JP5582701B2 - 被覆医薬製剤およびポリマー混合被覆した医薬製剤の製造のためのポリマー混合物の使用 - Google Patents
被覆医薬製剤およびポリマー混合被覆した医薬製剤の製造のためのポリマー混合物の使用 Download PDFInfo
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- JP5582701B2 JP5582701B2 JP2008512703A JP2008512703A JP5582701B2 JP 5582701 B2 JP5582701 B2 JP 5582701B2 JP 2008512703 A JP2008512703 A JP 2008512703A JP 2008512703 A JP2008512703 A JP 2008512703A JP 5582701 B2 JP5582701 B2 JP 5582701B2
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005024614.1 | 2005-05-25 | ||
| DE102005024614A DE102005024614A1 (de) | 2005-05-25 | 2005-05-25 | Verwendung von Polymermischungen zur Herstellung von überzogenen Arzneiformen sowie Arzneiform mit polymerem Mischüberzug |
| PCT/EP2006/001949 WO2006125483A1 (de) | 2005-05-25 | 2006-03-03 | Verwendung vom polymermischungen zur herstellung von überzogenen arzneiformen sowie arzneiform mit |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008542211A JP2008542211A (ja) | 2008-11-27 |
| JP2008542211A5 JP2008542211A5 (enExample) | 2010-03-18 |
| JP5582701B2 true JP5582701B2 (ja) | 2014-09-03 |
Family
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Family Applications (1)
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| JP2008512703A Expired - Fee Related JP5582701B2 (ja) | 2005-05-25 | 2006-03-03 | 被覆医薬製剤およびポリマー混合被覆した医薬製剤の製造のためのポリマー混合物の使用 |
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| EP (1) | EP1890682B1 (enExample) |
| JP (1) | JP5582701B2 (enExample) |
| KR (1) | KR101387835B1 (enExample) |
| CN (1) | CN101137354B (enExample) |
| BR (1) | BRPI0610206B8 (enExample) |
| CA (1) | CA2606587C (enExample) |
| DE (1) | DE102005024614A1 (enExample) |
| ES (1) | ES2628962T3 (enExample) |
| HU (1) | HUE032869T2 (enExample) |
| IL (1) | IL187535A0 (enExample) |
| MX (1) | MX363064B (enExample) |
| PL (1) | PL1890682T3 (enExample) |
| SI (1) | SI1890682T1 (enExample) |
| WO (1) | WO2006125483A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US8461187B2 (en) | 2004-06-16 | 2013-06-11 | Takeda Pharmaceuticals U.S.A., Inc. | Multiple PPI dosage form |
| WO2008070072A2 (en) * | 2006-12-01 | 2008-06-12 | Mutual Pharmaceutical Company, Inc. | Carvedilol forms, compositions, and methods of preparation thereof |
| CA2677053C (en) * | 2007-01-31 | 2016-03-15 | Methylation Sciences International Srl | Extended release pharmaceutical formulations of s-adenosylmethionine |
| ES2393934T3 (es) * | 2007-09-21 | 2013-01-02 | Evonik Röhm Gmbh | Composición farmacéutica opioide de lberación controlada dependiente del PH con resitencia frente a la influencia del etanol |
| CN101801356B (zh) | 2007-09-21 | 2016-10-19 | 赢创罗姆有限公司 | 耐受乙醇影响的非阿片类的pH依赖性受控释放的药物组合物 |
| RU2010119041A (ru) * | 2007-10-12 | 2011-11-20 | Такеда Фармасьютикалз Норт Америка, Инк. (Us) | Способы лечения нарушений желудочно-кишечного тракта, независимого от потребления пищи |
| EP2254556A2 (en) * | 2008-03-11 | 2010-12-01 | Takeda Pharmaceutical Company Limited | Orally-disintegrating solid preparation |
| RU2011102777A (ru) * | 2008-06-26 | 2012-08-10 | МакНЕЙЛ-ППС, ИНК. (US) | Частицы с покрытием, содержащие фармацевтически активные агенты |
| CN104984343B (zh) * | 2008-09-24 | 2019-04-02 | 赢创罗姆有限公司 | 耐受乙醇影响的非阿片类药物的pH依赖性受控释放的药物组合物 |
| KR101528957B1 (ko) * | 2008-09-24 | 2015-06-17 | 에보니크 룀 게엠베하 | 에탄올의 영향에 대하여 내성을 갖는 ｐｈ-의존성 조절 방출 제약학적 오피오이드 조성물 |
| EP2326313B1 (en) * | 2008-09-24 | 2015-03-04 | Evonik Röhm GmbH | Ph-dependent controlled release pharmaceutical composition for non-opioids with resistance against the influence of ethanol |
