KR101147672B1 - 경피 흡수 제제 - Google Patents

경피 흡수 제제 Download PDF

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Publication number
KR101147672B1
KR101147672B1 KR1020047019590A KR20047019590A KR101147672B1 KR 101147672 B1 KR101147672 B1 KR 101147672B1 KR 1020047019590 A KR1020047019590 A KR 1020047019590A KR 20047019590 A KR20047019590 A KR 20047019590A KR 101147672 B1 KR101147672 B1 KR 101147672B1
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KR
South Korea
Prior art keywords
propylene glycol
component
transdermal absorption
weight
drug
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1020047019590A
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English (en)
Korean (ko)
Other versions
KR20050024307A (ko
Inventor
나루이다카시
오미치가츠히로
오카다미노루
구라즈미도시아키
Original Assignee
히사미쓰 세이야꾸 가부시키가이샤
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication of KR20050024307A publication Critical patent/KR20050024307A/ko
Application granted granted Critical
Publication of KR101147672B1 publication Critical patent/KR101147672B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Anesthesiology (AREA)
  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020047019590A 2002-07-16 2003-07-02 경피 흡수 제제 Expired - Fee Related KR101147672B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JPJP-P-2002-00206565 2002-07-16
JP2002206565A JP4387639B2 (ja) 2002-07-16 2002-07-16 経皮吸収製剤
PCT/JP2003/008400 WO2004006960A1 (ja) 2002-07-16 2003-07-02 経皮吸収製剤

Publications (2)

Publication Number Publication Date
KR20050024307A KR20050024307A (ko) 2005-03-10
KR101147672B1 true KR101147672B1 (ko) 2012-05-21

Family

ID=30112800

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020047019590A Expired - Fee Related KR101147672B1 (ko) 2002-07-16 2003-07-02 경피 흡수 제제

Country Status (9)

Country Link
US (1) US20050255149A1 (enExample)
EP (1) EP1522316B1 (enExample)
JP (1) JP4387639B2 (enExample)
KR (1) KR101147672B1 (enExample)
CN (1) CN100341577C (enExample)
AU (1) AU2003244201A1 (enExample)
CA (1) CA2489188C (enExample)
TW (1) TW200403077A (enExample)
WO (1) WO2004006960A1 (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070166360A1 (en) * 2004-03-31 2007-07-19 Kowa Co., Ltd. External preparation
JP2005320282A (ja) * 2004-05-10 2005-11-17 Shiseido Co Ltd 局所麻酔用皮膚外用製剤
WO2007102243A1 (ja) 2006-03-08 2007-09-13 Nihon Nohyaku Co., Ltd. 外用の医薬組成物
BRPI0621386B8 (pt) 2006-03-08 2021-07-13 Nihon Nihyaku Co Ltd composição farmacêutica para o uso externo
PL2005958T3 (pl) 2006-03-08 2013-11-29 Nihon Nohyaku Co Ltd Kompozycja farmaceutyczna do stosowania zewnętrznego
HUE030028T2 (en) 2007-09-05 2017-04-28 Pola Pharma Inc Antifungal drug
KR20100075475A (ko) 2007-09-05 2010-07-02 가부시키가이샤 폴라 파마 의약 조성물
KR20100075476A (ko) * 2007-09-05 2010-07-02 가부시키가이샤 폴라 파마 항진균 조성물
CN102387785B (zh) 2009-04-09 2017-08-25 宝丽制药股份有限公司 抗真菌药物组合物
CN102387786B (zh) 2009-04-09 2015-09-09 宝丽制药股份有限公司 抗真菌药物组合物
US8952044B2 (en) 2009-08-25 2015-02-10 Pola Pharma Inc. Antimycotic pharmaceutical composition
JP5820207B2 (ja) * 2011-09-13 2015-11-24 日東電工株式会社 経皮吸収促進用組成物および貼付製剤
JP5820206B2 (ja) * 2011-09-13 2015-11-24 日東電工株式会社 経皮吸収促進用組成物および貼付製剤
JP5662495B2 (ja) * 2013-02-08 2015-01-28 株式会社ポーラファルマ 可溶化剤形の医薬組成物
NO2753788T3 (enExample) * 2013-05-10 2018-06-16
US9687455B2 (en) 2014-08-14 2017-06-27 John Daniel Dobak Sodium tetradecyl sulfate formulations for treatment of adipose tissue
US9351945B1 (en) 2015-02-27 2016-05-31 John Daniel Dobak, III Reduction of adipose tissue
CN108853312B (zh) * 2018-09-25 2021-04-16 陕西天宇制药有限公司 聚桂醇外用凝胶及其制备方法

