JP6391674B2 - セニクリビロック組成物並びにその製造及び使用方法 - Google Patents
セニクリビロック組成物並びにその製造及び使用方法 Download PDFInfo
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- JP6391674B2 JP6391674B2 JP2016514093A JP2016514093A JP6391674B2 JP 6391674 B2 JP6391674 B2 JP 6391674B2 JP 2016514093 A JP2016514093 A JP 2016514093A JP 2016514093 A JP2016514093 A JP 2016514093A JP 6391674 B2 JP6391674 B2 JP 6391674B2
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US61/823,766 | 2013-05-15 | ||
| PCT/US2014/038211 WO2014186581A1 (en) | 2013-05-15 | 2014-05-15 | Cenicriviroc compositions and methods of making and using the same |
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| JP2016518452A JP2016518452A (ja) | 2016-06-23 |
| JP2016518452A5 JP2016518452A5 (https=) | 2017-06-08 |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017509704A (ja) * | 2014-03-21 | 2017-04-06 | トビラ セラピューティクス， インコーポレイテッド | 線維症を処置するためのセニクリビロック |
| JP2017526713A (ja) * | 2014-09-12 | 2017-09-14 | トビラ セラピューティクス， インコーポレイテッド | 線維症を処置するためのセニクリビロック併用療法 |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20030329A1 (es) | 2001-08-08 | 2003-05-12 | Takeda Chemical Industries Ltd | Compuesto biciclico con actividad antagonista de ccr5 y produccion del mismo |
| JP6716568B2 (ja) * | 2014-12-23 | 2020-07-01 | トビラ セラピューティクス， インコーポレイテッド | セニクリビロックの製造方法及び関連類似体 |
| BR112017016388A2 (pt) * | 2015-02-10 | 2018-03-27 | Tobira Therapeutics, Inc. | cenicriviroc para o tratamento da fibrose |
| WO2016135740A1 (en) * | 2015-02-23 | 2016-09-01 | Natco Pharma Limited | Process for preparing stable oral compositions of everolimus |
| US20180360846A1 (en) * | 2015-09-16 | 2018-12-20 | Tobira Therapeutics, Inc. | Cenicriviroc combination therapy for the treatment of fibrosis |
| JP2019520427A (ja) | 2016-06-21 | 2019-07-18 | トビラ セラピューティクス， インコーポレイテッド | 精製されたセニクリビロク及びセニクリビロク製造のための精製された中間体 |
| US11045423B2 (en) | 2016-08-08 | 2021-06-29 | Hetero Labs Limited | Anti-retroviral compositions |
| MX2019002057A (es) | 2016-08-31 | 2019-11-18 | Tobira Therapeutics Inc | Formas solidas de mesilato de cenicriviroc y procesos para elaborar formas sólidas de mesilato de cenicriviroc. |
| US10736905B1 (en) | 2016-09-09 | 2020-08-11 | Shahin Fatholahi | Nefopam dosage forms and methods of treatment |
| JP7326161B2 (ja) | 2017-05-11 | 2023-08-15 | キング アブドラ ユニバーシティ オブ サイエンス アンド テクノロジー | 組織エンジニアリングおよびバイオプリンティングにおける使用のためのゲルを形成し得るペプチド |
| KR102418307B1 (ko) | 2017-05-11 | 2022-07-06 | 킹 압둘라 유니버시티 오브 사이언스 앤드 테크놀로지 | 미세유체공학-기반 3d 바이오프린팅용 장치 및 방법 |
| RU2662160C9 (ru) * | 2017-07-03 | 2018-10-22 | Александрович Иващенко Андрей | Комбинированный лекарственный препарат для терапии вирусных инфекций |
| US11446311B2 (en) | 2017-09-08 | 2022-09-20 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
| US10736874B1 (en) | 2017-09-08 | 2020-08-11 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
| WO2021133811A1 (en) * | 2019-12-26 | 2021-07-01 | Teva Pharmaceuticals International Gmbh | Solid state forms of cenicriviroc and process for preparation thereof |
