JP5144865B2 - ホスフィニト−オキサゾリン及び金属錯体 - Google Patents

ホスフィニト−オキサゾリン及び金属錯体 Download PDF

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Publication number
JP5144865B2
JP5144865B2 JP2001289902A JP2001289902A JP5144865B2 JP 5144865 B2 JP5144865 B2 JP 5144865B2 JP 2001289902 A JP2001289902 A JP 2001289902A JP 2001289902 A JP2001289902 A JP 2001289902A JP 5144865 B2 JP5144865 B2 JP 5144865B2
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formula
compound
alkyl
group
synthesis
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JP2001289902A
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Japanese (ja)
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JP2002187895A (ja
JP2002187895A5 (enExample
Inventor
プファルツ アンドレアス
エル ブランケンシュタイン イェルク
メンゲス フレデリック
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Solvias AG
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Solvias AG
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/10—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D263/14—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0033—Iridium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/653—Five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2001289902A 2000-09-21 2001-09-21 ホスフィニト−オキサゾリン及び金属錯体 Expired - Fee Related JP5144865B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH18332000 2000-09-21
CH20011177/01 2001-06-26
CH11772001 2001-06-26
CH20001833/00 2001-06-26

Publications (3)

Publication Number Publication Date
JP2002187895A JP2002187895A (ja) 2002-07-05
JP2002187895A5 JP2002187895A5 (enExample) 2008-09-18
JP5144865B2 true JP5144865B2 (ja) 2013-02-13

Family

ID=25738943

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001289902A Expired - Fee Related JP5144865B2 (ja) 2000-09-21 2001-09-21 ホスフィニト−オキサゾリン及び金属錯体

Country Status (7)

Country Link
US (2) US6498256B2 (enExample)
EP (1) EP1191030B1 (enExample)
JP (1) JP5144865B2 (enExample)
AT (1) ATE294806T1 (enExample)
DE (1) DE60110516T2 (enExample)
ES (1) ES2240297T3 (enExample)
PT (1) PT1191030E (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1748767B1 (en) 2004-05-28 2011-12-28 Unigen, Inc. 1-(3-methyl-2,4-dimethoxyphenyl)-3-(2',4'-dihydroxyphenyl)-propane as a potent tyrosinase inhibitor
ES2371653T3 (es) * 2004-12-22 2012-01-05 Dsm Ip Assets B.V. Hidrogenación asimétrica de alquenos usando complejos de iridio quirales.
US7528267B2 (en) 2005-08-01 2009-05-05 Girindus America, Inc. Method for enantioselective hydrogenation of chromenes
CN101565366B (zh) * 2008-04-25 2013-04-17 浙江九洲药业股份有限公司 铱络合物在不饱和羧酸不对称催化氢化中的应用
AU2009274158C1 (en) 2008-07-21 2019-09-05 Unigen, Inc. Series of skin-whitening (lightening) compounds
KR20130106374A (ko) 2010-08-23 2013-09-27 노파르티스 아게 Ｎｅｐ 억제제의 제조에 유용한 중간체의 신규한 제조 방법
US8586799B2 (en) 2011-03-24 2013-11-19 Unigen, Inc. Compounds and methods for preparation of diarylpropanes
CN102731572B (zh) * 2011-04-08 2015-08-05 中国科学院上海有机化学研究所 含全氟烷基的膦配体、其制备方法、应用以及金属络合物
BR112016021171B8 (pt) * 2014-03-18 2021-02-09 Sumitomo Chemical Co processo para fabricação de composto oticamente ativo
EP3350148A1 (en) * 2015-09-17 2018-07-25 DSM IP Assets B.V. Production of farnesol
CN116715699B (zh) * 2023-02-07 2025-08-08 无锡学院 噁唑啉型手性n,p配体及其制备方法和应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4243030A1 (de) * 1992-12-18 1994-06-23 Basf Ag Iminverbindungen
TW424089B (en) * 1996-01-16 2001-03-01 Du Pont Oxazoline arthropodicides
EP0989135B1 (en) * 1996-11-29 2003-03-05 Daiichi Fine Chemical Co., Ltd. Novel phosphinopyrrolidine compounds and process for producing the same
GB9905418D0 (en) * 1999-03-09 1999-05-05 Glaxo Group Ltd Process
GB9907895D0 (en) * 1999-04-08 1999-06-02 Texas A & M Univ Sys Novel ligands for chiral catalysis

Also Published As

Publication number Publication date
EP1191030B1 (en) 2005-05-04
DE60110516T2 (de) 2005-10-13
ATE294806T1 (de) 2005-05-15
PT1191030E (pt) 2005-09-30
EP1191030A2 (en) 2002-03-27
ES2240297T3 (es) 2005-10-16
US6498256B2 (en) 2002-12-24
US20020128486A1 (en) 2002-09-12
JP2002187895A (ja) 2002-07-05
DE60110516D1 (de) 2005-06-09
EP1191030A3 (en) 2002-07-17
US20020062027A1 (en) 2002-05-23
US6632954B2 (en) 2003-10-14

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