KR101444486B1 - 인돌 화합물 - Google Patents

인돌 화합물 Download PDF

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Publication number
KR101444486B1
KR101444486B1 KR1020097010151A KR20097010151A KR101444486B1 KR 101444486 B1 KR101444486 B1 KR 101444486B1 KR 1020097010151 A KR1020097010151 A KR 1020097010151A KR 20097010151 A KR20097010151 A KR 20097010151A KR 101444486 B1 KR101444486 B1 KR 101444486B1
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KR
South Korea
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group
substituted
alkyl
compound
optionally substituted
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Expired - Fee Related
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KR1020097010151A
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English (en)
Korean (ko)
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KR20090068292A (ko
Inventor
츠네오 야스마
오사무 우지카와
마사히로 이토
가즈코 아오키
Original Assignee
다케다 야쿠힌 고교 가부시키가이샤
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Publication of KR20090068292A publication Critical patent/KR20090068292A/ko
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433—Thidiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1020097010151A 2006-10-19 2007-10-18 인돌 화합물 Expired - Fee Related KR101444486B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JPJP-P-2006-285551 2006-10-19
JP2006285551 2006-10-19
PCT/JP2007/070772 WO2008050821A1 (en) 2006-10-19 2007-10-18 Indole compound

Publications (2)

Publication Number Publication Date
KR20090068292A KR20090068292A (ko) 2009-06-25
KR101444486B1 true KR101444486B1 (ko) 2014-09-24

Family

ID=39010108

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020097010151A Expired - Fee Related KR101444486B1 (ko) 2006-10-19 2007-10-18 인돌 화합물

Country Status (26)

Country Link
US (4) US7652133B2 (enExample)
EP (2) EP2508524A3 (enExample)
JP (1) JP5260507B2 (enExample)
KR (1) KR101444486B1 (enExample)
CN (1) CN101573357B (enExample)
AU (1) AU2007310064B2 (enExample)
BR (1) BRPI0717722A2 (enExample)
CA (1) CA2666973C (enExample)
CL (1) CL2008001017A1 (enExample)
CR (1) CR10748A (enExample)
EC (1) ECSP099330A (enExample)
GE (1) GEP20115241B (enExample)
IL (1) IL198154A (enExample)
MA (1) MA30890B1 (enExample)
ME (1) MEP11809A (enExample)
MX (1) MX2009003972A (enExample)
MY (1) MY158052A (enExample)
NO (1) NO20091948L (enExample)
NZ (1) NZ576570A (enExample)
PE (1) PE20090884A1 (enExample)
RU (1) RU2454415C9 (enExample)
TN (1) TN2009000129A1 (enExample)
TW (1) TWI460176B (enExample)
UA (1) UA97257C2 (enExample)
WO (1) WO2008050821A1 (enExample)
ZA (1) ZA200902585B (enExample)

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