JPS5839668A - １，５−ジフエニルピラゾリン−３−オン化合物、その製造法及び該化合物を含有する、抗アレルギ−作用を有する医薬品 - Google Patents
１，５−ジフエニルピラゾリン−３−オン化合物、その製造法及び該化合物を含有する、抗アレルギ−作用を有する医薬品Info
- Publication number
- JPS5839668A JPS5839668A JP57143479A JP14347982A JPS5839668A JP S5839668 A JPS5839668 A JP S5839668A JP 57143479 A JP57143479 A JP 57143479A JP 14347982 A JP14347982 A JP 14347982A JP S5839668 A JPS5839668 A JP S5839668A
- Authority
- JP
- Japan
- Prior art keywords
- group
- atom
- lower alkyl
- hydrogen atom
- alkyl group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Pulmonology (AREA)
- Animal Behavior & Ethology (AREA)
- Immunology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Detergent Compositions (AREA)
- Luminescent Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19813132915 DE3132915A1 (de) | 1981-08-20 | 1981-08-20 | 1,5-diphenylpyrazolin-3-on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| DE3132915.2 | 1981-08-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5839668A true JPS5839668A (ja) | 1983-03-08 |
| JPH0375542B2 JPH0375542B2 (US20100223739A1-20100909-C00005.png) | 1991-12-02 |
Family
ID=6139713
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP57143479A Granted JPS5839668A (ja) | 1981-08-20 | 1982-08-20 | １，５−ジフエニルピラゾリン−３−オン化合物、その製造法及び該化合物を含有する、抗アレルギ−作用を有する医薬品 |
Country Status (20)
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3442860A1 (de) * | 1984-11-24 | 1986-05-28 | Kali-Chemie Pharma Gmbh, 3000 Hannover | 5-alkyl-1-phenyl-2-piperazinoalkylpyrazolin-3- on-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| NZ524193A (en) * | 2000-08-14 | 2004-12-24 | Ortho Mcneil Pharm Inc | Substituted pyrazoles |
| CA2488202C (en) * | 2002-06-12 | 2011-03-08 | Chemocentryx, Inc. | 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders |
| US20050256130A1 (en) * | 2002-06-12 | 2005-11-17 | Chemocentryx, Inc. | Substituted piperazines |
| US7842693B2 (en) * | 2002-06-12 | 2010-11-30 | Chemocentryx, Inc. | Substituted piperazines |
| US7589199B2 (en) * | 2002-06-12 | 2009-09-15 | Chemocentryx, Inc. | Substituted piperazines |
| EP1720545B1 (en) * | 2004-03-03 | 2014-10-29 | ChemoCentryx, Inc. | Bicyclic and bridged nitrogen heterocycles |
| US7435831B2 (en) * | 2004-03-03 | 2008-10-14 | Chemocentryx, Inc. | Bicyclic and bridged nitrogen heterocycles |
| WO2011051958A1 (en) * | 2009-10-30 | 2011-05-05 | E.I. Du Pont De Nemours And Company | Fungicidal pyrazolones |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE74912C (US20100223739A1-20100909-C00005.png) * | ||||
| DE66610C (de) * | FARBWERKE VORM. MEISTER LUCIUS & BRÜNING in Höchst a. M | Verfahren zur Darstellung von Oxaethylmethylphenylpyrazolon | ||
| GB666578A (en) * | 1948-01-10 | 1952-02-13 | Luxema | Process for the preparation of derivatives of 1, 2, 3 substituted pyrazolones and derivatives obtained by this process |
| US3169966A (en) * | 1961-01-24 | 1965-02-16 | Ciba Geigy Corp | Aminopyrazoles |
| DE2824764A1 (de) * | 1978-06-06 | 1979-12-20 | Hoechst Ag | Neue pyridylpiperazinderivate und verfahren zu ihrer herstellung |
| DE2828529A1 (de) * | 1978-06-29 | 1980-01-17 | Kali Chemie Pharma Gmbh | Neue 5-phenylpyrazol-derivate, verfahren zu deren herstellung und arzneimittel |
-
1981
- 1981-08-20 DE DE19813132915 patent/DE3132915A1/de not_active Withdrawn
-
1982
- 1982-07-27 ZA ZA825381A patent/ZA825381B/xx unknown
- 1982-07-30 PT PT75353A patent/PT75353B/pt not_active IP Right Cessation
- 1982-08-09 AT AT82107193T patent/ATE43841T1/de not_active IP Right Cessation
- 1982-08-09 DE DE8282107193T patent/DE3279756D1/de not_active Expired
- 1982-08-09 EP EP82107193A patent/EP0072960B1/de not_active Expired
- 1982-08-10 CA CA000409072A patent/CA1208643A/en not_active Expired
- 1982-08-17 DD DD82242578A patent/DD202563A5/de unknown
- 1982-08-18 HU HU822675A patent/HU187572B/hu not_active IP Right Cessation
- 1982-08-18 GR GR69057A patent/GR76272B/el unknown
- 1982-08-18 PH PH27741A patent/PH19107A/en unknown
- 1982-08-18 GR GR69059A patent/GR78228B/el unknown
- 1982-08-19 ES ES515107A patent/ES8306143A1/es not_active Expired
- 1982-08-19 NZ NZ201643A patent/NZ201643A/xx unknown
- 1982-08-19 DK DK372382A patent/DK149947C/da not_active IP Right Cessation
- 1982-08-19 FI FI822883A patent/FI73673C/fi not_active IP Right Cessation
- 1982-08-19 AU AU87424/82A patent/AU555215B2/en not_active Ceased
- 1982-08-19 US US06/409,631 patent/US4442102A/en not_active Expired - Fee Related
- 1982-08-19 IE IE2002/82A patent/IE55377B1/en unknown
- 1982-08-19 IL IL66580A patent/IL66580A/xx unknown
- 1982-08-19 NO NO822827A patent/NO158185C/no unknown
- 1982-08-20 JP JP57143479A patent/JPS5839668A/ja active Granted
-
1983
- 1983-12-22 US US06/564,399 patent/US4515944A/en not_active Expired - Fee Related
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