| EP2364138A2 (en) * | 2008-12-08 | 2011-09-14 | Teva Pharmaceutical Industries Ltd. | Palonosetron formulation |
| JP5619130B2 (ja) | 2009-03-18 | 2014-11-05 | エボニック レーム ゲゼルシャフト ミット ベシュレンクテル ハフツングＥｖｏｎｉｋ ＲｏｅｈｍＧｍｂＨ | 中性ビニルポリマーおよび賦形剤を含むコーティングを使用するエタノールの影響に対する耐性を有する制御放出性医薬組成物 |
| US20110311631A1 (en) * | 2009-03-18 | 2011-12-22 | Evonik Röhm Gmbh | Controlled release pharmaceutical composition with resistance against the influence of ethanol employing a coating comprising a polymer mixture and excipients |
| CN105287434A (zh) * | 2009-03-18 | 2016-02-03 | 赢创罗姆有限公司 | 采用含有中性乙烯基聚合物和赋形剂的包衣的具有耐乙醇影响的控释药物组合物 |
| US20100303920A1 (en) * | 2009-05-27 | 2010-12-02 | Johan Hjartstam | Aqueous Film Coating Composition / 841 |
| US8329208B2 (en) | 2009-07-28 | 2012-12-11 | Methylation Sciences International Srl | Pharmacokinetics of S-adenosylmethionine formulations |
| DK2490675T3 (en) * | 2009-10-22 | 2019-04-29 | Synthon Bv | Pharmaceutical compositions with sevelamer |
| WO2012171884A1 (en) * | 2011-06-17 | 2012-12-20 | Evonik Röhm Gmbh | Gastric resistant pharmaceutical or nutraceutical composition with resistance against the influence of ethanol |
| KR101748053B1 (ko) | 2012-10-17 | 2017-06-15 | 메틸레이션 사이언시즈 인터내셔널 에스알엘 | S-아데노실메티오닌 및 갈산 에스테르가 포함된 조성물 |
| CA3018328A1 (en) | 2014-10-31 | 2016-04-30 | Purdue Pharma | Methods and compositions particularly for treatment of attention deficit disorder |
| US20170042806A1 (en) | 2015-04-29 | 2017-02-16 | Dexcel Pharma Technologies Ltd. | Orally disintegrating compositions |
| CA2986188A1 (en) | 2015-06-05 | 2016-12-08 | Evonik Rohm Gmbh | Pharmaceutical or nutraceutical composition with resistance against the influence of ethanol |
| US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
| JP6739275B2 (ja) * | 2016-08-02 | 2020-08-12 | 日本化薬株式会社 | ゲフィチニブを有効成分とする医薬組成物 |
| IT201700032367A1 (it) * | 2017-03-23 | 2018-09-23 | Lamberti Spa | Dispersioni poliuretaniche acquose |
| CN112469399A (zh) * | 2018-03-09 | 2021-03-09 | 赢创运营有限公司 | 耐受乙醇影响的聚合物混合物 |
| US10722473B2 (en) | 2018-11-19 | 2020-07-28 | Purdue Pharma L.P. | Methods and compositions particularly for treatment of attention deficit disorder |
| CN114026188A (zh) * | 2019-06-07 | 2022-02-08 | 日本曹达株式会社 | 微粒用的湿式涂布剂 |
| CN113950321A (zh) * | 2019-06-13 | 2022-01-18 | 赢创运营有限公司 | 包含共聚物混合物和水溶性纤维素的粉末组合物 |
| US12569481B2 (en) | 2020-06-12 | 2026-03-10 | Vanderbilt University | Methods of treatment for gastrointestinal motility disorders |
| CN111700871A (zh) * | 2020-06-24 | 2020-09-25 | 杭州巴洛特生物科技有限公司 | 一种美沙拉嗪组合物及其制备方法 |
| CN112237572A (zh) * | 2020-10-28 | 2021-01-19 | 海南卫康制药(潜山)有限公司 | 一种富马酸沃诺拉赞片剂及其制备方法 |
| CN114409998A (zh) * | 2021-12-24 | 2022-04-29 | 浙江普利特新材料有限公司 | 一种蜂窝状咖啡炭复合隔音降噪聚丙烯材料及其制备方法 |
| EP4712796A2 (en) | 2023-05-15 | 2026-03-25 | Bonafide Health, LLC | Sleep-improving compositions and methods of use |
| CN120204161A (zh) * | 2025-04-08 | 2025-06-27 | 江西英特科胜动保科技有限公司 | 一种氟尼辛葡甲胺颗粒及其制备方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5019397A (en) * | 1988-04-21 | 1991-05-28 | Alza Corporation | Aqueous emulsion for pharmaceutical dosage form |
| IT1227899B (it) * | 1988-12-23 | 1991-05-14 | Poli Ind Chimica Spa | Rivestimento totale o parziale di principi attivi farmaceutici e relative composizioni |
| DE9414066U1 (de) * | 1994-08-31 | 1994-11-03 | Röhm GmbH & Co. KG, 64293 Darmstadt | Überzugs- und Bindemittel für Arzneiformen sowie damit hergestellte Arzneiform |
