JP5766716B2 - 多環式グアニジン化合物の合成のための方法 - Google Patents

多環式グアニジン化合物の合成のための方法 Download PDF

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JP5766716B2
JP5766716B2 JP2012546076A JP2012546076A JP5766716B2 JP 5766716 B2 JP5766716 B2 JP 5766716B2 JP 2012546076 A JP2012546076 A JP 2012546076A JP 2012546076 A JP2012546076 A JP 2012546076A JP 5766716 B2 JP5766716 B2 JP 5766716B2
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guanidine
item
certain embodiments
optionally substituted
compound
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JP2013515728A5 (enExample
JP2013515728A (ja
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アレクセイ グリードネフ，
アレクセイ グリードネフ，
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ノボマー， インコーポレイテッド
ノボマー， インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/02—Guanidine; Salts, complexes or addition compounds thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
    • C07D251/40—Nitrogen atoms
    • C07D251/54—Three nitrogen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2012546076A 2009-12-24 2010-12-17 多環式グアニジン化合物の合成のための方法 Active JP5766716B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US29008709P 2009-12-24 2009-12-24
US61/290,087 2009-12-24
US29904710P 2010-01-28 2010-01-28
US61/299,047 2010-01-28
US42249210P 2010-12-13 2010-12-13
US61/422,492 2010-12-13
PCT/US2010/060985 WO2011079041A1 (en) 2009-12-24 2010-12-17 Methods for the synthesis of polycyclic guanidine compounds

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JP2013515728A JP2013515728A (ja) 2013-05-09
JP2013515728A5 JP2013515728A5 (enExample) 2014-02-13
JP5766716B2 true JP5766716B2 (ja) 2015-08-19

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US (2) US8642771B2 (enExample)
EP (1) EP2515648B1 (enExample)
JP (1) JP5766716B2 (enExample)
KR (1) KR101885503B1 (enExample)
CN (1) CN102665406B (enExample)
NO (1) NO2515648T3 (enExample)
WO (1) WO2011079041A1 (enExample)

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US8563560B2 (en) 2011-02-25 2013-10-22 Ppg Industries Ohio, Inc. Preparation of bicyclic guanidine salts in an aqueous media
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ES2633809T3 (es) 2013-01-30 2017-09-25 Basf Se Derivados de 2,6-bis-(aminometil)-piperidina (2,6-BAMP), derivados de 2,6-bis-(isocianometil)piperidin-(diisocianato) y derivados de 2,6-dicianopiperidina (derivados de 2,6-DCP) y su uso en la preparación de resinas epoxi, poliuretanos, polieteroles y poliamidas
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CN103172639B (zh) * 2013-03-18 2015-08-12 惠州市莱佛士制药技术有限公司 一种基于盐酸胍的六元二环胍的制备方法
US9688874B2 (en) 2013-10-25 2017-06-27 Ppg Industries Ohio, Inc. Method of making a bicyclic guanidine-cured acrylic coating
CN103539798A (zh) * 2013-11-12 2014-01-29 南京大学 一种双环胍（1,5,7-三氮杂双环[5.5.0]癸-5-烯）的合成方法
CN103755598A (zh) * 2014-01-23 2014-04-30 上海旭新化工科技有限公司 胍丁胺硫酸盐的合成方法
CN104844608B (zh) * 2015-04-13 2017-09-19 南京大学 相转移催化法合成双环胍tbd的工艺方法
WO2018128823A1 (en) 2017-01-03 2018-07-12 Chen Hwang Hsing Branched polymeric biguanide compounds and their uses
CN107325102B (zh) * 2017-08-11 2019-11-12 南京大学 自催化双亲混合溶剂中合成1,5,7-三氮杂双环[4.4.0]癸-5-烯的工艺方法
FI129024B (en) * 2017-11-08 2021-05-14 Helsingin Yliopisto Process for the preparation of bicyclic guanidine and its derivatives
WO2019126221A1 (en) 2017-12-22 2019-06-27 Saudi Aramco Technologies Company Catalysts for polycarbonate production
WO2020048604A1 (de) 2018-09-06 2020-03-12 Wacker Chemie Ag Verfahren zur herstellung bicyclischer guanidine
FI4048673T3 (fi) * 2019-10-22 2024-02-21 Basf Se Menetelmä syklisten guanidiinijohdannaisten tuottamiseksi
CN112094273A (zh) * 2020-08-07 2020-12-18 天津全和诚科技有限责任公司 一种的双环胍的合成方法
CN112961343B (zh) * 2021-02-19 2023-08-29 上海凯赛生物技术股份有限公司 一种戊二胺磷酸胍盐齐聚物、其制备方法及由其制得的抗菌聚合物
CN121752569A (zh) 2023-08-25 2026-03-27 赢创运营有限公司 制造双环胍的方法

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Publication number Publication date
US9738647B2 (en) 2017-08-22
CN102665406A (zh) 2012-09-12
KR101885503B1 (ko) 2018-08-07
EP2515648B1 (en) 2017-08-16
NO2515648T3 (enExample) 2018-01-13
JP2013515728A (ja) 2013-05-09
US20140194622A1 (en) 2014-07-10
EP2515648A1 (en) 2012-10-31
WO2011079041A1 (en) 2011-06-30
CN102665406B (zh) 2016-03-09
KR20120124419A (ko) 2012-11-13
US20120259112A1 (en) 2012-10-11
EP2515648A4 (en) 2014-08-27
US8642771B2 (en) 2014-02-04

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