KR101931204B1 - 알킬아미도티아졸, 상기 알킬아미도티아졸을 함유한 화장료 또는 피부학적 제제, 및 피부의 요망되지 않는 색소침착을 치료하거나 예방하기 위한 이의 용도 - Google Patents
알킬아미도티아졸, 상기 알킬아미도티아졸을 함유한 화장료 또는 피부학적 제제, 및 피부의 요망되지 않는 색소침착을 치료하거나 예방하기 위한 이의 용도 Download PDFInfo
- Publication number
- KR101931204B1 KR101931204B1 KR1020147010924A KR20147010924A KR101931204B1 KR 101931204 B1 KR101931204 B1 KR 101931204B1 KR 1020147010924 A KR1020147010924 A KR 1020147010924A KR 20147010924 A KR20147010924 A KR 20147010924A KR 101931204 B1 KR101931204 B1 KR 101931204B1
- Authority
- KR
- South Korea
- Prior art keywords
- alkyl
- dihydroxyphenyl
- branched
- thiazol
- linear
- Prior art date
Links
- WIDNAJNXDPHROL-UHFFFAOYSA-N CC(C)C(Nc1nc(-c(c(O)c2)ccc2O)c[s]1)=O Chemical compound CC(C)C(Nc1nc(-c(c(O)c2)ccc2O)c[s]1)=O WIDNAJNXDPHROL-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/02—Preparations for care of the skin for chemically bleaching or whitening the skin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102011083259.9 | 2011-09-23 | ||
| DE102011083259A DE102011083259A1 (de) | 2011-09-23 | 2011-09-23 | Alkylamidothiazole, deren kosmetische oder dermatologische Verwendung sowie kosmetische oder dermatologische Zubereitungen mit einem Gehalt an solchen Alkylamidothiazolen |
| PCT/EP2012/068362 WO2013041526A1 (de) | 2011-09-23 | 2012-09-18 | Alkylamidothiazole, sie enthaltende kosmetische oder dermatologische zubereitungen und deren verwendung zur bekämpfung und prophylaxe unerwünschter pigmentierung der haut |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20140065471A KR20140065471A (ko) | 2014-05-29 |
| KR101931204B1 true KR101931204B1 (ko) | 2018-12-21 |
Family
ID=46889035
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020147010924A KR101931204B1 (ko) | 2011-09-23 | 2012-09-18 | 알킬아미도티아졸, 상기 알킬아미도티아졸을 함유한 화장료 또는 피부학적 제제, 및 피부의 요망되지 않는 색소침착을 치료하거나 예방하기 위한 이의 용도 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9533963B2 (de) |
| EP (2) | EP2758381B1 (de) |
| JP (1) | JP6113171B2 (de) |
| KR (1) | KR101931204B1 (de) |
| CN (1) | CN103906737B (de) |
| AU (1) | AU2012311606C1 (de) |
| BR (1) | BR112014006455B1 (de) |
| CA (1) | CA2848599C (de) |
| DE (1) | DE102011083259A1 (de) |
| ES (2) | ES2735136T3 (de) |
| MX (1) | MX347203B (de) |
| PL (2) | PL3176156T3 (de) |
| WO (1) | WO2013041526A1 (de) |
| ZA (1) | ZA201400357B (de) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102013204081A1 (de) * | 2013-03-11 | 2014-09-11 | Beiersdorf Ag | Wirkstoffkombinationen aus Alkylamidothiazolen und einen oder mehreren kosmetisch oder dermatologisch unbedenklichen Konservierungsmitteln |
| DE102013204088A1 (de) * | 2013-03-11 | 2014-09-11 | Beiersdorf Ag | Wirkstoffkombinationen aus Alkylamidothiazolen und einen oder mehreren kosmetisch oder dermatologisch relevanten Duftstoffen |
