KR101386797B1 - 살진균 활성을 갖는 티에노-피리미딘 화합물 - Google Patents

살진균 활성을 갖는 티에노-피리미딘 화합물 Download PDF

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Publication number
KR101386797B1
KR101386797B1 KR1020077011335A KR20077011335A KR101386797B1 KR 101386797 B1 KR101386797 B1 KR 101386797B1 KR 1020077011335 A KR1020077011335 A KR 1020077011335A KR 20077011335 A KR20077011335 A KR 20077011335A KR 101386797 B1 KR101386797 B1 KR 101386797B1
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South Korea
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mmol
compound
solution
compounds
mixture
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Korean (ko)
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KR20070063602A (ko
Inventor
윌리암 커크랜드 브루스터
카를라 진 라스무센 클리티치
테리 윌리암 발코
네카 투에르 브록스
윌리암 란달 에릭슨
제임스 에드워드 헌터
크리스티안 토마스 로위
마이클 존 릭스
토마스 리만 시달
카를라 나네트 여케스
유안밍 쥬
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다우 아그로사이언시즈 엘엘씨
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
KR1020077011335A 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물 Expired - Fee Related KR101386797B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62157704P 2004-10-21 2004-10-21
US60/621,577 2004-10-21
PCT/US2005/038145 WO2006047397A1 (en) 2004-10-21 2005-10-21 Thieno-pyrimidine compounds having fungicidal activity

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020137034724A Division KR20140008471A (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물

Publications (2)

Publication Number Publication Date
KR20070063602A KR20070063602A (ko) 2007-06-19
KR101386797B1 true KR101386797B1 (ko) 2014-04-21

Family

ID=35722379

Family Applications (3)

Application Number Title Priority Date Filing Date
KR1020077011335A Expired - Fee Related KR101386797B1 (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물
KR1020147016709A Abandoned KR20140094626A (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물
KR1020137034724A Withdrawn KR20140008471A (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물

Family Applications After (2)

Application Number Title Priority Date Filing Date
KR1020147016709A Abandoned KR20140094626A (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물
KR1020137034724A Withdrawn KR20140008471A (ko) 2004-10-21 2005-10-21 살진균 활성을 갖는 티에노-피리미딘 화합물

Country Status (8)

Country Link
US (1) US8008487B2 (https=)
EP (1) EP1802632B1 (https=)
JP (2) JP5122293B2 (https=)
KR (3) KR101386797B1 (https=)
CN (1) CN101084224B (https=)
AT (1) ATE516291T1 (https=)
BR (1) BRPI0516242B1 (https=)
WO (1) WO2006047397A1 (https=)

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CN101084224B (zh) * 2004-10-21 2013-12-04 美国陶氏益农公司 具有杀真菌活性的噻吩并-嘧啶化合物
WO2007046809A1 (en) * 2005-10-21 2007-04-26 Dow Agrosciences Llc Thieno-pyrimidine compounds having fungicidal activity
MX2008013965A (es) 2006-05-22 2008-11-12 Basf Se Metodos insecticidas usando compuestos de 4-amino-5-cloro-tieno[2, 3-d]-pirimidina.
US8318384B2 (en) 2007-04-30 2012-11-27 The Governors Of The University Of Alberta Anode catalyst and methods of making and using the same
AU2009291783A1 (en) * 2008-09-10 2010-03-18 Alcon Research, Ltd Aminopyrimidine inhibitors of histamine receptors for the treatment of disease
US8586505B2 (en) 2009-07-16 2013-11-19 Sds Biotech K. K. 4-(3-butynyl)aminopyrimidine derivatives as pest control agents for agricultural and horticultural use
CN102596968B (zh) * 2009-07-30 2015-05-06 梅里亚有限公司 杀虫的4-氨基-噻吩并[2,3-d]-嘧啶化合物及其使用方法
NZ613449A (en) * 2011-01-14 2015-08-28 Sds Biotech Corp Agri-horticultural pest control compositions comprising 4-(3-butynyl)aminopyrimidine derivatives
ES2618813T3 (es) * 2011-06-27 2017-06-22 Merial, Inc. Compuestos y composiciones de éter amido-piridílico y uso contra los parásitos
MX2014000648A (es) 2011-07-19 2014-09-25 Infinity Pharmaceuticals Inc Compuestos heterociclicos y sus usos.
AR090037A1 (es) 2011-11-15 2014-10-15 Xention Ltd Derivados de tieno y/o furo-pirimidinas y piridinas inhibidores de los canales de potasio
CN105315296B (zh) * 2014-07-04 2018-04-03 沈阳中化农药化工研发有限公司 取代芳氧吡啶类化合物及其用途
CN104725398B (zh) * 2015-01-29 2017-01-18 杨威 一种jak/stat3磷酸化抑制剂及其制备方法与用途
CN109776427B (zh) * 2017-11-13 2022-08-23 沈阳中化农药化工研发有限公司 嘧啶双胺类化合物及其用途
WO2020180768A1 (en) * 2019-03-01 2020-09-10 Revolution Medicines, Inc. Bicyclic heteroaryl compounds and uses thereof
CN115626893B (zh) * 2022-10-10 2024-04-02 山西永津集团有限公司 一种2-羟基-5-羟甲基吡啶的合成方法

