KR101773070B1 - 아릴 및 헤테로아릴아세트산 유도체의 제조방법 - Google Patents

아릴 및 헤테로아릴아세트산 유도체의 제조방법 Download PDF

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KR101773070B1
KR101773070B1 KR1020127021635A KR20127021635A KR101773070B1 KR 101773070 B1 KR101773070 B1 KR 101773070B1 KR 1020127021635 A KR1020127021635 A KR 1020127021635A KR 20127021635 A KR20127021635 A KR 20127021635A KR 101773070 B1 KR101773070 B1 KR 101773070B1
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alkyl
propyl
ethyl
methyl
hydrogen
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KR20120116491A (ko
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토마스 히믈러
루카스 제이. 구쎈
베티나 지머만
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바이엘 인텔렉쳐 프로퍼티 게엠베하
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
    • C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
KR1020127021635A 2010-01-19 2011-01-14 아릴 및 헤테로아릴아세트산 유도체의 제조방법 Active KR101773070B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US29608110P 2010-01-19 2010-01-19
EP10151081 2010-01-19
US61/296,081 2010-01-19
EP10151081.6 2010-01-19
PCT/EP2011/050456 WO2011089072A1 (de) 2010-01-19 2011-01-14 Verfahren zur herstellung von aryl- und heteroarylessigsäure-derivaten

Publications (2)

Publication Number Publication Date
KR20120116491A KR20120116491A (ko) 2012-10-22
KR101773070B1 true KR101773070B1 (ko) 2017-09-12

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KR1020127021635A Active KR101773070B1 (ko) 2010-01-19 2011-01-14 아릴 및 헤테로아릴아세트산 유도체의 제조방법

Country Status (10)

Country Link
US (1) US8507688B2 (enExample)
EP (1) EP2526081B1 (enExample)
JP (1) JP5899119B2 (enExample)
KR (1) KR101773070B1 (enExample)
CN (1) CN102753513B (enExample)
DK (1) DK2526081T3 (enExample)
ES (1) ES2546487T3 (enExample)
IL (1) IL220787A (enExample)
IN (1) IN2012DN06383A (enExample)
WO (1) WO2011089072A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9096568B2 (en) * 2011-03-02 2015-08-04 Bayer Intellectual Property Gmbh Process for preparing aryl- and heteroarylacetic acid derivatives
BR112020019277B1 (pt) 2018-04-10 2024-01-16 Bayer Aktiengesellschaft Processo para produção de ácidos 2,6-dialquilfenil acéticos, e seus intermediários
CN113121341A (zh) * 2019-12-31 2021-07-16 江苏中旗科技股份有限公司 一种合成2,6-二乙基-4-甲基苯乙酸酯的方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001114763A (ja) * 1995-06-28 2001-04-24 Sanofi-Synthelabo 神経栄養活性および神経保護活性を有する４−アリール−１−フェニルアルキル−１，２，３，６−テトラヒドロピリジン
US20030203935A1 (en) * 1999-05-17 2003-10-30 Teijin Limited Cyanobiphenyl derivatives
JP2004524328A (ja) * 2001-03-09 2004-08-12 シュトゥディエンゲゼルシャフト・コーレ・ミット・ベシュレンクテル・ハフツング ビニル、アリールおよびヘテロアリール酢酸およびその誘導体の製造法
US20050038289A1 (en) * 2001-07-23 2005-02-17 Gordon Richard S Chemical reactions in compressed carbon dioxide

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2189877T3 (es) 1995-06-30 2003-07-16 Bayer Cropscience Ag Cetoenoles dialquil-halogenofenilsubstituidos para el empleo como herbicidas y pesticidas.

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001114763A (ja) * 1995-06-28 2001-04-24 Sanofi-Synthelabo 神経栄養活性および神経保護活性を有する４−アリール−１−フェニルアルキル−１，２，３，６−テトラヒドロピリジン
US20030203935A1 (en) * 1999-05-17 2003-10-30 Teijin Limited Cyanobiphenyl derivatives
JP2004524328A (ja) * 2001-03-09 2004-08-12 シュトゥディエンゲゼルシャフト・コーレ・ミット・ベシュレンクテル・ハフツング ビニル、アリールおよびヘテロアリール酢酸およびその誘導体の製造法
US20050038289A1 (en) * 2001-07-23 2005-02-17 Gordon Richard S Chemical reactions in compressed carbon dioxide

Also Published As

Publication number Publication date
CN102753513B (zh) 2015-03-18
WO2011089072A1 (de) 2011-07-28
EP2526081B1 (de) 2015-07-01
CN102753513A (zh) 2012-10-24
ES2546487T3 (es) 2015-09-24
JP2013517255A (ja) 2013-05-16
EP2526081A1 (de) 2012-11-28
IL220787A (en) 2015-05-31
US20110184180A1 (en) 2011-07-28
JP5899119B2 (ja) 2016-04-06
KR20120116491A (ko) 2012-10-22
IN2012DN06383A (enExample) 2015-10-02
DK2526081T3 (en) 2015-10-05
US8507688B2 (en) 2013-08-13

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