ITMI20052008A1 - Nuovi antimalarici derivati della 4-aminochinolina - Google Patents

Nuovi antimalarici derivati della 4-aminochinolina

Info

Publication number
ITMI20052008A1
ITMI20052008A1 IT002008A ITMI20052008A ITMI20052008A1 IT MI20052008 A1 ITMI20052008 A1 IT MI20052008A1 IT 002008 A IT002008 A IT 002008A IT MI20052008 A ITMI20052008 A IT MI20052008A IT MI20052008 A1 ITMI20052008 A1 IT MI20052008A1
Authority
IT
Italy
Prior art keywords
aminochinolina
antimalaric
derivatives
new
new antimalaric
Prior art date
Application number
IT002008A
Other languages
English (en)
Inventor
Fabio Sparatore
Original Assignee
Ctg Pharma S R L
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ctg Pharma S R L filed Critical Ctg Pharma S R L
Priority to IT002008A priority Critical patent/ITMI20052008A1/it
Priority to EP06809083A priority patent/EP1937686A1/en
Priority to PCT/IB2006/002946 priority patent/WO2007045987A1/en
Priority to CNA2006800486047A priority patent/CN101346381A/zh
Publication of ITMI20052008A1 publication Critical patent/ITMI20052008A1/it
Priority to AP2008004444A priority patent/AP2008004444A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT002008A 2005-10-21 2005-10-21 Nuovi antimalarici derivati della 4-aminochinolina ITMI20052008A1 (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
IT002008A ITMI20052008A1 (it) 2005-10-21 2005-10-21 Nuovi antimalarici derivati della 4-aminochinolina
EP06809083A EP1937686A1 (en) 2005-10-21 2006-10-20 New anti-malaria derivatives of 4-aminoquinoline
PCT/IB2006/002946 WO2007045987A1 (en) 2005-10-21 2006-10-20 New anti-malaria derivatives of 4-aminoquinoline
CNA2006800486047A CN101346381A (zh) 2005-10-21 2006-10-20 新颖的抗疟疾4-氨基喹啉衍生物
AP2008004444A AP2008004444A0 (en) 2005-10-21 2008-04-26 New anti-malaria derivatives of 4-aminoquinoline

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002008A ITMI20052008A1 (it) 2005-10-21 2005-10-21 Nuovi antimalarici derivati della 4-aminochinolina

Publications (1)

Publication Number Publication Date
ITMI20052008A1 true ITMI20052008A1 (it) 2007-04-22

Family

ID=37735214

Family Applications (1)

Application Number Title Priority Date Filing Date
IT002008A ITMI20052008A1 (it) 2005-10-21 2005-10-21 Nuovi antimalarici derivati della 4-aminochinolina

Country Status (5)

Country Link
EP (1) EP1937686A1 (it)
CN (1) CN101346381A (it)
AP (1) AP2008004444A0 (it)
IT (1) ITMI20052008A1 (it)
WO (1) WO2007045987A1 (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2743903A1 (en) 2008-11-18 2010-05-27 The Government Of The United States Of America D.B.A.The Department Of V Eterans Affairs Compounds for treating parasitic disease
EA023998B1 (ru) 2011-03-04 2016-08-31 Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед Аминохинолины в качестве ингибиторов киназ
TWI547494B (zh) 2011-08-18 2016-09-01 葛蘭素史克智慧財產發展有限公司 作為激酶抑制劑之胺基喹唑啉類
TW201425307A (zh) 2012-09-13 2014-07-01 Glaxosmithkline Llc 作為激酶抑制劑之胺基－喹啉類
AR092529A1 (es) 2012-09-13 2015-04-22 Glaxosmithkline Llc Compuesto de aminoquinazolina, composicion farmaceutica que lo comprende y uso de dicho compuesto para la preparacion de un medicamento
CN102898369A (zh) * 2012-11-05 2013-01-30 上海书亚医药科技有限公司 3-氨基-7-溴喹啉-2-甲酸乙酯及其制备方法
JP6301374B2 (ja) 2013-02-21 2018-03-28 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ キナーゼ阻害剤としてのキナゾリン類
CN106146466A (zh) * 2016-06-30 2016-11-23 珠海赛隆药业股份有限公司（长沙）医药研发中心 富马酸沃诺拉赞中间体、其制备方法和制备富马酸沃诺拉赞的方法
CN107915720B (zh) * 2016-10-08 2020-09-11 常州市第四制药厂有限公司 沃诺拉赞的新制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004533418A (ja) * 2001-03-14 2004-11-04 ザ・ユニヴァーシティ・オヴ・リヴァプール 抗マラリア化合物
ITMI20032044A1 (it) * 2003-10-21 2005-04-22 Univ Degli Studi Milano Chinolizidinil e chinolizidinilalchil-derivati della 4-ammino-chinolina ad attivita' antimalarica

Also Published As

Publication number Publication date
EP1937686A1 (en) 2008-07-02
CN101346381A (zh) 2009-01-14
WO2007045987A1 (en) 2007-04-26
AP2008004444A0 (en) 2008-04-30

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