JP5401463B2 - 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 - Google Patents

新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 Download PDF

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JP5401463B2
JP5401463B2 JP2010533467A JP2010533467A JP5401463B2 JP 5401463 B2 JP5401463 B2 JP 5401463B2 JP 2010533467 A JP2010533467 A JP 2010533467A JP 2010533467 A JP2010533467 A JP 2010533467A JP 5401463 B2 JP5401463 B2 JP 5401463B2
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formula
compound
administered
combination
crystalline hydrate
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JP2011503127A (ja
JP2011503127A5 (https=
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テーオドール・アンドレーアス・ヴォルマン
レジーナ・デューフィー
フランク・クルマン
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サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2010533467A 2007-11-13 2008-11-06 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用 Expired - Fee Related JP5401463B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DE102007054497.0 2007-11-13
DE102007054497A DE102007054497B3 (de) 2007-11-13 2007-11-13 Neue kristalline Diphenylazetidinonhydrate und Verfahren zu deren Herstellung
US99025507P 2007-11-26 2007-11-26
US60/990,255 2007-11-26
PCT/EP2008/009323 WO2009062619A1 (de) 2007-11-13 2008-11-06 Neue kristalline diphenylazetidinonhydrate, diese verbindungen enthaltende arzneimittel und deren verwendung

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JP2011503127A JP2011503127A (ja) 2011-01-27
JP2011503127A5 JP2011503127A5 (https=) 2011-12-22
JP5401463B2 true JP5401463B2 (ja) 2014-01-29

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JP2010533467A Expired - Fee Related JP5401463B2 (ja) 2007-11-13 2008-11-06 新規な結晶性ジフェニルアゼチジノン水和物、これらの化合物を含有する薬剤およびそれらの使用

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US (1) US8003636B2 (https=)
EP (1) EP2220040B1 (https=)
JP (1) JP5401463B2 (https=)
AR (1) AR069305A1 (https=)
CL (1) CL2008003358A1 (https=)
DE (2) DE102007054497B3 (https=)
PA (1) PA8803701A1 (https=)
PE (1) PE20091165A1 (https=)
TW (1) TW200936566A (https=)
UY (1) UY31469A1 (https=)
WO (1) WO2009062619A1 (https=)

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EP3954688A1 (en) * 2012-12-22 2022-02-16 Kbp Biosciences Pte. Ltd. Crystal forms of compound used as mineralocorticoid receptor antagonist and methods for their preparation
US10064871B2 (en) 2014-01-22 2018-09-04 Biomimetix Jv, Llc Methods of treating skin disorders
US10080759B2 (en) 2014-01-22 2018-09-25 Duke University Methods of treating pruritus

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AR069305A1 (es) 2010-01-13
US20090203578A1 (en) 2009-08-13
PE20091165A1 (es) 2009-08-31
TW200936566A (en) 2009-09-01
CL2008003358A1 (es) 2009-06-26
EP2220040B1 (de) 2013-01-16
JP2011503127A (ja) 2011-01-27
PA8803701A1 (es) 2009-06-23
WO2009062619A1 (de) 2009-05-22
US8003636B2 (en) 2011-08-23
EP2220040A1 (de) 2010-08-25
DE102007063671A1 (de) 2009-06-25

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