AU2019346158B2 - Process and intermediates for the preparation of fluensulfone - Google Patents

Process and intermediates for the preparation of fluensulfone Download PDF

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Publication number
AU2019346158B2
AU2019346158B2 AU2019346158A AU2019346158A AU2019346158B2 AU 2019346158 B2 AU2019346158 B2 AU 2019346158B2 AU 2019346158 A AU2019346158 A AU 2019346158A AU 2019346158 A AU2019346158 A AU 2019346158A AU 2019346158 B2 AU2019346158 B2 AU 2019346158B2
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formula
process according
cfx
reaction
solution
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AU2019346158A
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AU2019346158A1 (en
Inventor
Shlomi Cohen
Thomas Zell
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/36Sulfur atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AU2019346158A 2018-09-26 2019-09-26 Process and intermediates for the preparation of fluensulfone Active AU2019346158B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862736498P 2018-09-26 2018-09-26
US62/736,498 2018-09-26
PCT/IL2019/051063 WO2020065652A1 (en) 2018-09-26 2019-09-26 Process and intermediates for the preparation of fluensulfone

Publications (2)

Publication Number Publication Date
AU2019346158A1 AU2019346158A1 (en) 2021-05-06
AU2019346158B2 true AU2019346158B2 (en) 2025-01-30

Family

ID=68387378

Family Applications (1)

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AU2019346158A Active AU2019346158B2 (en) 2018-09-26 2019-09-26 Process and intermediates for the preparation of fluensulfone

Country Status (8)

Country Link
US (1) US11634397B2 (https=)
JP (1) JP7397070B2 (https=)
KR (1) KR102608979B1 (https=)
CN (1) CN112930342B (https=)
AR (1) AR116506A1 (https=)
AU (1) AU2019346158B2 (https=)
PY (1) PY1980072A (https=)
WO (1) WO2020065652A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114805240B (zh) * 2022-06-28 2022-09-16 湖南速博生物技术有限公司 一种一锅法合成氟烯线砜的方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998047884A1 (en) * 1997-04-24 1998-10-29 Zeneca Limited Process for the production of 5-chloro-2- (4,4-difluorobut-3-enylsulphonyl) thiazole and intermediates therefor
WO2003095401A1 (de) * 2002-05-13 2003-11-20 Bayer Cropscience Aktiengesellschaft Verfahren zur herstellung von substituierten trifluorethylenen

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2603647A (en) 1951-10-18 1952-07-15 Goodrich Co B F Preparation of 2-mercapto thiazoles
US2603648A (en) 1951-10-18 1952-07-15 Goodrich Co B F Preparation of 2-mercapto thiazoles
EP0228447A4 (en) 1985-06-20 1990-12-27 Fmc Corporation Pesticidal polyhaloalkene derivatives
IL112721A0 (en) * 1994-03-10 1995-05-26 Zeneca Ltd Azole derivatives
JP3899626B2 (ja) 1997-12-26 2007-03-28 宇部興産株式会社 2−メルカプトチアゾ−ルの製法
JP2001019685A (ja) 1999-07-06 2001-01-23 Nippon Bayer Agrochem Co Ltd 殺センチュウ性トリフルオロブテン類
JP2003113168A (ja) 2001-09-28 2003-04-18 Bayer Ag 殺センチュウ性トリフルオロブテン誘導体
DE10221119A1 (de) 2002-05-13 2003-12-04 Bayer Cropscience Ag Verfahren zur Herstellung von substituierten Trifluorethylenen
DE10229776A1 (de) 2002-07-03 2004-01-22 Bayer Cropscience Ag Verfahren zum Herstellen von heterocyclischen Fluoralkenylsulfonen
CN111670180A (zh) * 2017-12-20 2020-09-15 Pi工业有限公司 氟烯基化合物,制备方法及其用途

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998047884A1 (en) * 1997-04-24 1998-10-29 Zeneca Limited Process for the production of 5-chloro-2- (4,4-difluorobut-3-enylsulphonyl) thiazole and intermediates therefor
WO2003095401A1 (de) * 2002-05-13 2003-11-20 Bayer Cropscience Aktiengesellschaft Verfahren zur herstellung von substituierten trifluorethylenen

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
LI GUANGXIAO ET AL: "Fluoroalkane thioheterocyclic derivatives and their antitumor activity", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, ELSEVIER, AMSTERDAM, NL, vol. 93, 20 February 2015, pages 423 - 430, DOI: 10.1016/J.EJMECH.2015.02.031 *

Also Published As

Publication number Publication date
JP2022503882A (ja) 2022-01-12
US11634397B2 (en) 2023-04-25
US20220002258A1 (en) 2022-01-06
JP7397070B2 (ja) 2023-12-12
CN112930342A (zh) 2021-06-08
AR116506A1 (es) 2021-05-12
AU2019346158A1 (en) 2021-05-06
PY1980072A (es) 2020-06-05
CN112930342B (zh) 2024-10-11
BR112021005745A2 (pt) 2021-07-27
WO2020065652A1 (en) 2020-04-02
KR102608979B1 (ko) 2023-11-30
KR20210072010A (ko) 2021-06-16

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