KR100618743B1 - 융합된 비사이클릭 또는 트리사이클릭 아미노산 - Google Patents

융합된 비사이클릭 또는 트리사이클릭 아미노산 Download PDF

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Publication number
KR100618743B1
KR100618743B1 KR1020037013691A KR20037013691A KR100618743B1 KR 100618743 B1 KR100618743 B1 KR 100618743B1 KR 1020037013691 A KR1020037013691 A KR 1020037013691A KR 20037013691 A KR20037013691 A KR 20037013691A KR 100618743 B1 KR100618743 B1 KR 100618743B1
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South Korea
Prior art keywords
bicyclo
acetic acid
aminomethyl
hept
pain
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KR1020037013691A
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English (en)
Korean (ko)
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KR20030092088A (ko
Inventor
블라케모어데이비드클리브
브라이언즈저스틴스티븐
윌리엄즈소피카롤린
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워너-램버트 캄파니 엘엘씨
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Priority claimed from GB0109635A external-priority patent/GB2374595A/en
Priority claimed from GB0125807A external-priority patent/GB0125807D0/en
Application filed by 워너-램버트 캄파니 엘엘씨 filed Critical 워너-램버트 캄파니 엘엘씨
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    • C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • C07C45/292—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups with chromium derivatives
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
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    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
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    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/69—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by addition to carbon-to-carbon double or triple bonds
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    • C07C49/423—Saturated compounds containing a keto group being part of a ring polycyclic a keto group being part of a condensed ring system
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    • C07C49/423—Saturated compounds containing a keto group being part of a ring polycyclic a keto group being part of a condensed ring system
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    • C07C2602/24—All rings being cycloaliphatic the ring system containing nine carbon atoms, e.g. perhydroindane
KR1020037013691A 2001-04-19 2002-04-03 융합된 비사이클릭 또는 트리사이클릭 아미노산 KR100618743B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0109635.3 2001-04-19
GB0109635A GB2374595A (en) 2001-04-19 2001-04-19 Fused bicyclic or tricyclic amino acids
GB0125807A GB0125807D0 (en) 2001-10-26 2001-10-26 Fused bicyclic or tricyclic amino acids
GB0125807.8 2001-10-26
PCT/IB2002/001146 WO2002085839A1 (fr) 2001-04-19 2002-04-03 Acides amnines bicycliques ou tricycliques fondus

Publications (2)

Publication Number Publication Date
KR20030092088A KR20030092088A (ko) 2003-12-03
KR100618743B1 true KR100618743B1 (ko) 2006-08-31

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Country Status (33)

Country Link
US (1) US6596900B2 (fr)
EP (1) EP1379494B1 (fr)
JP (1) JP4121858B2 (fr)
KR (1) KR100618743B1 (fr)
AP (1) AP2002002521A0 (fr)
AR (1) AR035861A1 (fr)
AT (1) ATE460392T1 (fr)
BG (1) BG108182A (fr)
BR (1) BR0208922A (fr)
CA (1) CA2444053C (fr)
CZ (1) CZ20032764A3 (fr)
DE (1) DE60235619D1 (fr)
EA (1) EA006396B1 (fr)
EE (1) EE200300517A (fr)
GE (1) GEP20053545B (fr)
HR (1) HRP20030832A2 (fr)
HU (1) HUP0303808A2 (fr)
IL (1) IL157932A0 (fr)
IS (1) IS6955A (fr)
MA (1) MA27015A1 (fr)
MX (1) MXPA03009532A (fr)
MY (1) MY134865A (fr)
NO (1) NO20034642L (fr)
NZ (1) NZ528151A (fr)
OA (1) OA12504A (fr)
PA (1) PA8543501A1 (fr)
PE (1) PE20021031A1 (fr)
PL (1) PL366406A1 (fr)
SK (1) SK12822003A3 (fr)
TN (1) TNSN03094A1 (fr)
TW (1) TWI262909B (fr)
WO (1) WO2002085839A1 (fr)
YU (1) YU78803A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20190046892A (ko) * 2016-09-14 2019-05-07 스촨 하이스코 파마수티컬 씨오., 엘티디 융합 트리사이클릭 γ-아미노산 유도체, 그 제조방법, 및 그것의 의료 용도

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