CN102753513B - 制备芳基和杂芳基乙酸衍生物的方法 - Google Patents

制备芳基和杂芳基乙酸衍生物的方法 Download PDF

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Publication number
CN102753513B
CN102753513B CN201180009550.4A CN201180009550A CN102753513B CN 102753513 B CN102753513 B CN 102753513B CN 201180009550 A CN201180009550 A CN 201180009550A CN 102753513 B CN102753513 B CN 102753513B
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hydrogen
alkyl
compound
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Chinese (zh)
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CN102753513A (zh
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T·希姆勒
L·J·古森
B·齐默尔曼
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Bayer CropScience AG
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Bayer Intellectual Property GmbH
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
    • C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CN201180009550.4A 2010-01-19 2011-01-14 制备芳基和杂芳基乙酸衍生物的方法 Active CN102753513B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US29608110P 2010-01-19 2010-01-19
EP10151081 2010-01-19
US61/296,081 2010-01-19
EP10151081.6 2010-01-19
PCT/EP2011/050456 WO2011089072A1 (de) 2010-01-19 2011-01-14 Verfahren zur herstellung von aryl- und heteroarylessigsäure-derivaten

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CN102753513A CN102753513A (zh) 2012-10-24
CN102753513B true CN102753513B (zh) 2015-03-18

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US (1) US8507688B2 (enExample)
EP (1) EP2526081B1 (enExample)
JP (1) JP5899119B2 (enExample)
KR (1) KR101773070B1 (enExample)
CN (1) CN102753513B (enExample)
DK (1) DK2526081T3 (enExample)
ES (1) ES2546487T3 (enExample)
IL (1) IL220787A (enExample)
IN (1) IN2012DN06383A (enExample)
WO (1) WO2011089072A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9096568B2 (en) * 2011-03-02 2015-08-04 Bayer Intellectual Property Gmbh Process for preparing aryl- and heteroarylacetic acid derivatives
BR112020019277B1 (pt) 2018-04-10 2024-01-16 Bayer Aktiengesellschaft Processo para produção de ácidos 2,6-dialquilfenil acéticos, e seus intermediários
CN113121341A (zh) * 2019-12-31 2021-07-16 江苏中旗科技股份有限公司 一种合成2,6-二乙基-4-甲基苯乙酸酯的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2736053B1 (fr) * 1995-06-28 1997-09-19 Sanofi Sa Nouvelles 1-phenylalkyl-1,2,3,6-tetrahydropyridines
ES2189877T3 (es) 1995-06-30 2003-07-16 Bayer Cropscience Ag Cetoenoles dialquil-halogenofenilsubstituidos para el empleo como herbicidas y pesticidas.
AU4614100A (en) * 1999-05-17 2000-12-05 Teijin Limited Cyanobiphenyl derivatives
DE10111262A1 (de) 2001-03-09 2002-09-12 Studiengesellschaft Kohle Mbh Verfahren zur Herstellung von Vinyl- Aryl- und Heteroarylessigsäuren und ihrer Devivate
WO2003009936A2 (en) * 2001-07-23 2003-02-06 Andrew Bruce Holmes Palladium-catalysed carbon-carbon bond forming reactions in compressed carbon dioxide

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
E. Paetzold,et al..Efficient two-phase Suzuki reaction catalyzed by palladium complexes with water-soluble phosphine ligands and detergents as phase transfer reagents.《Journal of Molecular Catalysis A: Chemical》.2000,第152卷69-76. *
Pd-catalyzed synthesis of arylacetic acid derivatives from boronic acids;Lukas J. Gooßen;《Chemical Communication》;20010321;669–670 *

Also Published As

Publication number Publication date
WO2011089072A1 (de) 2011-07-28
EP2526081B1 (de) 2015-07-01
CN102753513A (zh) 2012-10-24
ES2546487T3 (es) 2015-09-24
JP2013517255A (ja) 2013-05-16
EP2526081A1 (de) 2012-11-28
IL220787A (en) 2015-05-31
US20110184180A1 (en) 2011-07-28
JP5899119B2 (ja) 2016-04-06
KR20120116491A (ko) 2012-10-22
IN2012DN06383A (enExample) 2015-10-02
DK2526081T3 (en) 2015-10-05
KR101773070B1 (ko) 2017-09-12
US8507688B2 (en) 2013-08-13

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