JP6572201B2 - 眼疾患を処置するための組成物、製剤、および方法 - Google Patents

眼疾患を処置するための組成物、製剤、および方法 Download PDF

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JP6572201B2
JP6572201B2 JP2016503207A JP2016503207A JP6572201B2 JP 6572201 B2 JP6572201 B2 JP 6572201B2 JP 2016503207 A JP2016503207 A JP 2016503207A JP 2016503207 A JP2016503207 A JP 2016503207A JP 6572201 B2 JP6572201 B2 JP 6572201B2
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ethyl
substituted
acid
phenylsulfamic acid
thiazol
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JP2016516068A (ja
JP2016516068A5 (enExample
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ケビン ペータース，
ケビン ペータース，
ロバート シャルウィッツ，
ロバート シャルウィッツ，
ジョン ジャヌス，
ジョン ジャヌス，
アレクサンダー スミス，
アレクサンダー スミス，
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エアーピオ セラピューティクス インコーポレイテッド
エアーピオ セラピューティクス インコーポレイテッド
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
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    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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JP2016503207A 2013-03-15 2014-03-14 眼疾患を処置するための組成物、製剤、および方法 Active JP6572201B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US201361792679P 2013-03-15 2013-03-15
US201361792868P 2013-03-15 2013-03-15
US61/792,868 2013-03-15
US61/792,679 2013-03-15
US201361882048P 2013-09-25 2013-09-25
US201361882056P 2013-09-25 2013-09-25
US61/882,048 2013-09-25
US61/882,056 2013-09-25
US201461934570P 2014-01-31 2014-01-31
US61/934,570 2014-01-31
PCT/US2014/029723 WO2014145068A1 (en) 2013-03-15 2014-03-14 Compositions, formulations and methods for treating ocular diseases

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