JPS61225181A - キノロンカルボン酸誘導体及びその製造方法 - Google Patents

キノロンカルボン酸誘導体及びその製造方法

Info

Publication number
JPS61225181A
JPS61225181A JP61022296A JP2229686A JPS61225181A JP S61225181 A JPS61225181 A JP S61225181A JP 61022296 A JP61022296 A JP 61022296A JP 2229686 A JP2229686 A JP 2229686A JP S61225181 A JPS61225181 A JP S61225181A
Authority
JP
Japan
Prior art keywords
formula
chloro
compound
bacteria
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP61022296A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0564955B2 (enrdf_load_stackoverflow
Inventor
Tsutomu Irikura
勉 入倉
Seigo Suzue
清吾 鈴江
Satoru Murayama
哲 村山
Keiji Hirai
敬二 平井
Takayoshi Ishizaki
孝義 石崎
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kyorin Pharmaceutical Co Ltd
Original Assignee
Kyorin Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Pharmaceutical Co Ltd filed Critical Kyorin Pharmaceutical Co Ltd
Priority to JP61022296A priority Critical patent/JPS61225181A/ja
Priority to AU54272/86A priority patent/AU5427286A/en
Priority to HU86888A priority patent/HUT40639A/hu
Priority to EP86102938A priority patent/EP0195316A1/en
Priority to FI860950A priority patent/FI85698C/fi
Priority to NO860870A priority patent/NO165071C/no
Priority to ES552802A priority patent/ES8704932A1/es
Priority to DK103986A priority patent/DK161383C/da
Priority to MX1780A priority patent/MX162668A/es
Priority to CN86102363A priority patent/CN1012613B/zh
Priority to PT82153A priority patent/PT82153B/pt
Priority to KR1019860001648A priority patent/KR930011036B1/ko
Publication of JPS61225181A publication Critical patent/JPS61225181A/ja
Publication of JPH0564955B2 publication Critical patent/JPH0564955B2/ja
Granted legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP61022296A 1985-03-08 1986-02-04 キノロンカルボン酸誘導体及びその製造方法 Granted JPS61225181A (ja)

Priority Applications (12)

Application Number Priority Date Filing Date Title
JP61022296A JPS61225181A (ja) 1986-02-04 1986-02-04 キノロンカルボン酸誘導体及びその製造方法
AU54272/86A AU5427286A (en) 1985-03-08 1986-03-04 7-(1-pyrrolidinyl)-3-quinolinecarboxylic acid derivatives
HU86888A HUT40639A (en) 1985-03-08 1986-03-04 Process for producing quinolon-carboxylic acid derivative and pharmaceutical composition containing them
EP86102938A EP0195316A1 (en) 1985-03-08 1986-03-06 Quinolonecarboxylic acid derivatives
FI860950A FI85698C (fi) 1985-03-08 1986-03-06 Foerfarande foer framstaellning av ett farmaceutiskt aktivt kinolonkarbonsyraderivat.
NO860870A NO165071C (no) 1985-03-08 1986-03-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive 7-(3-amino-1-pyrrolidinyl)-8-klor-1-cyklopropyl-6- fluor-1,4,-dihydro-4-okso-3-kinolin-karboksylsyre.
ES552802A ES8704932A1 (es) 1985-03-08 1986-03-07 Procedimiento para preparar un derivado de acido quinoloncarboxilico
DK103986A DK161383C (da) 1985-03-08 1986-03-07 Quinolincarboxylsyre-derivat, fremgangsmaade til fremstilling heraf samt antibakterielle farmaceutiske praeparater indeholdende dette
MX1780A MX162668A (es) 1985-03-08 1986-03-07 Procedimiento para preparar un derivado de acido quinoloncarboxilico
CN86102363A CN1012613B (zh) 1985-03-08 1986-03-07 喹诺酮羧酸衍生物的制备方法
PT82153A PT82153B (pt) 1985-03-08 1986-03-07 Processo para a preparacao de acido 7-(3-amino-1-pirrolidinil)-8-cloro-1-ciclopropil-6-fluor-1,4-dihidro-4-oxo-3-quinolino-carboxilico e seus hidratos e sais farmaceuticamente aceitaveis
KR1019860001648A KR930011036B1 (ko) 1985-03-08 1986-03-08 퀴놀론카복실산 유도체의 제조방법