| JPH09323926A (ja) * | 1996-03-15 | 1997-12-16 | Nikken Chem Co Ltd | バルプロ酸ナトリウムの徐放性錠剤 |
| CA2388560A1 (en) * | 1999-08-31 | 2001-03-08 | Grunenthal Gmbh | Sustained-release form of administration containing tramadol saccharinate |
| DE10013029A1 (de) * | 2000-03-17 | 2001-09-20 | Roehm Gmbh | Mehrschichtige Arzneiform für die Colonfreigabe |
| EP1416922A1 (en) * | 2001-07-16 | 2004-05-12 | AstraZeneca AB | Pharmaceutical formulation comprising a proton pump inhibitor and antacids |
| CA2460132A1 (en) * | 2001-10-15 | 2003-04-24 | Roehm Gmbh & Co. Kg | Use of a copolymer to produce a galenic form containing a peptide or a protein as active agent |
| WO2004041255A1 (en) * | 2002-10-31 | 2004-05-21 | Alza Corporation | Dosage form providing ascending release of liquid formulation |
| ES2645930T3 (es) * | 2003-01-03 | 2017-12-11 | Supernus Pharmaceuticals, Inc. | Utilización de una mezcla de dos o más materiales entéricos para regular la liberación de fármacos a través de una membrana o matriz para terapias sistémicas |
| MXPA04010956A (es) * | 2003-01-30 | 2005-01-25 | Roehm Gmbh | Forma de dosis farmaceutica y metodo para la produccion de la misma. |
| BRPI0415557A (pt) * | 2003-10-31 | 2006-12-26 | Hexal Ag | formulação contendo ingrediente ativo farmacêutico com revestimento |
-
2005
- 2005-05-25 DE DE102005024614A patent/DE102005024614A1/de not_active Withdrawn
-
2006
- 2006-03-03 PL PL06723193T patent/PL1890682T3/pl unknown
- 2006-03-03 KR KR1020077027199A patent/KR101387835B1/ko not_active Expired - Fee Related
- 2006-03-03 CA CA2606587A patent/CA2606587C/en not_active Expired - Lifetime
- 2006-03-03 SI SI200632186T patent/SI1890682T1/sl unknown
- 2006-03-03 WO PCT/EP2006/001949 patent/WO2006125483A1/de not_active Ceased
- 2006-03-03 ES ES06723193.6T patent/ES2628962T3/es not_active Expired - Lifetime
- 2006-03-03 JP JP2008512703A patent/JP5582701B2/ja not_active Expired - Fee Related
- 2006-03-03 EP EP06723193.6A patent/EP1890682B1/de not_active Expired - Lifetime
- 2006-03-03 HU HUE06723193A patent/HUE032869T2/en unknown
- 2006-03-03 US US11/909,315 patent/US20080193522A1/en not_active Abandoned
- 2006-03-03 BR BRPI0610206A patent/BRPI0610206B8/pt not_active IP Right Cessation
- 2006-03-03 CN CN200680007508.8A patent/CN101137354B/zh not_active Expired - Fee Related
- 2006-03-03 MX MX2007014024A patent/MX363064B/es unknown
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2007
- 2007-11-21 IL IL187535A patent/IL187535A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20080009213A (ko) | 2008-01-25 |
| ES2628962T3 (es) | 2017-08-04 |
| BRPI0610206A2 (pt) | 2010-06-01 |
| HK1116341A1 (en) | 2008-12-19 |
| MX2007014024A (es) | 2008-04-09 |
| SI1890682T1 (sl) | 2017-10-30 |
| KR101387835B1 (ko) | 2014-04-25 |
| JP2008542211A (ja) | 2008-11-27 |
| WO2006125483A1 (de) | 2006-11-30 |
| CA2606587C (en) | 2015-05-26 |
| MX363064B (es) | 2019-03-06 |
| EP1890682B1 (de) | 2017-05-03 |
| DE102005024614A1 (de) | 2006-11-30 |
| IL187535A0 (en) | 2008-03-20 |
| BRPI0610206B8 (pt) | 2022-07-05 |
| US20080193522A1 (en) | 2008-08-14 |
| CN101137354B (zh) | 2014-06-11 |
| EP1890682A1 (de) | 2008-02-27 |
| PL1890682T3 (pl) | 2017-10-31 |
| BRPI0610206B1 (pt) | 2020-10-06 |
| CA2606587A1 (en) | 2006-11-30 |
| HUE032869T2 (en) | 2017-11-28 |
| CN101137354A (zh) | 2008-03-05 |
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