JP7014736B2 - がんの処置のためのピラゾロピリジン誘導体 - Google Patents

がんの処置のためのピラゾロピリジン誘導体 Download PDF

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JP7014736B2
JP7014736B2 JP2018561557A JP2018561557A JP7014736B2 JP 7014736 B2 JP7014736 B2 JP 7014736B2 JP 2018561557 A JP2018561557 A JP 2018561557A JP 2018561557 A JP2018561557 A JP 2018561557A JP 7014736 B2 JP7014736 B2 JP 7014736B2
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mmol
compound
salt
pharmaceutically acceptable
mixture
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JP2019516759A (ja
JP2019516759A5 (https=
Inventor
パトリック シール，
サラ ブロナー，
エフ． アントニー ロメロ，
スティーブン マグヌソン，
ビッキー シャオ－ウェイ ツイ，
ジェレミー エム． マレー，
ジョン ワイ，
クォン ワー ライ，
フェイ ワン，
ケビン エックス． チェン，
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Constellation Pharmaceuticals Inc
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Constellation Pharmaceuticals Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
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  • Psychiatry (AREA)
  • Obesity (AREA)
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  • Transplantation (AREA)
  • Toxicology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
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JP2018561557A 2016-05-24 2017-05-24 がんの処置のためのピラゾロピリジン誘導体 Expired - Fee Related JP7014736B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2016083118 2016-05-24
CNPCT/CN2016/083118 2016-05-24
PCT/US2017/034326 WO2017205538A1 (en) 2016-05-24 2017-05-24 Pyrazolopyridine derivatives for the treatment of cancer

Publications (3)

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JP2019516759A JP2019516759A (ja) 2019-06-20
JP2019516759A5 JP2019516759A5 (https=) 2020-07-02
JP7014736B2 true JP7014736B2 (ja) 2022-02-01

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JP2018561557A Expired - Fee Related JP7014736B2 (ja) 2016-05-24 2017-05-24 がんの処置のためのピラゾロピリジン誘導体

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US (2) US11247989B2 (https=)
EP (1) EP3464286B1 (https=)
JP (1) JP7014736B2 (https=)
CN (1) CN109476663B (https=)
MA (1) MA45146A (https=)
WO (1) WO2017205538A1 (https=)

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