KR101300831B1 - 이미다조[1,2-ａ]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 - Google Patents

이미다조[1,2-ａ]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 Download PDF

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Publication number
KR101300831B1
KR101300831B1 KR1020077023609A KR20077023609A KR101300831B1 KR 101300831 B1 KR101300831 B1 KR 101300831B1 KR 1020077023609 A KR1020077023609 A KR 1020077023609A KR 20077023609 A KR20077023609 A KR 20077023609A KR 101300831 B1 KR101300831 B1 KR 101300831B1
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Prior art keywords
pyridin
imidazo
hydroxy
delete delete
acrylamide
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Korean (ko)
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KR20080005207A (ko
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켄 치 릭 리
에릭 티 선
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에스*바이오 피티이 리미티드
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Assigned to 메이 파마, 아이엔씨. reassignment 메이 파마, 아이엔씨. 권리의 전부이전등록 Assignors: 에스*바이오 피티이 리미티드
Assigned to 헬신 헬스케어 에스아 reassignment 헬신 헬스케어 에스아 권리의 전부이전등록 Assignors: 메이 파마, 아이엔씨.
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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KR1020077023609A 2005-03-21 2006-03-20 이미다조[1,2-ａ]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도 Expired - Fee Related KR101300831B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US66326505P 2005-03-21 2005-03-21
US60/663,265 2005-03-21
US75954406P 2006-01-18 2006-01-18
US60/759,544 2006-01-18
PCT/SG2006/000064 WO2006101455A1 (en) 2005-03-21 2006-03-20 Imidazo[1,2-a]pyridine derivatives: preparation and pharmaceutical applications

Publications (2)

Publication Number Publication Date
KR20080005207A KR20080005207A (ko) 2008-01-10
KR101300831B1 true KR101300831B1 (ko) 2013-08-30

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ID=37024054

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KR1020077023609A Expired - Fee Related KR101300831B1 (ko) 2005-03-21 2006-03-20 이미다조[1,2-ａ]피리딘 유도체, 이의 제조 방법 및 그의약학적 용도

Country Status (12)

Country Link
EP (1) EP1863811B1 (https=)
JP (1) JP5206405B2 (https=)
KR (1) KR101300831B1 (https=)
CN (1) CN101218238B (https=)
AR (1) AR056187A1 (https=)
AU (1) AU2006225355B2 (https=)
CA (1) CA2602328C (https=)
ES (1) ES2470766T3 (https=)
MX (1) MX2007011710A (https=)
MY (1) MY147647A (https=)
TW (1) TW200714600A (https=)
WO (1) WO2006101455A1 (https=)

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EP2601191A4 (en) * 2010-08-03 2013-07-31 Univ California COMPOUNDS AND COMPOSITIONS FOR MITIGATING WEB DAMAGE AND LETALITY
US9000186B2 (en) 2011-02-01 2015-04-07 Kyowa Hakko Kirin Co., Ltd. Ring-fused heterocyclic derivative
CA2831356A1 (en) * 2011-03-31 2012-10-04 Emblem Technology Transfer Gmbh Imidazo [1,2-a]pyridine_compounds for use in therapy
US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
CN104619707A (zh) 2012-07-31 2015-05-13 协和发酵麒麟株式会社 稠环杂环化合物
US9073921B2 (en) 2013-03-01 2015-07-07 Novartis Ag Salt forms of bicyclic heterocyclic derivatives
JP2016520047A (ja) * 2013-04-30 2016-07-11 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ ピラゾールアミドのＰｄ触媒カップリング
EP3004088A1 (en) * 2013-05-24 2016-04-13 Iomet Pharma Ltd. Slc2a transporter inhibitors
CA2913785C (en) * 2013-06-25 2021-08-31 F. Hoffmann-La Roche Ag Compounds for treating spinal muscular atrophy
EP3062783B1 (en) 2013-10-18 2020-08-12 The General Hospital Corporation Imaging histone deacetylases with a radiotracer using positron emission tomography
US10723705B2 (en) 2015-08-14 2020-07-28 Incyte Corporation Heterocyclic compounds and uses thereof
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JP5206405B2 (ja) 2013-06-12
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MY147647A (en) 2012-12-31
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