KR100939890B1 - N-[1-(2-에톡시에틸)-5-(N-에틸-N-메틸아미노)-7-(4-메틸피리딘-2-일-아미노)-1H-피라졸로[4,3-d]피리미딘-3-카르보닐]메탄술폰아미드의 무수 결정 형태 - Google Patents

N-[1-(2-에톡시에틸)-5-(N-에틸-N-메틸아미노)-7-(4-메틸피리딘-2-일-아미노)-1H-피라졸로[4,3-d]피리미딘-3-카르보닐]메탄술폰아미드의 무수 결정 형태 Download PDF

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KR100939890B1
KR100939890B1 KR1020077026098A KR20077026098A KR100939890B1 KR 100939890 B1 KR100939890 B1 KR 100939890B1 KR 1020077026098 A KR1020077026098 A KR 1020077026098A KR 20077026098 A KR20077026098 A KR 20077026098A KR 100939890 B1 KR100939890 B1 KR 100939890B1
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amino
ethoxyethyl
pyrimidine
ethyl
methanesulfonamide
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KR20080004593A (ko
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데이비드 앤드류 앤트위슬
피터 발렌스 마샬
스테판 콜린 존 테일러
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화이자 인코포레이티드
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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KR1020077026098A 2005-05-12 2006-05-03 N-[1-(2-에톡시에틸)-5-(N-에틸-N-메틸아미노)-7-(4-메틸피리딘-2-일-아미노)-1H-피라졸로[4,3-d]피리미딘-3-카르보닐]메탄술폰아미드의 무수 결정 형태 Expired - Fee Related KR100939890B1 (ko)

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Application Number Priority Date Filing Date Title
US68044505P 2005-05-12 2005-05-12
US60/680,445 2005-05-12
US68171105P 2005-05-17 2005-05-17
US60/681,711 2005-05-17

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KR20080004593A KR20080004593A (ko) 2008-01-09
KR100939890B1 true KR100939890B1 (ko) 2010-01-29

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US8227475B2 (en) 2012-07-24
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