JP6005140B2 - ２型糖尿病患者の治療において使用するための組合せ医薬 - Google Patents
２型糖尿病患者の治療において使用するための組合せ医薬 Download PDFInfo
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- JP6005140B2 JP6005140B2 JP2014509759A JP2014509759A JP6005140B2 JP 6005140 B2 JP6005140 B2 JP 6005140B2 JP 2014509759 A JP2014509759 A JP 2014509759A JP 2014509759 A JP2014509759 A JP 2014509759A JP 6005140 B2 JP6005140 B2 JP 6005140B2
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
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- A—HUMAN NECESSITIES
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- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/2278—Vasoactive intestinal peptide [VIP]; Related peptides (e.g. Exendin)
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| EP11166052.8 | 2011-05-13 | ||
| EP11166052 | 2011-05-13 | ||
| PCT/EP2012/058779 WO2012156312A1 (en) | 2011-05-13 | 2012-05-11 | Pharmaceutical combination for use in the treatment of diabetes type 2 |
Publications (3)
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| JP2014518860A JP2014518860A (ja) | 2014-08-07 |
| JP2014518860A5 JP2014518860A5 (OSRAM) | 2015-06-18 |
| JP6005140B2 true JP6005140B2 (ja) | 2016-10-12 |
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| US (1) | US20130040878A1 (OSRAM) |
| EP (1) | EP2709652A1 (OSRAM) |
| JP (1) | JP6005140B2 (OSRAM) |
| KR (1) | KR20140041553A (OSRAM) |
| CN (2) | CN109045283A (OSRAM) |
| AR (1) | AR086356A1 (OSRAM) |
| AU (1) | AU2012257780B2 (OSRAM) |
| BR (1) | BR112013029256A8 (OSRAM) |
| CA (1) | CA2835336A1 (OSRAM) |
| MX (1) | MX356728B (OSRAM) |
| RU (2) | RU2017129878A (OSRAM) |
| WO (1) | WO2012156312A1 (OSRAM) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
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| LT2349324T (lt) | 2008-10-17 | 2017-12-27 | Sanofi-Aventis Deutschland Gmbh | Insulino ir glp-1 agonisto derinys |
| JP5832439B2 (ja) | 2009-11-13 | 2015-12-16 | サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | Ｇｌｐ−１アゴニスト、インスリン及びメチオニンを含む薬学的組成物 |
| CN102711804B (zh) | 2009-11-13 | 2015-09-16 | 赛诺菲-安万特德国有限公司 | 包含glp-1激动剂和甲硫氨酸的药物组合物 |
| US20110118178A1 (en) * | 2009-11-13 | 2011-05-19 | Sanofi-Aventis Deutschland Gmbh | Method of treatment of diabetes type 2 comprising add-on therapy to insulin glargine and metformin |
| CN103179978A (zh) | 2010-08-30 | 2013-06-26 | 赛诺菲-安万特德国有限公司 | Ave0010用于制造供治疗2型糖尿病用的药物的用途 |
| US9821032B2 (en) | 2011-05-13 | 2017-11-21 | Sanofi-Aventis Deutschland Gmbh | Pharmaceutical combination for improving glycemic control as add-on therapy to basal insulin |
| WO2013030160A1 (en) | 2011-08-29 | 2013-03-07 | Sanofi-Aventis Deutschland Gmbh | Pharmaceutical combination for use in glycemic control in diabetes type 2 patients |
| TWI559929B (en) | 2011-09-01 | 2016-12-01 | Sanofi Aventis Deutschland | Pharmaceutical composition for use in the treatment of a neurodegenerative disease |
| MX366685B (es) * | 2013-01-17 | 2019-07-19 | Vtv Therapeutics Llc | Combinaciones de un agonista de glp1r y metformina, y uso de los mismos para el tratamiento de la diabetes tipo 2 y otros trastornos. |
| TWI641381B (zh) | 2013-02-04 | 2018-11-21 | 法商賽諾菲公司 | 胰島素類似物及／或胰島素衍生物之穩定化醫藥調配物 |
| JP6735674B2 (ja) | 2014-01-09 | 2020-08-05 | サノフイＳａｎｏｆｉ | インスリンアスパルトの安定化された医薬製剤 |
