Patents

Pyridin- og pyrimidinderivater og deres anvendelse som inhibitorer af cytokin-medieret sygdom

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Publication number
DK1165566T3
DK1165566T3 DK00912750T DK00912750T DK1165566T3 DK 1165566 T3 DK1165566 T3 DK 1165566T3 DK 00912750 T DK00912750 T DK 00912750T DK 00912750 T DK00912750 T DK 00912750T DK 1165566 T3 DK1165566 T3 DK 1165566T3
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halo
hydroxy
amino
hydrogen
group
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DK00912750T
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English (en)
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John Graham Cumming
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Astrazeneca Ab
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Publication of DK1165566T3 publication Critical patent/DK1165566T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P11/06—Antiasthmatics
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    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
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    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Engineering & Computer Science (AREA)
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  • Cardiology (AREA)
  • Oncology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • AIDS & HIV (AREA)
  • Psychiatry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
DK00912750T 1999-03-23 2000-03-17 Pyridin- og pyrimidinderivater og deres anvendelse som inhibitorer af cytokin-medieret sygdom DK1165566T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9906566.6A GB9906566D0 (en) 1999-03-23 1999-03-23 Chemical compounds
PCT/GB2000/001006 WO2000056738A1 (en) 1999-03-23 2000-03-17 Pyridine and pyrimidine derivatives and their use as inhibitors of cytokine mediated disease

Publications (1)

Publication Number Publication Date
DK1165566T3 true DK1165566T3 (da) 2003-11-24

Family

ID=10850125

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00912750T DK1165566T3 (da) 1999-03-23 2000-03-17 Pyridin- og pyrimidinderivater og deres anvendelse som inhibitorer af cytokin-medieret sygdom

Country Status (20)

Country Link
US (1) US6784174B1 (da)
EP (1) EP1165566B1 (da)
JP (1) JP2002540112A (da)
KR (1) KR20010103798A (da)
CN (3) CN1911931A (da)
AT (1) ATE247661T1 (da)
AU (1) AU757028B2 (da)
BR (1) BR0009223A (da)
CA (1) CA2367866A1 (da)
DE (1) DE60004655T2 (da)
DK (1) DK1165566T3 (da)
ES (1) ES2204539T3 (da)
GB (1) GB9906566D0 (da)
HK (2) HK1041886A1 (da)
IL (1) IL145303A0 (da)
NO (1) NO20014589L (da)
NZ (1) NZ514042A (da)
PT (1) PT1165566E (da)
WO (1) WO2000056738A1 (da)
ZA (1) ZA200107501B (da)

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NO20014589D0 (no) 2001-09-21
WO2000056738A1 (en) 2000-09-28
CN1911931A (zh) 2007-02-14
HK1078849A1 (en) 2006-03-24
CN1308329C (zh) 2007-04-04
ATE247661T1 (de) 2003-09-15
ZA200107501B (en) 2003-02-26
EP1165566A1 (en) 2002-01-02
PT1165566E (pt) 2004-01-30
US6784174B1 (en) 2004-08-31
KR20010103798A (ko) 2001-11-23
AU757028B2 (en) 2003-01-30
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NO20014589L (no) 2001-11-21
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AU3440100A (en) 2000-10-09
CN1351604A (zh) 2002-05-29
CN1660849A (zh) 2005-08-31
IL145303A0 (en) 2002-06-30
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