| EP4093380A1 (en) | 2020-01-23 | 2022-11-30 | Lupin Limited | Pharmaceutical compositions of raltegravir |
| US12109327B2 (en) | 2020-08-20 | 2024-10-08 | King Abdullah University Of Science And Technology | Scaffolds from self-assembling tetrapeptides support 3D spreading, osteogenic differentiation and angiogenesis of mesenchymal stem cells |
| US11673324B2 (en) | 2020-08-20 | 2023-06-13 | King Abdullah University Of Science And Technology | Nozzle for 3D bioprinting |
| US12590121B2 (en) | 2020-08-20 | 2026-03-31 | King Abdullah University Of Science And Technology | Peptide compound with repetitive sequences |
| JP2022108727A (ja) * | 2021-01-13 | 2022-07-26 | 日曹商事株式会社 | フマル酸含有固形製剤 |
Family Cites Families (7)
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| RU2167649C2 (ru) * | 1995-08-11 | 2001-05-27 | Ниссан Кемикал Индастриз, Лтд. | Способ получения твердой дисперсии умеренно водорастворимого лекарственного вещества (варианты) и фармацевтическая композиция |
| AU9461898A (en) * | 1997-10-20 | 1999-05-10 | Dainippon Pharmaceutical Co. Ltd. | Stable drug composition |
| CA2244097A1 (en) * | 1998-08-21 | 2000-02-21 | Bernard Charles Sherman | Pharmaceutical composition comprising bupropion hydrochloride and fumaric acid |
| WO2000061109A1 (fr) * | 1999-04-12 | 2000-10-19 | Shionogi & Co., Ltd. | Procede de production de composition medicamenteuse renfermant un compose medicamenteux hydrophobe basique |
| WO2006059716A1 (ja) * | 2004-12-03 | 2006-06-08 | Takeda Pharmaceutical Company Limited | 固形製剤 |
| EP2552429A1 (en) * | 2010-04-02 | 2013-02-06 | Phivco-1 LLC | Combination therapy comprising a ccr5 antagonist, a hiv-1 protease inhibitor and a pharmacokinetic enhancer |
| HK1232147A1 (zh) * | 2014-03-21 | 2018-01-05 | Tobira Therapeutics, Inc. | 用於治疗纤维化的赛尼克韦罗 |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017509704A (ja) * | 2014-03-21 | 2017-04-06 | トビラ セラピューティクス， インコーポレイテッド | 線維症を処置するためのセニクリビロック |
| JP2017526713A (ja) * | 2014-09-12 | 2017-09-14 | トビラ セラピューティクス， インコーポレイテッド | 線維症を処置するためのセニクリビロック併用療法 |
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| CA2911212A1 (en) | 2014-11-20 |
| AU2014265327A1 (en) | 2015-11-26 |
| MY180145A (en) | 2020-11-23 |
| CN105263498B (zh) | 2019-04-26 |
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| BR112015028644A2 (pt) | 2017-07-25 |
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| NZ713981A (en) | 2021-03-26 |
| RU2014150327A (ru) | 2016-07-10 |
| HK1214171A1 (zh) | 2016-07-22 |
| MX383706B (es) | 2025-03-14 |
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| PH12015502539B1 (en) | 2016-02-22 |
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| EP2996694A1 (en) | 2016-03-23 |
| RU2633069C2 (ru) | 2017-10-11 |
| CN105263498A (zh) | 2016-01-20 |
| WO2014186581A1 (en) | 2014-11-20 |
| AU2014265327B2 (en) | 2019-08-15 |
| CL2015003346A1 (es) | 2016-09-16 |
| EP2996694A4 (en) | 2016-12-07 |
| US20160081985A1 (en) | 2016-03-24 |
| SG11201509136YA (en) | 2015-12-30 |
| PH12015502539A1 (en) | 2016-02-22 |
| SG10201708595YA (en) | 2017-11-29 |
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