JPS5826758B2 - チエノチアジンユウドウタイノセイゾウホウホウ - Google Patents

チエノチアジンユウドウタイノセイゾウホウホウ

Info

Publication number
JPS5826758B2
JPS5826758B2 JP50102635A JP10263575A JPS5826758B2 JP S5826758 B2 JPS5826758 B2 JP S5826758B2 JP 50102635 A JP50102635 A JP 50102635A JP 10263575 A JP10263575 A JP 10263575A JP S5826758 B2 JPS5826758 B2 JP S5826758B2
Authority
JP
Japan
Prior art keywords
methyl
group
pyridyl
lower alkyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP50102635A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5148694A (OSRAM
Inventor
ホロマトカ オツトー
ビンダー デイーター
ツエラー パウル
フイスター ルドルフ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1158274A external-priority patent/CH608500A5/de
Priority claimed from CH1215774A external-priority patent/CH608501A5/de
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of JPS5148694A publication Critical patent/JPS5148694A/ja
Publication of JPS5826758B2 publication Critical patent/JPS5826758B2/ja
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/34—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Electroplating Methods And Accessories (AREA)
  • Manufacturing Of Printed Wiring (AREA)
JP50102635A 1974-08-26 1975-08-26 チエノチアジンユウドウタイノセイゾウホウホウ Expired JPS5826758B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1158274A CH608500A5 (en) 1974-08-26 1974-08-26 Process for the preparation of thiazine derivatives
CH1215774A CH608501A5 (en) 1974-09-09 1974-09-09 Process for the preparation of thiazine derivatives

Publications (2)

Publication Number Publication Date
JPS5148694A JPS5148694A (OSRAM) 1976-04-26
JPS5826758B2 true JPS5826758B2 (ja) 1983-06-04

Family

ID=25708582

Family Applications (1)

Application Number Title Priority Date Filing Date
JP50102635A Expired JPS5826758B2 (ja) 1974-08-26 1975-08-26 チエノチアジンユウドウタイノセイゾウホウホウ

Country Status (20)

Country Link
JP (1) JPS5826758B2 (OSRAM)
AR (1) AR216288A1 (OSRAM)
AT (1) AT350064B (OSRAM)
BR (1) BR7505463A (OSRAM)
DD (1) DD124119A5 (OSRAM)
DE (1) DE2537070A1 (OSRAM)
DK (1) DK137835B (OSRAM)
FI (1) FI59253C (OSRAM)
FR (3) FR2282893A1 (OSRAM)
GB (1) GB1519811A (OSRAM)
HU (1) HU173739B (OSRAM)
IE (1) IE41457B1 (OSRAM)
IL (1) IL47877A (OSRAM)
LU (2) LU73257A1 (OSRAM)
NL (2) NL183582C (OSRAM)
NO (1) NO146096C (OSRAM)
PL (1) PL106076B1 (OSRAM)
SE (1) SE412066B (OSRAM)
SU (1) SU603338A3 (OSRAM)
YU (1) YU40266B (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2704485A1 (de) * 1977-02-03 1978-08-10 Thomae Gmbh Dr K Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
LU78009A1 (de) 1977-08-22 1979-05-23 Hoffmann La Roche Verfahren zur herstellung von thiazinderivaten
ZA784958B (en) * 1977-09-06 1979-08-29 Hoffmann La Roche Thiazine derivatives
AU518216B2 (en) 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
DE2838377A1 (de) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung
AU5811280A (en) * 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
JPS58109492A (ja) * 1981-12-22 1983-06-29 Mitsui Toatsu Chem Inc チエノチアジン誘導体およびそれを含有する医薬組成物
DE3371082D1 (de) * 1982-09-09 1987-05-27 Hoffmann La Roche Thieno(2,3-e)-1,2-thiazine derivatives
ATA39088A (de) 1988-02-18 1990-06-15 Binder Dieter Dr Basisch substituierte thienoisothiazol-3(2h)-on-1,1-dioxide und ihre pharmazeutisch vertraeglichen salze, verfahren zu ihrer herstellung und ihre verwendung
AT400437B (de) * 1993-12-14 1995-12-27 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
AT400568B (de) * 1994-05-18 1996-01-25 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
EP0658559A1 (de) * 1993-12-14 1995-06-21 Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. Thienothiazinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als 5-dipoxygenase und Cyclooxygenaseinhibitoren
US5538966A (en) * 1994-01-21 1996-07-23 Alcon Laboratories, Inc. Carbonic anhydrase inhibitors
IT1308633B1 (it) 1999-03-02 2002-01-09 Nicox Sa Nitrossiderivati.
CN1171892C (zh) * 2001-06-25 2004-10-20 李晶 具有抗炎镇痛活性的噻吩并噻嗪化合物及其制备方法和用途

Also Published As

Publication number Publication date
IE41457B1 (en) 1980-01-02
AT350064B (de) 1979-05-10
DE2537070A1 (de) 1976-03-18
FR2303803A1 (fr) 1976-10-08
FR2282893A1 (fr) 1976-03-26
LU73257A1 (OSRAM) 1977-04-15
NL930080I2 (nl) 1994-01-03
YU216675A (en) 1982-08-31
DE2537070C2 (OSRAM) 1987-06-25
NO146096C (no) 1982-07-28
AR216288A1 (es) 1979-12-14
NL183582C (nl) 1988-12-01
LU88312I2 (de) 1994-09-09
NL7510057A (nl) 1976-03-01
NL930080I1 (nl) 1993-09-16
IL47877A (en) 1978-10-31
ATA655975A (de) 1978-10-15
FI59253B (fi) 1981-03-31
NO146096B (no) 1982-04-19
FR2309558B1 (OSRAM) 1979-05-04
DK137835B (da) 1978-05-16
NO752932L (OSRAM) 1976-02-27
FI752398A7 (OSRAM) 1976-02-27
GB1519811A (en) 1978-08-02
SE7509446L (sv) 1976-02-27
IL47877A0 (en) 1975-11-25
HU173739B (hu) 1979-08-28
NL183582B (nl) 1988-07-01
DK381175A (OSRAM) 1976-02-27
AU8418675A (en) 1977-02-24
JPS5148694A (OSRAM) 1976-04-26
YU40266B (en) 1985-12-31
PL106076B1 (pl) 1979-11-30
DD124119A5 (OSRAM) 1977-02-02
IE41457L (en) 1976-02-26
SE412066B (sv) 1980-02-18
FR2303803B1 (OSRAM) 1979-07-13
FR2309558A1 (fr) 1976-11-26
DK137835C (OSRAM) 1978-10-16
BR7505463A (pt) 1976-08-03
FR2282893B1 (OSRAM) 1980-05-16
SU603338A3 (ru) 1978-04-15
FI59253C (fi) 1981-07-10

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