CN102596321B - 可用作dpp-1抑制剂的炔基衍生物 - Google Patents

可用作dpp-1抑制剂的炔基衍生物 Download PDF

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Publication number
CN102596321B
CN102596321B CN201080049814.4A CN201080049814A CN102596321B CN 102596321 B CN102596321 B CN 102596321B CN 201080049814 A CN201080049814 A CN 201080049814A CN 102596321 B CN102596321 B CN 102596321B
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phenyl
base
methyl
alkyl
compound
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CN102596321A (zh
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M·H·帕克
D·J·赫拉斯塔
黄义方
A·B·雷茨
E·C·劳森
C·舒伯特
E·斯特罗贝尔
B·通格
K·怀特
M·P·温特斯
S·高希
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Janssen Pharmaceutica NV
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    • C07C237/16—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and unsaturated
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CN201080049814.4A 2009-10-29 2010-10-28 可用作dpp-1抑制剂的炔基衍生物 Expired - Fee Related CN102596321B (zh)

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US25617109P 2009-10-29 2009-10-29
US61/256171 2009-10-29
US61/256,171 2009-10-29
PCT/US2010/054445 WO2011059731A1 (en) 2009-10-29 2010-10-28 Alkynyl derivatives useful as dpp-1 inhibitors

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CN102596321A CN102596321A (zh) 2012-07-18
CN102596321B true CN102596321B (zh) 2014-11-19

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