JP5815542B2 - Ｄｐｐ−１阻害剤として有用なアルキニル誘導体 - Google Patents

Ｄｐｐ−１阻害剤として有用なアルキニル誘導体 Download PDF

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JP5815542B2
JP5815542B2 JP2012537052A JP2012537052A JP5815542B2 JP 5815542 B2 JP5815542 B2 JP 5815542B2 JP 2012537052 A JP2012537052 A JP 2012537052A JP 2012537052 A JP2012537052 A JP 2012537052A JP 5815542 B2 JP5815542 B2 JP 5815542B2
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phenyl
methyl
alkyl
group
oxy
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JP2013509423A (ja
JP2013509423A5 (enExample
Inventor
パーカー，マイケル，エィチ．
ラスタ，デニス，ジェィ．
フアン，イファン
ライツ，アレン，ビー．
ローソン，エドワード，シー．
シューベルト，カルステン
ストゥロベル，エリック
タング，ブレット
ホワイト，キンバリー
ウィンターズ，マイケル，ピー．
ゴッシュ，シャマリ
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ヤンセン ファーマシューティカ エヌ．ベー．
ヤンセン ファーマシューティカ エヌ．ベー．
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/16—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and unsaturated
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JP2012537052A 2009-10-29 2010-10-28 Ｄｐｐ−１阻害剤として有用なアルキニル誘導体 Expired - Fee Related JP5815542B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25617109P 2009-10-29 2009-10-29
US61/256,171 2009-10-29
PCT/US2010/054445 WO2011059731A1 (en) 2009-10-29 2010-10-28 Alkynyl derivatives useful as dpp-1 inhibitors

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JP2013509423A JP2013509423A (ja) 2013-03-14
JP2013509423A5 JP2013509423A5 (enExample) 2013-12-19
JP5815542B2 true JP5815542B2 (ja) 2015-11-17

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US8633322B2 (en) 2014-01-21

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