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP61022296A JPS61225181A (ja) 1986-02-04 1986-02-04 キノロンカルボン酸誘導体及びその製造方法

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP60046216A Division JPS61205258A (ja) 1985-03-08 1985-03-08 キノロンカルボン酸誘導体及びその製造方法

Publications (2)

Publication Number Publication Date
JPS61225181A true JPS61225181A (ja) 1986-10-06
JPH0564955B2 JPH0564955B2 (enrdf_load_stackoverflow) 1993-09-16

Family

ID=12078778

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61022296A Granted JPS61225181A (ja) 1985-03-08 1986-02-04 キノロンカルボン酸誘導体及びその製造方法

Country Status (1)

Country Link
JP (1) JPS61225181A (enrdf_load_stackoverflow)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH01146880A (ja) * 1982-09-09 1989-06-08 Warner Lambert Co 抗菌性化合物
JP2001516756A (ja) * 1997-09-15 2001-10-02 ザ プロクター アンド ギャンブル カンパニー 抗微生物キノロン類、その組成物およびその使用
WO2010111116A1 (en) 2009-03-25 2010-09-30 Bausch & Lomb Incorporated Fluoroquinolone carboxylic acid molecular crystals
US8039485B2 (en) 2006-03-28 2011-10-18 Warner Chilcott Company, Llc Malate salts, and polymorphs of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
US8158798B2 (en) 2006-03-28 2012-04-17 Taigen Biotechnology Co., Ltd. Coupling process for preparing quinolone intermediates
US8518935B2 (en) 2009-12-11 2013-08-27 Bausch & Lomb Incorporated Amorphous besifloxacin solid

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS611667A (ja) * 1984-06-04 1986-01-07 バイエル・アクチエンゲゼルシヤフト ７‐アミノ‐１‐シクロプロピル‐６，８‐ジハロゲノ‐１，４‐ジヒドロ‐４‐オキソ‐３‐キノリンカルボン酸類、それらの製造方法およびそれらを含有する抗バクテリア剤

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS611667A (ja) * 1984-06-04 1986-01-07 バイエル・アクチエンゲゼルシヤフト ７‐アミノ‐１‐シクロプロピル‐６，８‐ジハロゲノ‐１，４‐ジヒドロ‐４‐オキソ‐３‐キノリンカルボン酸類、それらの製造方法およびそれらを含有する抗バクテリア剤

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH01146880A (ja) * 1982-09-09 1989-06-08 Warner Lambert Co 抗菌性化合物
JP2001516756A (ja) * 1997-09-15 2001-10-02 ザ プロクター アンド ギャンブル カンパニー 抗微生物キノロン類、その組成物およびその使用
US7868021B2 (en) 1997-09-15 2011-01-11 Warner Chilcott Company, Llc Antimicrobial quinolones, their compositions and uses
US8039485B2 (en) 2006-03-28 2011-10-18 Warner Chilcott Company, Llc Malate salts, and polymorphs of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
US8158798B2 (en) 2006-03-28 2012-04-17 Taigen Biotechnology Co., Ltd. Coupling process for preparing quinolone intermediates
WO2010111116A1 (en) 2009-03-25 2010-09-30 Bausch & Lomb Incorporated Fluoroquinolone carboxylic acid molecular crystals
US8481526B2 (en) 2009-03-25 2013-07-09 Bausch & Lomb Incorporated Fluoroquinolone carboxylic acid molecular crystals
US8518935B2 (en) 2009-12-11 2013-08-27 Bausch & Lomb Incorporated Amorphous besifloxacin solid

Also Published As

Publication number Publication date
JPH0564955B2 (enrdf_load_stackoverflow) 1993-09-16

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