JP5327518B2 - ５−リポキシゲナーゼ−活性化タンパク質（ｆｌａｐ）阻害剤 - Google Patents

５−リポキシゲナーゼ−活性化タンパク質（ｆｌａｐ）阻害剤 Download PDF

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JP5327518B2
JP5327518B2 JP2008535605A JP2008535605A JP5327518B2 JP 5327518 B2 JP5327518 B2 JP 5327518B2 JP 2008535605 A JP2008535605 A JP 2008535605A JP 2008535605 A JP2008535605 A JP 2008535605A JP 5327518 B2 JP5327518 B2 JP 5327518B2
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compound
leukotriene
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JP2009521399A (ja
JP2009521399A5 (enExample
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ハチンソン，ジョン，エイチ．
プラシト，ペティブーン，ペッピ
モラン，マーク
エヴァンス，ジュリアン，エフ．
ズニック，ジャスミン，エレノア
ストック，ニコラス，サイモン
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パンミラ ファーマシューティカルズ，エルエルシー．
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings

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  • Health & Medical Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP2008535605A 2005-10-11 2006-10-05 ５−リポキシゲナーゼ−活性化タンパク質（ｆｌａｐ）阻害剤 Expired - Fee Related JP5327518B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US72557305P 2005-10-11 2005-10-11
US60/725,573 2005-10-11
US11/538,762 2006-10-04
US11/538,762 US7405302B2 (en) 2005-10-11 2006-10-04 5-lipoxygenase-activating protein (FLAP) inhibitors
PCT/US2006/039421 WO2007047207A2 (en) 2005-10-11 2006-10-05 5-lipoxygenase-activating protein (flap) inhibitors

Publications (3)

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JP2009521399A JP2009521399A (ja) 2009-06-04
JP2009521399A5 JP2009521399A5 (enExample) 2009-11-12
JP5327518B2 true JP5327518B2 (ja) 2013-10-30

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US (2) US7405302B2 (enExample)
EP (1) EP1933842B1 (enExample)
JP (1) JP5327518B2 (enExample)
ES (1) ES2399702T3 (enExample)
WO (1) WO2007047207A2 (enExample)

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JP2013501064A (ja) 2009-08-04 2013-01-10 アミラ ファーマシューティカルス，インコーポレーテッド リゾホスファチジン酸受容体アンタゴニストとしての化合物
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