JP6301374B2 - キナーゼ阻害剤としてのキナゾリン類 - Google Patents
キナーゼ阻害剤としてのキナゾリン類 Download PDFInfo
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- JP6301374B2 JP6301374B2 JP2015558582A JP2015558582A JP6301374B2 JP 6301374 B2 JP6301374 B2 JP 6301374B2 JP 2015558582 A JP2015558582 A JP 2015558582A JP 2015558582 A JP2015558582 A JP 2015558582A JP 6301374 B2 JP6301374 B2 JP 6301374B2
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- butylsulfonyl
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| TWI547494B (zh) | 2011-08-18 | 2016-09-01 | 葛蘭素史克智慧財產發展有限公司 | 作為激酶抑制劑之胺基喹唑啉類 |
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| TWI592417B (zh) | 2012-09-13 | 2017-07-21 | 葛蘭素史克智慧財產發展有限公司 | 胺基喹唑啉激酶抑制劑之前藥 |
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| JP2019514878A (ja) * | 2016-04-20 | 2019-06-06 | グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ | Ｒｉｐｋ２阻害剤を含むコンジュゲート |
| CN112638905A (zh) * | 2018-08-28 | 2021-04-09 | 南京明德新药研发有限公司 | 作为rip2激酶抑制剂的喹唑啉类衍生物 |
| WO2025092821A1 (zh) * | 2023-11-01 | 2025-05-08 | 成都赜灵生物医药科技有限公司 | 喹唑啉衍生物类ripk2抑制剂及其用途 |
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| JP6301374B2 (ja) | 2013-02-21 | 2018-03-28 | グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ | キナーゼ阻害剤としてのキナゾリン類 |
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| EP2958911A1 (en) | 2015-12-30 |
| RU2015139758A (ru) | 2017-03-24 |
| CN105143208A (zh) | 2015-12-09 |
| JP2016509051A (ja) | 2016-03-24 |
| WO2014128622A1 (en) | 2014-08-28 |
| CN105143208B (zh) | 2017-09-26 |
| RU2662810C2 (ru) | 2018-07-31 |
| ES2654100T3 (es) | 2018-02-12 |
| BR112015019624A2 (pt) | 2017-07-18 |
| TW201444824A (zh) | 2014-12-01 |
| CA2902132A1 (en) | 2014-08-28 |
| US20150361069A1 (en) | 2015-12-17 |
| KR20150118152A (ko) | 2015-10-21 |
| AU2014220300A1 (en) | 2015-08-06 |
| AR094707A1 (es) | 2015-08-19 |
| AU2014220300B2 (en) | 2016-10-13 |
| EP2958911B1 (en) | 2017-10-18 |
| TWI630203B (zh) | 2018-07-21 |
| US9650364B2 (en) | 2017-05-16 |
| CA2902132C (en) | 2020-09-22 |
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