CA2902132C - Quinazolines as kinase inhibitors - Google Patents
Quinazolines as kinase inhibitors Download PDFInfo
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- CA2902132C CA2902132C CA2902132A CA2902132A CA2902132C CA 2902132 C CA2902132 C CA 2902132C CA 2902132 A CA2902132 A CA 2902132A CA 2902132 A CA2902132 A CA 2902132A CA 2902132 C CA2902132 C CA 2902132C
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- disease
- compound
- pharmaceutically acceptable
- sarcoidosis
- tert
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Classifications
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Landscapes
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| PCT/IB2014/059094 WO2014128622A1 (en) | 2013-02-21 | 2014-02-19 | Quinazolines as kinase inhibitors |
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| US9604963B2 (en) | 2011-03-04 | 2017-03-28 | Glaxosmithkline Intellectual Property Development Limited | Amino-quinolines as kinase inhibitors |
| TWI547494B (zh) | 2011-08-18 | 2016-09-01 | 葛蘭素史克智慧財產發展有限公司 | 作為激酶抑制劑之胺基喹唑啉類 |
| TW201425307A (zh) | 2012-09-13 | 2014-07-01 | Glaxosmithkline Llc | 作為激酶抑制劑之胺基－喹啉類 |
| AR092529A1 (es) | 2012-09-13 | 2015-04-22 | Glaxosmithkline Llc | Compuesto de aminoquinazolina, composicion farmaceutica que lo comprende y uso de dicho compuesto para la preparacion de un medicamento |
| CA2902132C (en) | 2013-02-21 | 2020-09-22 | Glaxosmithkline Intellectual Property Development Limited | Quinazolines as kinase inhibitors |
| GB201506872D0 (en) | 2015-04-22 | 2015-06-03 | Ge Oil & Gas Uk Ltd | Novel compounds |
| GB201516243D0 (en) | 2015-09-14 | 2015-10-28 | Glaxosmithkline Ip Dev Ltd | Novel compounds |
| AU2017253560B2 (en) * | 2016-04-20 | 2019-03-21 | Glaxosmithkline Intellectual Property Development Limited | Conjugates comprising RIPK2 inhibitors |
| WO2020043122A1 (zh) * | 2018-08-28 | 2020-03-05 | 南京明德新药研发有限公司 | 作为rip2激酶抑制剂的喹唑啉类衍生物 |
| WO2025092821A1 (zh) * | 2023-11-01 | 2025-05-08 | 成都赜灵生物医药科技有限公司 | 喹唑啉衍生物类ripk2抑制剂及其用途 |
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| US4916135A (en) | 1989-05-08 | 1990-04-10 | Hoechst Roussel Pharmaceuticals Inc. | N-heteroaryl-4-quinolinamines |
| US5710158A (en) | 1991-05-10 | 1998-01-20 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Aryl and heteroaryl quinazoline compounds which inhibit EGF and/or PDGF receptor tyrosine kinase |
| PT100905A (pt) | 1991-09-30 | 1994-02-28 | Eisai Co Ltd | Compostos heterociclicos azotados biciclicos contendo aneis de benzeno, ciclo-hexano ou piridina e de pirimidina, piridina ou imidazol substituidos e composicoes farmaceuticas que os contem |
| GB9300059D0 (en) | 1992-01-20 | 1993-03-03 | Zeneca Ltd | Quinazoline derivatives |
| GB9510757D0 (en) | 1994-09-19 | 1995-07-19 | Wellcome Found | Therapeuticaly active compounds |
| US5747498A (en) | 1996-05-28 | 1998-05-05 | Pfizer Inc. | Alkynyl and azido-substituted 4-anilinoquinazolines |
| US6046206A (en) | 1995-06-07 | 2000-04-04 | Cell Pathways, Inc. | Method of treating a patient having a precancerous lesions with amide quinazoline derivatives |
| AR007857A1 (es) | 1996-07-13 | 1999-11-24 | Glaxo Group Ltd | Compuestos heterociclicos fusionados como inhibidores de proteina tirosina quinasa, sus metodos de preparacion, intermediarios uso en medicina ycomposiciones farmaceuticas que los contienen. |
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-
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- 2014-02-19 EP EP14708681.3A patent/EP2958911B1/en active Active
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- 2014-02-19 ES ES14708681.3T patent/ES2654100T3/es active Active
- 2014-02-19 US US14/762,905 patent/US9650364B2/en not_active Expired - Fee Related
- 2014-02-19 TW TW103105395A patent/TWI630203B/zh not_active IP Right Cessation
- 2014-02-19 BR BR112015019624A patent/BR112015019624A2/pt not_active Application Discontinuation
- 2014-02-19 RU RU2015139758A patent/RU2662810C2/ru not_active IP Right Cessation
- 2014-02-19 AU AU2014220300A patent/AU2014220300B2/en not_active Ceased
- 2014-02-19 JP JP2015558582A patent/JP6301374B2/ja not_active Expired - Fee Related
- 2014-02-19 WO PCT/IB2014/059094 patent/WO2014128622A1/en not_active Ceased
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Also Published As
| Publication number | Publication date |
|---|---|
| JP6301374B2 (ja) | 2018-03-28 |
| EP2958911B1 (en) | 2017-10-18 |
| AU2014220300B2 (en) | 2016-10-13 |
| TWI630203B (zh) | 2018-07-21 |
| RU2662810C2 (ru) | 2018-07-31 |
| BR112015019624A2 (pt) | 2017-07-18 |
| KR20150118152A (ko) | 2015-10-21 |
| JP2016509051A (ja) | 2016-03-24 |
| ES2654100T3 (es) | 2018-02-12 |
| WO2014128622A1 (en) | 2014-08-28 |
| AR094707A1 (es) | 2015-08-19 |
| TW201444824A (zh) | 2014-12-01 |
| CN105143208B (zh) | 2017-09-26 |
| AU2014220300A1 (en) | 2015-08-06 |
| CN105143208A (zh) | 2015-12-09 |
| RU2015139758A (ru) | 2017-03-24 |
| US9650364B2 (en) | 2017-05-16 |
| CA2902132A1 (en) | 2014-08-28 |
| US20150361069A1 (en) | 2015-12-17 |
| EP2958911A1 (en) | 2015-12-30 |
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