KR100309754B1 - 벤젠유도체및이를함유하는약제학적조성물 - Google Patents

벤젠유도체및이를함유하는약제학적조성물 Download PDF

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Publication number
KR100309754B1
KR100309754B1 KR1019970705095A KR19970705095A KR100309754B1 KR 100309754 B1 KR100309754 B1 KR 100309754B1 KR 1019970705095 A KR1019970705095 A KR 1019970705095A KR 19970705095 A KR19970705095 A KR 19970705095A KR 100309754 B1 KR100309754 B1 KR 100309754B1
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KR
South Korea
Prior art keywords
group
formula
methyl
hydrogen atom
compound
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Expired - Fee Related
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KR1019970705095A
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English (en)
Korean (ko)
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KR19980701699A (ko
Inventor
마사이치 하세가와
다쿠미 다케야스
나오키 쓰치야
나오키 하세
가쓰시 다카하시
다카시 가미무라
Original Assignee
야스이 쇼사꾸
데이진 가부시키가이샤
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Publication of KR19980701699A publication Critical patent/KR19980701699A/ko
Application granted granted Critical
Publication of KR100309754B1 publication Critical patent/KR100309754B1/ko
Anticipated expiration legal-status Critical
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/38—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019970705095A 1995-11-27 1996-11-26 벤젠유도체및이를함유하는약제학적조성물 Expired - Fee Related KR100309754B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP30722295 1995-11-27
JP95-307222 1995-11-27
JP22836796 1996-08-29
JP96-228367 1996-08-29
PCT/JP1996/003456 WO1997019910A1 (en) 1995-11-27 1996-11-26 Benzene derivatives

Publications (2)

Publication Number Publication Date
KR19980701699A KR19980701699A (ko) 1998-06-25
KR100309754B1 true KR100309754B1 (ko) 2002-05-30

Family

ID=26528211

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019970705095A Expired - Fee Related KR100309754B1 (ko) 1995-11-27 1996-11-26 벤젠유도체및이를함유하는약제학적조성물

Country Status (12)

Country Link
US (1) US5808144A (enExample)
EP (1) EP0806412B1 (enExample)
JP (1) JP3117466B2 (enExample)
KR (1) KR100309754B1 (enExample)
CN (1) CN1081623C (enExample)
AT (1) ATE191458T1 (enExample)
AU (1) AU703092B2 (enExample)
CA (1) CA2210579C (enExample)
DE (1) DE69607597T2 (enExample)
ES (1) ES2144786T3 (enExample)
TW (1) TW346483B (enExample)
WO (1) WO1997019910A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6649656B1 (en) * 1998-07-24 2003-11-18 Teijin Limited Anthranilic acid derivatives
US6627743B1 (en) * 1999-12-03 2003-09-30 Abbott Laboratories 6-O-methylerythromycin A crystal form III
AU2001234089B2 (en) * 2000-02-15 2005-08-11 Teijin Limited Cancer remedy comprising anthranilic acid derivative as active ingredient
GB0319124D0 (en) * 2003-08-14 2003-09-17 Smithkline Beecham Corp Chemical compounds
WO2020252195A1 (en) * 2019-06-11 2020-12-17 The Wistar Institute Of Anatomy And Biology Telomerase reverse transcriptase degraders and methods of use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE736787A (fr) * 1968-08-02 1970-01-30 Roussel Uclaf Dérivés de l'acide anthranilique et procédé de préparation
JPS60116657A (ja) * 1983-11-30 1985-06-24 Ono Pharmaceut Co Ltd アニリン誘導体
WO1993015043A1 (fr) 1992-01-24 1993-08-05 Yoshitomi Pharmaceutical Industries, Ltd. Compose arylalkananilide et utilisation pharmaceutique
US5783593A (en) * 1993-11-04 1998-07-21 Abbott Laboratories Inhibitors of squalene synthetase and protein farnesyltransferase

Also Published As

Publication number Publication date
ATE191458T1 (de) 2000-04-15
US5808144A (en) 1998-09-15
CN1081623C (zh) 2002-03-27
DE69607597T2 (de) 2000-08-24
AU7590296A (en) 1997-06-19
EP0806412B1 (en) 2000-04-05
EP0806412A1 (en) 1997-11-12
KR19980701699A (ko) 1998-06-25
CA2210579A1 (en) 1997-06-05
WO1997019910A1 (en) 1997-06-05
EP0806412A4 (enExample) 1997-11-12
CA2210579C (en) 2003-03-11
ES2144786T3 (es) 2000-06-16
CN1173169A (zh) 1998-02-11
TW346483B (en) 1998-12-01
JP3117466B2 (ja) 2000-12-11
AU703092B2 (en) 1999-03-18
DE69607597D1 (de) 2000-05-11

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