| RU2552529C1 (ru) * | 2013-11-29 | 2015-06-10 | Федеральное государственное бюджетное учреждение "Медицинский радиологический научный центр" Министерства здравоохранения Российской Федерации (ФГБУ МРНЦ Минздрава России) | Вазопрессорное средство |
| DE102013226746A1 (de) * | 2013-12-19 | 2015-06-25 | Beiersdorf Ag | Verwendung von Alkylamidothiazolen als Antioxidans oder Radikalfänger in kosmetischen oder dermatologischen Zubereitungen |
| DE102013226711A1 (de) * | 2013-12-19 | 2015-06-25 | Beiersdorf Ag | Verwendung von Alkylamidothiazolen in kosmetischen oder dermatologischen Zubereitungen zur Prophylaxe vor und Behandlung von sensibler Haut |
| KR101700946B1 (ko) | 2014-11-11 | 2017-02-02 | 연세대학교 산학협력단 | Ｃｘｃｒ４ 길항제를 포함하는 피부 색소침착의 예방 또는 개선용 조성물 |
| CH713170B1 (de) * | 2017-05-22 | 2018-05-31 | La Prairie Group Ag | Kosmetische oder dermatologische Zubereitung, enthaltend einen wässrigen und einen lipophilen Fischeiextrakt. |
| DE102018211412A1 (de) * | 2018-07-10 | 2020-01-16 | Beiersdorf Ag | Selbstklebende flächige Produkte enthaltend ein oder mehrere Alkylamidothiazole |
| DE202018004125U1 (de) | 2018-09-05 | 2018-10-11 | Beiersdorf Ag | Alkylamidothiazole in Polypropylen-haltigen Packmitteln |
| MX2022015522A (es) | 2020-06-15 | 2023-01-16 | Dsm Ip Assets Bv | Proceso para la elaboracion de alquilamidotiazoles. |
| DE102020210535A1 (de) | 2020-08-19 | 2022-03-24 | Beiersdorf Aktiengesellschaft | Neue Isobutyramidderivate, kosmetische und/oder dermatologischen Zubereitungen, solche Verbindungen enthaltend, sowie deren Verwendung zur Prophylaxe vor und Behandlung von sensibler, insbesondere entzündeter Haut bzw. entzündlichen Hautzuständen |
| CN111943908B (zh) * | 2020-08-24 | 2022-07-19 | 泰州瑞仕诺医药科技有限公司 | 一种制备异丁酰胺基噻唑基间苯二酚的方法 |
| DE102022209937A1 (de) | 2022-09-21 | 2024-03-21 | Beiersdorf Aktiengesellschaft | Wirkstoffkombinationen aus Alkylamidothiazolen und einem oder mehreren Biopolymeren |
| CN116554122B (zh) * | 2023-06-29 | 2023-09-19 | 南京桦冠生物技术有限公司 | α-酮酸酰胺或取代草酸酰胺酯类化合物及其组合物 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090258915A1 (en) * | 2008-04-08 | 2009-10-15 | Yun Yen | Ribonucleotide reductase inhibitors and methods of use |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH07215952A (ja) * | 1993-12-06 | 1995-08-15 | Otsuka Pharmaceut Factory Inc | カテコール誘導体 |
| EP1027050B1 (de) * | 1997-10-27 | 2004-01-14 | Takeda Chemical Industries, Ltd. | 1,3-thiazole als adenosine a3 rezeptor antagonisten zur behandlung von asthma, allergien und diabetes |
| US20040224992A1 (en) * | 2003-02-27 | 2004-11-11 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| US20070042997A1 (en) | 2003-07-16 | 2007-02-22 | Akiko Itai | Medicament for treatment of dermal pigmentation |
| AU2007301126A1 (en) | 2006-09-28 | 2008-04-03 | Banyu Pharmaceutical Co., Ltd. | Diaryl ketimine derivative |
| ES2655305T3 (es) | 2008-02-08 | 2018-02-19 | Shiseido Company, Ltd. | Agente para blanqueamiento de la piel |
