JP6775516B2 - 新奇な３−インドール置換誘導体、医薬組成物、および使用方法 - Google Patents

新奇な３−インドール置換誘導体、医薬組成物、および使用方法 Download PDF

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JP6775516B2
JP6775516B2 JP2017548261A JP2017548261A JP6775516B2 JP 6775516 B2 JP6775516 B2 JP 6775516B2 JP 2017548261 A JP2017548261 A JP 2017548261A JP 2017548261 A JP2017548261 A JP 2017548261A JP 6775516 B2 JP6775516 B2 JP 6775516B2
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isothiazole
fluoro
indole
methyl
dioxide
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JP2018511587A (ja
JP2018511587A5 (https=
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ニンコヴィッチ サッシャ
ニンコヴィッチ サッシャ
クロシグナニ ステファノ
クロシグナニ ステファノ
アン スケイルズ ステファニー
アン スケイルズ ステファニー
ジェームズ マケルピン インドラワン
ジェームズ マケルピン インドラワン
レイモンド コリンズ マイケル
レイモンド コリンズ マイケル
マデルナ アンドレアス
マデルナ アンドレアス
ワイセス マーティン
ワイセス マーティン
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ファイザー・インク
アイティーオス セラペウティクス
アイティーオス セラペウティクス
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Gastroenterology & Hepatology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2017548261A 2015-03-17 2016-03-17 新奇な３−インドール置換誘導体、医薬組成物、および使用方法 Expired - Fee Related JP6775516B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
PCT/IB2015/051957 WO2015140717A1 (en) 2014-03-18 2015-03-17 Novel 3-indol substituted derivatives, pharmaceutical compositions and methods for use
IBPCT/IB2015/051957 2015-03-17
US201562203032P 2015-08-10 2015-08-10
US62/203,032 2015-08-10
PCT/IB2016/051509 WO2016147144A1 (en) 2015-03-17 2016-03-17 Novel 3-indol substituted derivatives, pharmaceutical compositions and methods for use

Publications (3)

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JP2018511587A JP2018511587A (ja) 2018-04-26
JP2018511587A5 JP2018511587A5 (https=) 2019-04-25
JP6775516B2 true JP6775516B2 (ja) 2020-10-28

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US (1) US9873690B2 (https=)
EP (1) EP3271354A1 (https=)
JP (1) JP6775516B2 (https=)
KR (1) KR102013512B1 (https=)
CN (1) CN107635990A (https=)
AU (1) AU2016231832B2 (https=)
BR (1) BR112017019699A2 (https=)
CA (1) CA2979616C (https=)
HK (1) HK1243999A1 (https=)
IL (1) IL254124A0 (https=)
MX (1) MX2017011951A (https=)
RU (1) RU2672252C1 (https=)
SG (1) SG11201706992TA (https=)
WO (1) WO2016147144A1 (https=)

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WO2016147144A1 (en) 2016-09-22
BR112017019699A2 (pt) 2018-09-04
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US9873690B2 (en) 2018-01-23
EP3271354A1 (en) 2018-01-24
US20160272628A1 (en) 2016-09-22
CN107635990A (zh) 2018-01-26
AU2016231832A1 (en) 2017-09-14
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