JP5524084B2 - Ｈｓｐ９０阻害剤としてのオキシム誘導体 - Google Patents

Ｈｓｐ９０阻害剤としてのオキシム誘導体 Download PDF

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JP5524084B2
JP5524084B2 JP2010545233A JP2010545233A JP5524084B2 JP 5524084 B2 JP5524084 B2 JP 5524084B2 JP 2010545233 A JP2010545233 A JP 2010545233A JP 2010545233 A JP2010545233 A JP 2010545233A JP 5524084 B2 JP5524084 B2 JP 5524084B2
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alkyl
hetero
aryl
cycloalkyl
amino
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JP2011511003A5 (OSRAM
JP2011511003A (ja
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チェン、ヤング、ケー．
ワン コー、エリック
グントゥパッリ、プラスナ
デイビッド ローソン、ジョン
ラインハルト ルートヴィヒ ノッツ、ウォルフガング
エー． スタッフォード、ジェフリー
トン−ヌー、フォーン−トゥ
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Takeda Pharmaceutical Co Ltd
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Takeda Pharmaceutical Co Ltd
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
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    • C07D239/72—Quinazolines; Hydrogenated quinazolines
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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JP2010545233A 2008-02-01 2009-01-30 Ｈｓｐ９０阻害剤としてのオキシム誘導体 Expired - Fee Related JP5524084B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US2572508P 2008-02-01 2008-02-01
US61/025,725 2008-02-01
US10159508P 2008-09-30 2008-09-30
US61/101,595 2008-09-30
PCT/US2009/032728 WO2009097578A1 (en) 2008-02-01 2009-01-30 Oxim derivatives as hsp90 inhibitors

Publications (3)

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JP2011511003A JP2011511003A (ja) 2011-04-07
JP2011511003A5 JP2011511003A5 (OSRAM) 2012-03-15
JP5524084B2 true JP5524084B2 (ja) 2014-06-18

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JP2010545233A Expired - Fee Related JP5524084B2 (ja) 2008-02-01 2009-01-30 Ｈｓｐ９０阻害剤としてのオキシム誘導体

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US (4) US8071766B2 (OSRAM)
EP (1) EP2252595B1 (OSRAM)
JP (1) JP5524084B2 (OSRAM)
KR (1) KR20100116206A (OSRAM)
CN (1) CN101983191B (OSRAM)
AR (1) AR071452A1 (OSRAM)
AU (1) AU2009208947B2 (OSRAM)
BR (1) BRPI0906598A2 (OSRAM)
CA (1) CA2713658C (OSRAM)
CL (1) CL2009000228A1 (OSRAM)
CR (1) CR11659A (OSRAM)
DO (1) DOP2010000236A (OSRAM)
EA (1) EA019156B1 (OSRAM)
EC (1) ECSP10010434A (OSRAM)
ES (1) ES2475206T3 (OSRAM)
GE (1) GEP20125718B (OSRAM)
IL (1) IL207227A0 (OSRAM)
MA (1) MA32104B1 (OSRAM)
MX (1) MX2010008269A (OSRAM)
MY (1) MY150596A (OSRAM)
NZ (1) NZ587207A (OSRAM)
PE (1) PE20091371A1 (OSRAM)
SG (1) SG187502A1 (OSRAM)
TW (1) TW200946531A (OSRAM)
WO (1) WO2009097578A1 (OSRAM)
ZA (1) ZA201005435B (OSRAM)

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