KR101977920B1 - 제초 작용을 가지는 3-페닐이속사졸린 유도체 - Google Patents

제초 작용을 가지는 3-페닐이속사졸린 유도체 Download PDF

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KR101977920B1
KR101977920B1 KR1020157010148A KR20157010148A KR101977920B1 KR 101977920 B1 KR101977920 B1 KR 101977920B1 KR 1020157010148 A KR1020157010148 A KR 1020157010148A KR 20157010148 A KR20157010148 A KR 20157010148A KR 101977920 B1 KR101977920 B1 KR 101977920B1
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methyl
dihydro
oxazole
chlorine
fluorine
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KR20150063445A (ko
Inventor
비르기트 쿤
로타르 빌름스
토마스 프렌젤
클라우스 베른하르트 하프
스테판 다비트 린델
한스외르크 디트리히
디르크 슈무츨러
엘마르 가츠바일러
크리스토퍼 휴 로징거
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바이엘 크롭사이언스 악티엔게젤샤프트
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1020157010148A 2012-09-25 2013-09-19 제초 작용을 가지는 3-페닐이속사졸린 유도체 Active KR101977920B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12185768 2012-09-25
EP12185768.4 2012-09-25
PCT/EP2013/069453 WO2014048827A1 (de) 2012-09-25 2013-09-19 Herbizid wirksame 3-phenylisoxazolinderivate

Publications (2)

Publication Number Publication Date
KR20150063445A KR20150063445A (ko) 2015-06-09
KR101977920B1 true KR101977920B1 (ko) 2019-05-13

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KR1020157010148A Active KR101977920B1 (ko) 2012-09-25 2013-09-19 제초 작용을 가지는 3-페닐이속사졸린 유도체

Country Status (13)

Country Link
US (1) US9585392B2 (https=)
EP (1) EP2900645B1 (https=)
JP (1) JP6472382B2 (https=)
KR (1) KR101977920B1 (https=)
CN (1) CN104812739B (https=)
BR (1) BR112015006573B1 (https=)
DK (1) DK2900645T3 (https=)
ES (1) ES2747483T3 (https=)
IL (1) IL237685B (https=)
IN (1) IN2015DN01315A (https=)
MX (1) MX378312B (https=)
TW (1) TWI598344B (https=)
WO (1) WO2014048827A1 (https=)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014048882A1 (de) 2012-09-25 2014-04-03 Bayer Cropscience Ag Herbizid und fungizid wirksame 5-oxy-substituierte 3-phenylisoxazolin-5-carboxamide und 5-oxy-substituierte 3-phenylisoxazolin-5-thioamide
JP6397820B2 (ja) 2012-09-25 2018-09-26 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 除草活性と殺菌活性を示す3−ヘテロアリール−イソオキサゾリン−5−カルボキサミド類及び3−ヘテロアリール−イソオキサゾリン−5−チオアミド類
CN105753853B (zh) 2014-12-16 2020-08-04 沈阳中化农药化工研发有限公司 一种含异恶唑啉的脲嘧啶类化合物及其用途
CN105198824B (zh) * 2015-10-09 2018-08-31 苏州大学 一种二氢异噁唑啉化合物及其制备方法和应用
CN110799511B (zh) 2017-06-13 2023-09-01 拜耳公司 除草活性的四氢和二氢呋喃甲酰胺的3-苯基异噁唑啉-5-甲酰胺
WO2018228985A1 (de) 2017-06-13 2018-12-20 Bayer Aktiengesellschaft Herbizid wirksame 3-phenylisoxazolin-5-carboxamide von tetrahydro- und dihydrofurancarbonsäuren und -estern
CN111164077B (zh) 2017-08-17 2023-12-19 拜耳公司 除草活性的环戊基羧酸和其酯的3-苯基-5-三氟甲基异噁唑啉-5-甲酰胺
EA202091774A1 (ru) * 2018-01-25 2020-12-07 Байер Акциенгезельшафт Гербицидно-активные 3-фенилизоксазолин-5-карбоксамиды производных циклопентенилкарбоновой кислоты
CA3133025A1 (en) 2019-03-12 2020-09-17 Bayer Aktiengesellschaft Herbicidally active 3-phenylisoxazoline-5-carboxamides of s-containing cyclopentenyl carboxylic acid esters
CN112745269B (zh) * 2019-10-29 2023-01-24 沈阳中化农药化工研发有限公司 一种苯基异恶唑啉类化合物及其用途
ES3009408T3 (en) 2020-04-14 2025-03-26 Basf Se Beta-lactams and their use as herbicides
CN115515962B (zh) 2020-05-05 2025-04-29 巴斯夫欧洲公司 稠合异噁唑啉衍生物及其作为除草剂的用途
IL301695A (en) 2020-10-01 2023-05-01 Bayer Ag Benzaldehyde oximes and method for producing same
CN116568673A (zh) * 2020-11-24 2023-08-08 先正达农作物保护股份公司 除草化合物
KR20230155446A (ko) 2021-03-09 2023-11-10 바스프 에스이 말론아미드 및 제초제로서의 그의 용도
EP4363407B1 (de) * 2021-06-29 2025-04-16 Bayer Aktiengesellschaft Verfahren zur herstellung von isoxazolincarbonsäure-derivaten
EP4441035A1 (de) * 2021-12-03 2024-10-09 Bayer Aktiengesellschaft Verfahren zur herstellung von isoxazolin-5,5-vinylcarbonsäure-derivaten
CN114436834A (zh) * 2021-12-16 2022-05-06 江苏阿尔法药业股份有限公司 一种利用连续流微通道反应器合成瑞舒伐他汀钙中间体的方法
AU2023206316A1 (en) 2022-01-14 2024-08-29 Enko Chem, Inc. Protoporphyrinogen oxidase inhibitors
AU2024283657A1 (en) 2023-06-04 2026-01-22 Jiangsu Flag Chemical Industry Co., Ltd. 3-phenylisoxazoline-5-carboxamide compound, and preparation method therefor, herbicidal composition thereof and use thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001510835A (ja) * 1997-07-23 2001-08-07 ビーエーエスエフ アクチェンゲゼルシャフト 置換3−フェニルイソオキサゾリン