| DE102010012594A1 (de) * | 2010-03-23 | 2011-09-29 | Beiersdorf Ag | Kosmetische oder dermatologische Zubereitungen mit einem Gehalt an einem oder mehreren Thiazolderivaten |
-
2011
- 2011-09-23 DE DE102011083259A patent/DE102011083259A1/de not_active Withdrawn
-
2012
- 2012-09-18 EP EP12762266.0A patent/EP2758381B1/de active Active
- 2012-09-18 KR KR1020147010924A patent/KR101931204B1/ko active IP Right Grant
- 2012-09-18 AU AU2012311606A patent/AU2012311606C1/en active Active
- 2012-09-18 PL PL16204983T patent/PL3176156T3/pl unknown
- 2012-09-18 WO PCT/EP2012/068362 patent/WO2013041526A1/de active Application Filing
- 2012-09-18 CN CN201280045929.5A patent/CN103906737B/zh active Active
- 2012-09-18 BR BR112014006455A patent/BR112014006455B1/pt active IP Right Grant
- 2012-09-18 ES ES16204983T patent/ES2735136T3/es active Active
- 2012-09-18 MX MX2014003448A patent/MX347203B/es active IP Right Grant
- 2012-09-18 PL PL12762266T patent/PL2758381T3/pl unknown
- 2012-09-18 JP JP2014531196A patent/JP6113171B2/ja active Active
- 2012-09-18 ES ES12762266.0T patent/ES2626609T3/es active Active
- 2012-09-18 US US14/126,078 patent/US9533963B2/en active Active
- 2012-09-18 EP EP16204983.7A patent/EP3176156B1/de active Active
- 2012-09-18 CA CA2848599A patent/CA2848599C/en active Active
-
2014
- 2014-01-16 ZA ZA2014/00357A patent/ZA201400357B/en unknown
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090258915A1 (en) * | 2008-04-08 | 2009-10-15 | Yun Yen | Ribonucleotide reductase inhibitors and methods of use |
Non-Patent Citations (2)
| Title |
|---|
| Heteroatom Chemistry., 2006, Vol.17, No.4, pp 254-260* |
| STN Database Registry [Online; 1998.05.27.]* |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2013041526A1 (de) | 2013-03-28 |
| KR20140065471A (ko) | 2014-05-29 |
| MX2014003448A (es) | 2014-09-22 |
| AU2012311606B2 (en) | 2016-12-15 |
| AU2012311606A1 (en) | 2014-02-20 |
| PL3176156T3 (pl) | 2019-10-31 |
| CA2848599A1 (en) | 2013-03-28 |
| NZ620487A (en) | 2016-02-26 |
| EP3176156B1 (de) | 2019-06-12 |
| MX347203B (es) | 2017-04-19 |
| CN103906737A (zh) | 2014-07-02 |
| CN103906737B (zh) | 2016-09-28 |
| BR112014006455A2 (pt) | 2017-03-28 |
| ES2626609T3 (es) | 2017-07-25 |
| US9533963B2 (en) | 2017-01-03 |
| BR112014006455B1 (pt) | 2019-08-13 |
| EP3176156A1 (de) | 2017-06-07 |
| CA2848599C (en) | 2019-10-01 |
| EP2758381A1 (de) | 2014-07-30 |
| JP2014526535A (ja) | 2014-10-06 |
| PL2758381T3 (pl) | 2017-08-31 |
| JP6113171B2 (ja) | 2017-04-12 |
| ZA201400357B (en) | 2015-09-30 |
| EP2758381B1 (de) | 2017-03-01 |
| DE102011083259A1 (de) | 2013-03-28 |
| AU2012311606C1 (en) | 2018-05-17 |
| ES2735136T3 (es) | 2019-12-16 |
| US20140121250A1 (en) | 2014-05-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A201 | Request for examination | ||
| E902 | Notification of reason for refusal | ||
| E701 | Decision to grant or registration of patent right |