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07285861A (ja) * 1994-04-20 1995-10-31 Dot:Kk 外用剤
JPH10182450A (ja) * 1996-12-27 1998-07-07 Ss Pharmaceut Co Ltd 外用組成物
US5932227A (en) * 1992-07-23 1999-08-03 Hisamitsu Pharmaceutical Co., Inc. Percutaneously administrable base composition and drug composition prepared therefrom

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5850964B2 (ja) * 1978-03-07 1983-11-14 東興薬品工業株式会社 ステロイド含有クリ−ム製剤およびその製造方法
JPS58225009A (ja) * 1982-06-23 1983-12-27 Shionogi & Co Ltd コルチコステロイド外用製剤
JPS62238216A (ja) * 1986-04-03 1987-10-19 Otsuka Pharmaceut Factory Inc ステロイドクリ−ム製剤
JP2860306B2 (ja) * 1989-12-26 1999-02-24 株式会社資生堂 皮膚外用製剤
JPH05178763A (ja) * 1991-02-19 1993-07-20 Nippon Saafuakutanto Kogyo Kk 難溶解性薬物溶解剤組成物
JP2986966B2 (ja) * 1991-06-26 1999-12-06 ポーラ化成工業株式会社 メラニン生成抑制剤
JPH06239740A (ja) * 1993-02-18 1994-08-30 Hiroshi Hibino ミコフェノール酸含有外用治療薬
US5858398A (en) * 1994-11-03 1999-01-12 Isomed Inc. Microparticular pharmaceutical compositions
AU5578096A (en) * 1995-04-28 1996-11-18 Pharmetrix, Inc. Compositions and methods for inducing dermal analgesia
JP4138910B2 (ja) * 1997-07-02 2008-08-27 帝國製薬株式会社 経皮吸収性が良好で且つ皮膚刺激性の少ない塩酸アゼラスチン含有経皮製剤
AU1689999A (en) * 1997-12-25 1999-07-19 Daiichi Pharmaceutical Co., Ltd. Medicinal composition for percutaneous administration
JP4275768B2 (ja) * 1998-06-18 2009-06-10 久光製薬株式会社 水性粘着膏体
US5994330A (en) * 1998-11-09 1999-11-30 El Khoury; Georges F. Topical application of muscarinic agents such as neostigmine for treatment of acne and other inflammatory conditions
JP2001026553A (ja) * 1999-07-09 2001-01-30 Lion Corp 外用剤組成物
GB0008785D0 (en) * 2000-04-10 2000-05-31 Novartis Ag Organic compounds
JP2003093152A (ja) * 2001-09-26 2003-04-02 Lion Corp 化粧料含浸シート

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5932227A (en) * 1992-07-23 1999-08-03 Hisamitsu Pharmaceutical Co., Inc. Percutaneously administrable base composition and drug composition prepared therefrom
JPH07285861A (ja) * 1994-04-20 1995-10-31 Dot:Kk 外用剤
JPH10182450A (ja) * 1996-12-27 1998-07-07 Ss Pharmaceut Co Ltd 外用組成物

Also Published As

Publication number Publication date
CA2489188C (en) 2011-11-15
WO2004006960A1 (ja) 2004-01-22
TW200403077A (en) 2004-03-01
KR20050024307A (ko) 2005-03-10
TWI314458B (enExample) 2009-09-11
JP4387639B2 (ja) 2009-12-16
EP1522316B1 (en) 2018-02-21
AU2003244201A1 (en) 2004-02-02
CN1668334A (zh) 2005-09-14
EP1522316A4 (en) 2011-02-23
JP2004051487A (ja) 2004-02-19
EP1522316A1 (en) 2005-04-13
US20050255149A1 (en) 2005-11-17
CN100341577C (zh) 2007-10-10
CA2489188A1 (en) 2004-01-22

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