KR101480279B1 - 피리딜 피페리딘 오렉신 수용체 길항제 - Google Patents

피리딜 피페리딘 오렉신 수용체 길항제 Download PDF

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KR101480279B1
KR101480279B1 KR1020097024362A KR20097024362A KR101480279B1 KR 101480279 B1 KR101480279 B1 KR 101480279B1 KR 1020097024362 A KR1020097024362 A KR 1020097024362A KR 20097024362 A KR20097024362 A KR 20097024362A KR 101480279 B1 KR101480279 B1 KR 101480279B1
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methyl
methoxy
pyridine
carbonyl
piperidin
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KR20100019984A (ko
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마이클 제이. 브레슬린
폴 제이. 콜먼
크리스토퍼 디. 콕스
존 디. 슈라이어
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머크 샤프 앤드 돔 코포레이션
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
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    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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KR1020097024362A 2007-05-23 2008-05-22 피리딜 피페리딘 오렉신 수용체 길항제 Expired - Fee Related KR101480279B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US93145807P 2007-05-23 2007-05-23
US60/931,458 2007-05-23
PCT/US2008/006563 WO2008147518A1 (en) 2007-05-23 2008-05-22 Pyridyl piperidine orexin receptor antagonists

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KR20100019984A KR20100019984A (ko) 2010-02-19
KR101480279B1 true KR101480279B1 (ko) 2015-01-09

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