JP5206405B2 - イミダゾ［１，２−ａ］ピリジン誘導体：製造および医薬用途 - Google Patents

イミダゾ［１，２−ａ］ピリジン誘導体：製造および医薬用途 Download PDF

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JP5206405B2
JP5206405B2 JP2008502953A JP2008502953A JP5206405B2 JP 5206405 B2 JP5206405 B2 JP 5206405B2 JP 2008502953 A JP2008502953 A JP 2008502953A JP 2008502953 A JP2008502953 A JP 2008502953A JP 5206405 B2 JP5206405 B2 JP 5206405B2
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group
alkyl
aryl
optionally substituted
compound
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JP2008533198A5 (https=
JP2008533198A (ja
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リ，ケン・チ・リク
サン，エリック・ティー
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Lite Strategy Inc
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Mei Pharma Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
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    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
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  • Virology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biotechnology (AREA)
  • Transplantation (AREA)
  • Obesity (AREA)
JP2008502953A 2005-03-21 2006-03-20 イミダゾ［１，２−ａ］ピリジン誘導体：製造および医薬用途 Expired - Fee Related JP5206405B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US66326505P 2005-03-21 2005-03-21
US60/663,265 2005-03-21
US75954406P 2006-01-18 2006-01-18
US60/759,544 2006-01-18
PCT/SG2006/000064 WO2006101455A1 (en) 2005-03-21 2006-03-20 Imidazo[1,2-a]pyridine derivatives: preparation and pharmaceutical applications

Publications (3)

Publication Number Publication Date
JP2008533198A JP2008533198A (ja) 2008-08-21
JP2008533198A5 JP2008533198A5 (https=) 2009-05-07
JP5206405B2 true JP5206405B2 (ja) 2013-06-12

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JP2008502953A Expired - Fee Related JP5206405B2 (ja) 2005-03-21 2006-03-20 イミダゾ［１，２−ａ］ピリジン誘導体：製造および医薬用途

Country Status (12)

Country Link
EP (1) EP1863811B1 (https=)
JP (1) JP5206405B2 (https=)
KR (1) KR101300831B1 (https=)
CN (1) CN101218238B (https=)
AR (1) AR056187A1 (https=)
AU (1) AU2006225355B2 (https=)
CA (1) CA2602328C (https=)
ES (1) ES2470766T3 (https=)
MX (1) MX2007011710A (https=)
MY (1) MY147647A (https=)
TW (1) TW200714600A (https=)
WO (1) WO2006101455A1 (https=)

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WO2008068392A1 (fr) * 2006-12-07 2008-06-12 Commissariat A L'energie Atomique Nouveaux derives fluorophores imidazo [1,2-a] pyridin-3-yl-amine et leur procede de preparation
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DE102007040336A1 (de) 2007-08-27 2009-03-05 Johann Wolfgang Goethe-Universität Frankfurt am Main Neue Inhibitoren der 5-Lipoxygenase und deren Verwendungen
BRPI0817897A2 (pt) * 2007-11-02 2019-09-24 Methylgene Inc composto, composição, e, métodos de inibição da atividade hdac, e de tratamento de uma doença responsiva a um inibidor de atividade hdac
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WO2010032195A1 (en) 2008-09-16 2010-03-25 Csir Imidazopyridines and imidazopyrimidines as hiv-i reverse transcriptase inhibitors
US20110212943A1 (en) * 2008-10-15 2011-09-01 Orchid Research Laboratories Limited Novel bridged cyclic compounds as histone deacetylase inhibitors
EP2601191A4 (en) * 2010-08-03 2013-07-31 Univ California COMPOUNDS AND COMPOSITIONS FOR MITIGATING WEB DAMAGE AND LETALITY
US9000186B2 (en) 2011-02-01 2015-04-07 Kyowa Hakko Kirin Co., Ltd. Ring-fused heterocyclic derivative
CA2831356A1 (en) * 2011-03-31 2012-10-04 Emblem Technology Transfer Gmbh Imidazo [1,2-a]pyridine_compounds for use in therapy
US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
CN104619707A (zh) 2012-07-31 2015-05-13 协和发酵麒麟株式会社 稠环杂环化合物
US9073921B2 (en) 2013-03-01 2015-07-07 Novartis Ag Salt forms of bicyclic heterocyclic derivatives
JP2016520047A (ja) * 2013-04-30 2016-07-11 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ ピラゾールアミドのＰｄ触媒カップリング
EP3004088A1 (en) * 2013-05-24 2016-04-13 Iomet Pharma Ltd. Slc2a transporter inhibitors
CA2913785C (en) * 2013-06-25 2021-08-31 F. Hoffmann-La Roche Ag Compounds for treating spinal muscular atrophy
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US10723705B2 (en) 2015-08-14 2020-07-28 Incyte Corporation Heterocyclic compounds and uses thereof
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TW200714600A (en) 2007-04-16
AU2006225355B2 (en) 2010-12-09
MX2007011710A (es) 2007-11-20
CN101218238A (zh) 2008-07-09
EP1863811A4 (en) 2008-11-12
WO2006101455A1 (en) 2006-09-28
KR101300831B1 (ko) 2013-08-30
MY147647A (en) 2012-12-31
CA2602328A1 (en) 2006-09-28
CN101218238B (zh) 2011-10-26
JP2008533198A (ja) 2008-08-21
AU2006225355A1 (en) 2006-09-28
CA2602328C (en) 2014-07-29
ES2470766T3 (es) 2014-06-24
EP1863811B1 (en) 2014-03-12
KR20080005207A (ko) 2008-01-10
AR056187A1 (es) 2007-09-26
EP1863811A1 (en) 2007-12-12

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