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8422701D0 (en) * 1984-09-07 1984-10-10 Shell Int Research Ether herbicides
GB8423252D0 (en) * 1984-09-14 1984-10-17 Shell Int Research Ether herbicides
JPS62103070A (ja) * 1985-10-29 1987-05-13 Mitsui Toatsu Chem Inc イソオキサゾリン誘導体および植物生長調節剤
DE3541722A1 (de) * 1985-11-26 1987-05-27 Basf Ag Chinolinderivate und ihre verwendung zur bekaempfung von unerwuenschtem pflanzenwachstum
US4956006A (en) * 1988-12-27 1990-09-11 Ici Americas Inc. Substituted 1-phenyl pyrrolidones and their use as herbicides
DE4026018A1 (de) * 1990-08-17 1992-02-20 Hoechst Ag Isoxazoline oder isothiazoline enthaltende pflanzenschuetzende mittel und neue isoxazoline und isothiazoline
WO1995014680A1 (en) * 1993-11-26 1995-06-01 Pfizer Inc. 3-aryl-2-isoxazolines as antiinflammatory agents
ATE154932T1 (de) * 1993-11-26 1997-07-15 Pfizer Isoxazolinverbindungen als entzündungshemmende mittel
US5939418A (en) 1995-12-21 1999-08-17 The Dupont Merck Pharmaceutical Company Isoxazoline, isothiazoline and pyrazoline factor Xa inhibitors
ATE318801T1 (de) * 1999-08-10 2006-03-15 Kumiai Chemical Industry Co Isoxazolin derivate und herbizide, die diese als aktiven bestandteil enthalten
KR100594544B1 (ko) 2003-08-27 2006-06-30 주식회사 엘지생명과학 이소옥사졸린 구조를 갖는 캐스파제 저해제
JP2007504123A (ja) 2003-08-29 2007-03-01 ランバクシー ラボラトリーズ リミテッド Iv型ホスホジエステラーゼの阻害剤
JP2005112840A (ja) * 2003-09-16 2005-04-28 Nissan Chem Ind Ltd 新規ピラゾールスルホニルウレア化合物および除草剤
EP1694655A2 (en) * 2003-11-26 2006-08-30 Ranbaxy Laboratories Limited Phosphodiesterase inhibitors
EA200900472A1 (ru) * 2006-09-22 2009-10-30 Ранбакси Лабораторис Лимитед Ингибиторы фосфодиэстеразы iv типа
US9078442B2 (en) 2011-03-31 2015-07-14 Bayer Intellectual Property Gmbh Herbicidally and fungicidally active 3-phenylisoxazoline-5-carboxamides and 3-phenylisoxazoline-5-thioamides
WO2014048882A1 (de) 2012-09-25 2014-04-03 Bayer Cropscience Ag Herbizid und fungizid wirksame 5-oxy-substituierte 3-phenylisoxazolin-5-carboxamide und 5-oxy-substituierte 3-phenylisoxazolin-5-thioamide
JP6397820B2 (ja) 2012-09-25 2018-09-26 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 除草活性と殺菌活性を示す3−ヘテロアリール−イソオキサゾリン−5−カルボキサミド類及び3−ヘテロアリール−イソオキサゾリン−5−チオアミド類

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001510835A (ja) * 1997-07-23 2001-08-07 ビーエーエスエフ アクチェンゲゼルシャフト 置換3−フェニルイソオキサゾリン

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
J. Med. Chem. 1999, 42, 2760-2773 "Design and Synthesis of Isoxazoline Derivatives as Factor Xa Inhibitors"
Pestycydy/Pesticides, 2010, (1-4), 21-31. "Synthesis and fungicidal activity of substituted isoxazolecarboxamides"

Also Published As

Publication number Publication date
JP2015530397A (ja) 2015-10-15
KR20150063445A (ko) 2015-06-09
EP2900645B1 (de) 2019-08-21
CN104812739A (zh) 2015-07-29
BR112015006573B1 (pt) 2020-11-03
EP2900645A1 (de) 2015-08-05
US9585392B2 (en) 2017-03-07
IL237685A0 (en) 2015-05-31
US20150245615A1 (en) 2015-09-03
IN2015DN01315A (https=) 2015-07-03
MX2015003538A (es) 2015-10-12
IL237685B (en) 2019-11-28
WO2014048827A1 (de) 2014-04-03
TWI598344B (zh) 2017-09-11
DK2900645T3 (da) 2019-10-14
ES2747483T3 (es) 2020-03-10
MX378312B (es) 2025-03-10
TW201418231A (zh) 2014-05-16
JP6472382B2 (ja) 2019-02-20
CN104812739B (zh) 2017-12-12
BR112015006573A2 (pt) 2017-07-04

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