Citations (2)

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US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
EP0447891A1 (de) * 1990-03-19 1991-09-25 BASF Aktiengesellschaft Thieno[2,3-d]pyrimidinderivate

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GB2043061B (en) 1979-03-05 1983-05-11 Ici Ltd Thienopyrimidine and quinazoline derivatives
JPS5942387A (ja) * 1982-07-21 1984-03-08 Sankyo Co Ltd チエノピリミジン誘導体および殺虫、殺ダニ剤
DE3663945D1 (en) 1985-03-02 1989-07-20 Basf Ag Thiophene derivatives
JPS6267A (ja) * 1985-03-14 1987-01-06 Sankyo Co Ltd フエノキシアルキルアミン誘導体、その製法および殺虫殺ダニ剤
US5141941A (en) * 1988-11-21 1992-08-25 Ube Industries, Ltd. Aralkylamine derivatives, and fungicides containing the same
JPH075569B2 (ja) * 1989-08-02 1995-01-25 宇部興産株式会社 アラルキルアミン誘導体、その製法及び殺菌、殺虫剤
US5124333A (en) * 1989-08-02 1992-06-23 Ube Industries, Ltd. Aminopyrimidine derivatives and harmful organisms preventive agent
JPH0363265A (ja) * 1989-08-02 1991-03-19 Ube Ind Ltd アルキルアミノピリミジン誘導体、その製造法及び殺虫・殺ダニ・殺線虫剤
EP0424125A3 (en) 1989-10-18 1991-10-09 Ube Industries, Ltd. Aralkylamine derivatives, preparation method thereof and fungicides containing the same
BR9101256A (pt) * 1990-03-30 1991-11-05 Dowelanco Composto,composicao fungicida,processo fungicida,composicao inseticida ou acaricida e processo inseticida ou acaricida
US5137879A (en) * 1990-03-30 1992-08-11 Dowelanco Furopyrimidin-4-imine derivatives
JP2730019B2 (ja) * 1990-04-06 1998-03-25 宇部興産株式会社 アラルキルアミン誘導体，その製造法及び殺菌剤
JP2762430B2 (ja) 1991-01-18 1998-06-04 宇部興産株式会社 アラルキルアミノピリミジン類の製法
EP0519211A1 (de) * 1991-05-17 1992-12-23 Hoechst Schering AgrEvo GmbH Substituierte 4-Aminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel
JP3063266B2 (ja) 1991-08-30 2000-07-12 セイコーエプソン株式会社 液晶パネル及びその製造方法
JPH0710712A (ja) * 1993-06-25 1995-01-13 Ube Ind Ltd 花卉園芸用殺菌剤
US5679683A (en) * 1994-01-25 1997-10-21 Warner-Lambert Company Tricyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
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CA2333770A1 (en) * 1998-06-04 1999-12-09 Abbott Laboratories Cell adhesion-inhibiting antinflammatory compounds
US6232320B1 (en) * 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
JP2004509059A (ja) * 1999-06-03 2004-03-25 アボット・ラボラトリーズ 細胞接着抑制性抗炎症化合物
AU2002336462A1 (en) * 2001-09-06 2003-03-24 Millennium Pharmaceuticals, Inc. Piperazine and homopiperazine compounds
EP1463507A1 (en) 2001-12-19 2004-10-06 SmithKline Beecham Corporation Thienopyrimidine compounds as protein tyrosine kinase inhibitors
WO2004092123A2 (en) * 2003-04-10 2004-10-28 Microbia, Inc. Inhibitors of fungal invasion
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
PL1641803T6 (pl) * 2003-06-11 2011-04-29 Xention Ltd Pochodne tienopirymidyny jako inhibitory kanału potasowego
CN101084224B (zh) * 2004-10-21 2013-12-04 美国陶氏益农公司 具有杀真菌活性的噻吩并-嘧啶化合物

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
EP0447891A1 (de) * 1990-03-19 1991-09-25 BASF Aktiengesellschaft Thieno[2,3-d]pyrimidinderivate

Also Published As

Publication number Publication date
ATE516291T1 (de) 2011-07-15
JP2012180362A (ja) 2012-09-20
KR20140094626A (ko) 2014-07-30
HK1118534A1 (en) 2009-02-13
JP5122293B2 (ja) 2013-01-16
JP2008517936A (ja) 2008-05-29
WO2006047397A1 (en) 2006-05-04
CN101084224A (zh) 2007-12-05
BRPI0516242A (pt) 2008-08-26
US8008487B2 (en) 2011-08-30
BRPI0516242B1 (pt) 2014-10-07
KR20070063602A (ko) 2007-06-19
CN101084224B (zh) 2013-12-04
KR20140008471A (ko) 2014-01-21
JP5572664B2 (ja) 2014-08-13
US20060089370A1 (en) 2006-04-27
EP1802632B1 (en) 2011-07-13
EP1802632A1 (en) 2007-07-04

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