KR102598775B1 - Ｒｏｒ감마 조절제 - Google Patents
Ｒｏｒ감마 조절제 Download PDFInfo
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- KR102598775B1 KR102598775B1 KR1020197015082A KR20197015082A KR102598775B1 KR 102598775 B1 KR102598775 B1 KR 102598775B1 KR 1020197015082 A KR1020197015082 A KR 1020197015082A KR 20197015082 A KR20197015082 A KR 20197015082A KR 102598775 B1 KR102598775 B1 KR 102598775B1
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Landscapes
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| MX392163B (es) | 2016-10-27 | 2025-03-21 | Escalier Biosciences Bv | Moduladores de ror gamma. |
| WO2019177997A1 (en) | 2018-03-12 | 2019-09-19 | Escalier Biosciences B.V. | Spirocyclic ror-gamma modulators |
| US11230555B2 (en) | 2018-03-12 | 2022-01-25 | Escalier Biosciences B.V. | Bicyclic RORγ modulators |
| JP2022554390A (ja) * | 2019-11-05 | 2022-12-28 | デルミラ インコーポレイテッド | Ｒｏｒガンマｔ阻害剤およびその局所使用 |
| CN115867267A (zh) * | 2020-06-30 | 2023-03-28 | 德米拉公司 | RORγt抑制剂和其局部用途 |
| CN111892599B (zh) * | 2020-08-14 | 2023-01-13 | 黄芳 | 一种2,5-二氮杂双环[2.2.2]辛烷-2-羧酸叔丁酯的合成方法 |
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| US20140187554A1 (en) * | 2011-05-16 | 2014-07-03 | The Scripps Research Institute | Modulators of the nuclear hormone receptor ror |
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| AU2003280558A1 (en) * | 2002-10-11 | 2004-05-04 | Kowa Co., Ltd. | Method for treatment of cancer |
| HUP1100166A2 (en) * | 2011-03-29 | 2012-12-28 | Sanofi Sa | Reductive amination process for preparation of dronedarone using amine intermediary compound |
| JP2014526494A (ja) * | 2011-09-19 | 2014-10-06 | イーティーエイチ・チューリッヒ | ＲＯＲγ修飾剤 |
| TW201408652A (zh) | 2012-07-11 | 2014-03-01 | Hoffmann La Roche | 作爲ＲＯＲｃ調節劑之芳基磺內醯胺衍生物 |
| CN107614062A (zh) * | 2015-03-12 | 2018-01-19 | 加利福尼亚大学董事会 | 用RORγ抑制剂治疗癌症的方法 |
| MX392163B (es) | 2016-10-27 | 2025-03-21 | Escalier Biosciences Bv | Moduladores de ror gamma. |
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009138438A1 (en) | 2008-05-15 | 2009-11-19 | N.V. Organon | N- (1, 1, 1, 3, 3, 3-hexafluoro-2-hydroxypropan-2-yl) benzyl-n' -arylcarbonylpiperaz ine derivatives |
| US20140187554A1 (en) * | 2011-05-16 | 2014-07-03 | The Scripps Research Institute | Modulators of the nuclear hormone receptor ror |
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| US20210069182A1 (en) | 2021-03-11 |
| CN110139652A (zh) | 2019-08-16 |
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| US20190269674A1 (en) | 2019-09-05 |
| CN110139652B (zh) | 2022-10-11 |
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| RU2753490C2 (ru) | 2021-08-17 |
| US20230277527A1 (en) | 2023-09-07 |
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