KR102239649B1 - 염증성 장 질환의 치료를 위한 티아졸로 피리미딘온의 용도 - Google Patents

염증성 장 질환의 치료를 위한 티아졸로 피리미딘온의 용도 Download PDF

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KR102239649B1
KR102239649B1 KR1020157033744A KR20157033744A KR102239649B1 KR 102239649 B1 KR102239649 B1 KR 102239649B1 KR 1020157033744 A KR1020157033744 A KR 1020157033744A KR 20157033744 A KR20157033744 A KR 20157033744A KR 102239649 B1 KR102239649 B1 KR 102239649B1
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compound
pharmaceutical composition
composition
dose
present
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KR1020157033744A
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Korean (ko)
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KR20160008571A (ko
Inventor
차이타냐 두트
비제이 차우타이왈르
람 굽타
시타르쿠마르 잠바드
샤일레시 데시판드
지그네스 코테차
라메시 굽타
산제이 스리바스타바
락스미칸트 치파
자야 아브라함
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토렌트 파마슈티칼스 리미티드
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
KR1020157033744A 2013-05-14 2014-05-12 염증성 장 질환의 치료를 위한 티아졸로 피리미딘온의 용도 Expired - Fee Related KR102239649B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN1718MU2013 2013-05-14
IN1718/MUM/2013 2013-05-14
IN2309MU2013 2013-07-09
IN2309/MUM/2013 2013-07-09
PCT/IB2014/000707 WO2014184631A1 (en) 2013-05-14 2014-05-12 Use of a thiazolo pyrimidinone for the treatment of inflammatory bowel disease

Publications (2)

Publication Number Publication Date
KR20160008571A KR20160008571A (ko) 2016-01-22
KR102239649B1 true KR102239649B1 (ko) 2021-04-12

Family

ID=50896342

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020157033744A Expired - Fee Related KR102239649B1 (ko) 2013-05-14 2014-05-12 염증성 장 질환의 치료를 위한 티아졸로 피리미딘온의 용도

Country Status (28)

Country Link
US (2) US9610247B2 (https=)
EP (1) EP2996693B1 (https=)
JP (1) JP6407974B2 (https=)
KR (1) KR102239649B1 (https=)
CN (1) CN105209043B (https=)
AU (1) AU2014266968B2 (https=)
BR (1) BR112015028581B1 (https=)
CA (1) CA2912011C (https=)
CY (1) CY1121280T1 (https=)
DK (1) DK2996693T3 (https=)
EA (1) EA030590B1 (https=)
ES (1) ES2712705T3 (https=)
HR (1) HRP20190315T1 (https=)
HU (1) HUE042691T2 (https=)
IL (1) IL242490B (https=)
LT (1) LT2996693T (https=)
MX (1) MX358198B (https=)
MY (1) MY179215A (https=)
PH (1) PH12015502560B1 (https=)
PL (1) PL2996693T3 (https=)
PT (1) PT2996693T (https=)
RS (1) RS58423B1 (https=)
SG (1) SG11201509275PA (https=)
SI (1) SI2996693T1 (https=)
SM (1) SMT201900111T1 (https=)
TW (1) TWI661828B (https=)
UA (1) UA117244C2 (https=)
WO (1) WO2014184631A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11324829B2 (en) * 2016-03-14 2022-05-10 Santen Pharmaceutical Co., Ltd. Antiseptic agent comprising meglumine or salt thereof

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009002533A1 (en) * 2007-06-27 2008-12-31 The Brigham And Women's Hospital, Inc. Inflammatory bowel disease therapies
US20110130414A1 (en) * 2009-11-27 2011-06-02 Torrent Pharmaceuticals Limited Novel fused thiazolo and oxazolo pyrimidinones

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI500623B (zh) * 2009-10-13 2015-09-21 Torrent Pharmaceuticals Ltd 新穎稠合噻唑及噁唑嘧啶酮

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009002533A1 (en) * 2007-06-27 2008-12-31 The Brigham And Women's Hospital, Inc. Inflammatory bowel disease therapies
US20110130414A1 (en) * 2009-11-27 2011-06-02 Torrent Pharmaceuticals Limited Novel fused thiazolo and oxazolo pyrimidinones

Also Published As

Publication number Publication date
CN105209043B (zh) 2019-07-02
ES2712705T3 (es) 2019-05-14
HUE042691T2 (hu) 2019-07-29
US10471005B2 (en) 2019-11-12
SG11201509275PA (en) 2015-12-30
SI2996693T1 (sl) 2019-04-30
AU2014266968B2 (en) 2019-09-19
TW201513866A (zh) 2015-04-16
RS58423B1 (sr) 2019-04-30
MX358198B (es) 2018-08-08
MY179215A (en) 2020-11-02
NZ714098A (en) 2020-12-18
DK2996693T3 (en) 2019-03-18
PL2996693T3 (pl) 2019-05-31
JP2016518440A (ja) 2016-06-23
SMT201900111T1 (it) 2019-02-28
WO2014184631A1 (en) 2014-11-20
LT2996693T (lt) 2019-03-12
EP2996693B1 (en) 2018-12-12
PT2996693T (pt) 2019-02-27
US20170157129A1 (en) 2017-06-08
US20160120801A1 (en) 2016-05-05
EP2996693A1 (en) 2016-03-23
PH12015502560A1 (en) 2016-02-22
AU2014266968A1 (en) 2015-12-03
JP6407974B2 (ja) 2018-10-17
US9610247B2 (en) 2017-04-04
PH12015502560B1 (en) 2016-02-22
BR112015028581B1 (pt) 2022-05-03
CN105209043A (zh) 2015-12-30
CA2912011C (en) 2021-10-26
CY1121280T1 (el) 2020-05-29
EA201592159A1 (ru) 2016-04-29
IL242490B (en) 2018-11-29
TWI661828B (zh) 2019-06-11
UA117244C2 (uk) 2018-07-10
CA2912011A1 (en) 2014-11-20
HRP20190315T1 (hr) 2019-04-05
MX2015015682A (es) 2016-07-20
EA030590B1 (ru) 2018-08-31
BR112015028581A2 (pt) 2017-07-25
KR20160008571A (ko) 2016-01-22

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