JP5311673B2 - Ｍｅｋ阻害剤の使用方法 - Google Patents

Ｍｅｋ阻害剤の使用方法 Download PDF

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Publication number
JP5311673B2
JP5311673B2 JP2009541420A JP2009541420A JP5311673B2 JP 5311673 B2 JP5311673 B2 JP 5311673B2 JP 2009541420 A JP2009541420 A JP 2009541420A JP 2009541420 A JP2009541420 A JP 2009541420A JP 5311673 B2 JP5311673 B2 JP 5311673B2
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alkyl
optionally substituted
formula
optionally
amino
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JP2010513288A (ja
JP2010513288A5 (enExample
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ピーター ランブ，
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エグゼリクシス， インコーポレイテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2009541420A 2006-12-14 2007-12-14 Ｍｅｋ阻害剤の使用方法 Expired - Fee Related JP5311673B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US87541206P 2006-12-14 2006-12-14
US60/875,412 2006-12-14
PCT/US2007/025751 WO2008076415A1 (en) 2006-12-14 2007-12-14 Methods of using mek inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013102016A Division JP2013151569A (ja) 2006-12-14 2013-05-14 Ｍｅｋ阻害剤の使用方法

Publications (3)

Publication Number Publication Date
JP2010513288A JP2010513288A (ja) 2010-04-30
JP2010513288A5 JP2010513288A5 (enExample) 2011-04-28
JP5311673B2 true JP5311673B2 (ja) 2013-10-09

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JP2009541420A Expired - Fee Related JP5311673B2 (ja) 2006-12-14 2007-12-14 Ｍｅｋ阻害剤の使用方法
JP2013102016A Pending JP2013151569A (ja) 2006-12-14 2013-05-14 Ｍｅｋ阻害剤の使用方法

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JP2013102016A Pending JP2013151569A (ja) 2006-12-14 2013-05-14 Ｍｅｋ阻害剤の使用方法

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US (1) US7999006B2 (enExample)
EP (1) EP2101759B1 (enExample)
JP (2) JP5311673B2 (enExample)
CN (3) CN105106199A (enExample)
AU (1) AU2007334402B2 (enExample)
CA (1) CA2671982C (enExample)
ES (1) ES2703723T3 (enExample)
HK (1) HK1218256A1 (enExample)
PL (1) PL2101759T3 (enExample)
TR (1) TR201900306T4 (enExample)
WO (1) WO2008076415A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020045535A1 (ja) * 2018-09-01 2020-03-05 富士フイルム株式会社 感活性光線性又は感放射線性樹脂組成物、感活性光線性又は感放射線性膜、パターン形成方法、フォトマスク、電子デバイスの製造方法、及び化合物

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US20080166359A1 (en) 2008-07-10
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