| EP3091995B1 (en) | 2014-01-09 | 2024-03-20 | Sanofi | Stabilized pharmaceutical formulations of insulin aspart |
| US9895424B2 (en) | 2014-01-09 | 2018-02-20 | Sanofi | Stabilized pharmaceutical formulations of insulin analogues and/or insulin derivatives |
| MA41138B1 (fr) | 2014-12-12 | 2023-07-31 | Sanofi Aventis Deutschland | Formulation à rapport fixe d'insuline glargine/lixisenatide |
| TWI748945B (zh) | 2015-03-13 | 2021-12-11 | 德商賽諾菲阿凡提斯德意志有限公司 | 第２型糖尿病病患治療 |
| TW201705975A (zh) | 2015-03-18 | 2017-02-16 | 賽諾菲阿凡提斯德意志有限公司 | 第２型糖尿病病患之治療 |
| US12421245B2 (en) | 2020-04-01 | 2025-09-23 | Hangzhou Zhongmei Huadong Pharmaceutical Co., Ltd. | Pharmaceutically acceptable acid salt of free base of GLP1 receptor agonist, and preparation method therefor |
| JP2023528565A (ja) | 2020-04-01 | 2023-07-05 | ハンジョウ ジョンメイ フアドン ファーマシューティカル シーオー．，エルティーディー． | Ｇｌｐ－１受容体アゴニストの結晶形ａおよびその調製法 |
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| EP1076066A1 (en) | 1999-07-12 | 2001-02-14 | Zealand Pharmaceuticals A/S | Peptides for lowering blood glucose levels |
| US20110118178A1 (en) * | 2009-11-13 | 2011-05-19 | Sanofi-Aventis Deutschland Gmbh | Method of treatment of diabetes type 2 comprising add-on therapy to insulin glargine and metformin |
| EP2324853B1 (en) * | 2009-11-13 | 2015-08-26 | Sanofi-Aventis Deutschland GmbH | Lixisenatide as add-on to metformin in the treatment of diabetes type 2 |
| US20110118180A1 (en) * | 2009-11-13 | 2011-05-19 | Sanofi-Aventis Deutschland Gmbh | Method of treatment of diabetes type 2 comprising add-on therapy to metformin |
| JP5980466B2 (ja) * | 2009-11-13 | 2016-08-31 | サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | インスリングラルギン及びメトホルミンへの付加療法を含む２型糖尿病の治療方法 |
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2012
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- 2012-05-11 AR ARP120101668A patent/AR086356A1/es unknown
- 2012-05-11 RU RU2017129878A patent/RU2017129878A/ru not_active Application Discontinuation
- 2012-05-11 MX MX2013013198A patent/MX356728B/es active IP Right Grant
- 2012-05-11 KR KR1020137033311A patent/KR20140041553A/ko not_active Ceased
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- 2012-05-11 WO PCT/EP2012/058779 patent/WO2012156312A1/en not_active Ceased
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- 2012-05-11 BR BR112013029256A patent/BR112013029256A8/pt not_active Application Discontinuation
- 2012-05-11 JP JP2014509759A patent/JP6005140B2/ja not_active Expired - Fee Related
- 2012-05-11 CA CA2835336A patent/CA2835336A1/en not_active Abandoned
- 2012-05-11 AU AU2012257780A patent/AU2012257780B2/en not_active Ceased
- 2012-05-11 EP EP12720196.0A patent/EP2709652A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| BR112013029256A8 (pt) | 2018-01-16 |
| MX2013013198A (es) | 2014-02-20 |
| MX356728B (es) | 2018-06-12 |
| WO2012156312A1 (en) | 2012-11-22 |
| US20130040878A1 (en) | 2013-02-14 |
| RU2013155480A (ru) | 2015-06-20 |
| CN103648519A (zh) | 2014-03-19 |
| RU2017129878A (ru) | 2019-02-05 |
| CN109045283A (zh) | 2018-12-21 |
| AU2012257780B2 (en) | 2017-06-01 |
| EP2709652A1 (en) | 2014-03-26 |
| AR086356A1 (es) | 2013-12-04 |
| KR20140041553A (ko) | 2014-04-04 |
| BR112013029256A2 (pt) | 2016-11-29 |
| JP2014518860A (ja) | 2014-08-07 |
| CA2835336A1 (en) | 2012-11-22 |
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