JP5380293B2 - 選択的グリコシダーゼ阻害剤およびその使用 - Google Patents

選択的グリコシダーゼ阻害剤およびその使用 Download PDF

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JP5380293B2
JP5380293B2 JP2009525881A JP2009525881A JP5380293B2 JP 5380293 B2 JP5380293 B2 JP 5380293B2 JP 2009525881 A JP2009525881 A JP 2009525881A JP 2009525881 A JP2009525881 A JP 2009525881A JP 5380293 B2 JP5380293 B2 JP 5380293B2
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tetrahydro
compounds
glcnac
nmr
compound
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JP2010501598A5 (enExample
JP2010501598A (ja
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デイビッド・ボカドロ
アーネスト・マクイーチャーン
ガレット・ホイットワース
マシュー・マコーレー
ジュリア・ヘイノネン
キース・スタッブス
トン−シュアン・リ
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Simon Fraser University
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    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/68—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids
    • G01N33/6803—General methods of protein analysis not limited to specific proteins or families of proteins
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    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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    • C07H9/06—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing nitrogen as ring hetero atoms

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JP2009525881A 2006-08-31 2007-08-31 選択的グリコシダーゼ阻害剤およびその使用 Expired - Fee Related JP5380293B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US84119606P 2006-08-31 2006-08-31
US60/841,196 2006-08-31
US89566307P 2007-03-19 2007-03-19
US60/895,663 2007-03-19
PCT/CA2007/001554 WO2008025170A1 (en) 2006-08-31 2007-08-31 Selective glycosidase inhibitors and uses thereof

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JP2010501598A JP2010501598A (ja) 2010-01-21
JP2010501598A5 JP2010501598A5 (enExample) 2010-10-21
JP5380293B2 true JP5380293B2 (ja) 2014-01-08

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US (2) US8334310B2 (enExample)
EP (2) EP2057171A4 (enExample)
JP (2) JP5380293B2 (enExample)
AU (1) AU2007291870B2 (enExample)
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AU2012298949B2 (en) * 2011-08-25 2016-09-22 Merck Patent Gmbh Pyrano [3, 2 - D] [1, 3] thiazole as glycosidase inhibitors
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KR102108586B1 (ko) * 2012-05-08 2020-05-07 머크 샤프 앤드 돔 코포레이션 투과성 글리코시다제 억제제 및 그의 용도
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US20120316207A1 (en) 2012-12-13
AU2007291870A1 (en) 2008-03-06
US8334310B2 (en) 2012-12-18
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US8962664B2 (en) 2015-02-24
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