JP7397070B2 - フルエンスルホンの製造のための方法及び中間体 - Google Patents
フルエンスルホンの製造のための方法及び中間体 Download PDFInfo
- Publication number
- JP7397070B2 JP7397070B2 JP2021517567A JP2021517567A JP7397070B2 JP 7397070 B2 JP7397070 B2 JP 7397070B2 JP 2021517567 A JP2021517567 A JP 2021517567A JP 2021517567 A JP2021517567 A JP 2021517567A JP 7397070 B2 JP7397070 B2 JP 7397070B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- reaction
- cfx
- organic solvent
- mercaptothiazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862736498P | 2018-09-26 | 2018-09-26 | |
| US62/736,498 | 2018-09-26 | ||
| PCT/IL2019/051063 WO2020065652A1 (en) | 2018-09-26 | 2019-09-26 | Process and intermediates for the preparation of fluensulfone |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022503882A JP2022503882A (ja) | 2022-01-12 |
| JP2022503882A5 JP2022503882A5 (https=) | 2023-02-07 |
| JP7397070B2 true JP7397070B2 (ja) | 2023-12-12 |
Family
ID=68387378
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021517567A Active JP7397070B2 (ja) | 2018-09-26 | 2019-09-26 | フルエンスルホンの製造のための方法及び中間体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US11634397B2 (https=) |
| JP (1) | JP7397070B2 (https=) |
| KR (1) | KR102608979B1 (https=) |
| CN (1) | CN112930342B (https=) |
| AR (1) | AR116506A1 (https=) |
| AU (1) | AU2019346158B2 (https=) |
| PY (1) | PY1980072A (https=) |
| WO (1) | WO2020065652A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN114805240B (zh) * | 2022-06-28 | 2022-09-16 | 湖南速博生物技术有限公司 | 一种一锅法合成氟烯线砜的方法 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005525418A (ja) | 2002-05-13 | 2005-08-25 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | 置換トリフルオロエチレンの製造方法 |
| JP2011063599A (ja) | 2002-07-03 | 2011-03-31 | Makhteshim Chemical Works Ltd | ヘテロ環式フルオロアルケニルスルホンの製造方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2603647A (en) | 1951-10-18 | 1952-07-15 | Goodrich Co B F | Preparation of 2-mercapto thiazoles |
| US2603648A (en) | 1951-10-18 | 1952-07-15 | Goodrich Co B F | Preparation of 2-mercapto thiazoles |
| EP0228447A4 (en) | 1985-06-20 | 1990-12-27 | Fmc Corporation | Pesticidal polyhaloalkene derivatives |
| IL112721A0 (en) * | 1994-03-10 | 1995-05-26 | Zeneca Ltd | Azole derivatives |
| GB9708280D0 (en) | 1997-04-24 | 1997-06-18 | Zeneca Ltd | Novel process |
| JP3899626B2 (ja) | 1997-12-26 | 2007-03-28 | 宇部興産株式会社 | ２−メルカプトチアゾ−ルの製法 |
| JP2001019685A (ja) | 1999-07-06 | 2001-01-23 | Nippon Bayer Agrochem Co Ltd | 殺センチュウ性トリフルオロブテン類 |
| JP2003113168A (ja) | 2001-09-28 | 2003-04-18 | Bayer Ag | 殺センチュウ性トリフルオロブテン誘導体 |
| DE10221120A1 (de) | 2002-05-13 | 2003-11-27 | Bayer Cropscience Ag | Verfahren zur Herstellung von substituierten Trifluorethylenen |
| CN111670180A (zh) * | 2017-12-20 | 2020-09-15 | Pi工业有限公司 | 氟烯基化合物，制备方法及其用途 |
-
2019
- 2019-09-25 PY PY201901980072A patent/PY1980072A/es unknown
- 2019-09-25 AR ARP190102726A patent/AR116506A1/es unknown
- 2019-09-26 KR KR1020217011965A patent/KR102608979B1/ko active Active
- 2019-09-26 CN CN201980069064.8A patent/CN112930342B/zh active Active
- 2019-09-26 US US17/280,146 patent/US11634397B2/en active Active
- 2019-09-26 JP JP2021517567A patent/JP7397070B2/ja active Active
- 2019-09-26 WO PCT/IL2019/051063 patent/WO2020065652A1/en not_active Ceased
- 2019-09-26 AU AU2019346158A patent/AU2019346158B2/en active Active
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005525418A (ja) | 2002-05-13 | 2005-08-25 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | 置換トリフルオロエチレンの製造方法 |
| JP2011063599A (ja) | 2002-07-03 | 2011-03-31 | Makhteshim Chemical Works Ltd | ヘテロ環式フルオロアルケニルスルホンの製造方法 |
Non-Patent Citations (1)
| Title |
|---|
| LI, G et al.，Fluoroalkane thioheterocyclic derivatives and their antitumor activity，European Journal of Medicinal Chemistry，2015年02月20日，Vol. 93，pp. 423-430 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2022503882A (ja) | 2022-01-12 |
| US11634397B2 (en) | 2023-04-25 |
| US20220002258A1 (en) | 2022-01-06 |
| CN112930342A (zh) | 2021-06-08 |
| AR116506A1 (es) | 2021-05-12 |
| AU2019346158A1 (en) | 2021-05-06 |
| PY1980072A (es) | 2020-06-05 |
| CN112930342B (zh) | 2024-10-11 |
| BR112021005745A2 (pt) | 2021-07-27 |
| WO2020065652A1 (en) | 2020-04-02 |
| KR102608979B1 (ko) | 2023-11-30 |
| KR20210072010A (ko) | 2021-06-16 |
| AU2019346158B2 (en) | 2025-01-30 |
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